Index by author
December 01, 2017; Volume 363,Issue 3
A
Abdullah, Rehab A.
- You have accessInvestigation of Diacylglycerol Lipase Alpha Inhibition in the Mouse Lipopolysaccharide Inflammatory Pain ModelJenny L. Wilkerson, Giulia Donvito, Travis W. Grim, Rehab A. Abdullah, Daisuke Ogasawara, Benjamin F. Cravatt and Aron H. LichtmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 394-401; DOI: https://doi.org/10.1124/jpet.117.243808
Adams, David F.
- You have accessDiscovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor–Prolyl Hydroxylase Inhibitor for AnemiaJennifer L. Ariazi, Kevin J. Duffy, David F. Adams, Duke M. Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-MillerJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 336-347; DOI: https://doi.org/10.1124/jpet.117.242503
Aher, Jayant
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Alapafuja, Shakiru O.
- You have accessCannabinoid CB1 Discrimination: Effects of Endocannabinoids and Catabolic Enzyme InhibitorsMichael Z. Leonard, Shakiru O. Alapafuja, Lipin Ji, Vidyanand G. Shukla, Yingpeng Liu, Spyros P. Nikas, Alexandros Makriyannis, Jack Bergman and Brian D. KangasJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 314-323; DOI: https://doi.org/10.1124/jpet.117.244392
Albright, Charlie F.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Ariazi, Jennifer L.
- You have accessDiscovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor–Prolyl Hydroxylase Inhibitor for AnemiaJennifer L. Ariazi, Kevin J. Duffy, David F. Adams, Duke M. Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-MillerJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 336-347; DOI: https://doi.org/10.1124/jpet.117.242503
B
Bastia, Tanmaya
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Bendayan, Reina
- You have accessXenobiotic Nuclear Receptors Pregnane X Receptor and Constitutive Androstane Receptor Regulate Antiretroviral Drug Efflux Transporters at the Blood-Testis BarrierSana-Kay Whyte-Allman, Md Tozammel Hoque, Mohammad-Ali Jenabian, Jean-Pierre Routy and Reina BendayanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 324-335; DOI: https://doi.org/10.1124/jpet.117.243584
Bergman, Jack
- You have accessCannabinoid CB1 Discrimination: Effects of Endocannabinoids and Catabolic Enzyme InhibitorsMichael Z. Leonard, Shakiru O. Alapafuja, Lipin Ji, Vidyanand G. Shukla, Yingpeng Liu, Spyros P. Nikas, Alexandros Makriyannis, Jack Bergman and Brian D. KangasJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 314-323; DOI: https://doi.org/10.1124/jpet.117.244392
Biernat, Marzena C.
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Biju, Mangatt
- You have accessDiscovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor–Prolyl Hydroxylase Inhibitor for AnemiaJennifer L. Ariazi, Kevin J. Duffy, David F. Adams, Duke M. Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-MillerJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 336-347; DOI: https://doi.org/10.1124/jpet.117.242503
Bookbinder, Mark
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Bristow, Linda J.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Bronson, Joanne J.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Brown, Jeffrey M.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
C
Chamorro, Pablo Aníbal Ferreira
- You have accessTreatment with Sulforaphane Produces Antinociception and Improves Morphine Effects during Inflammatory Pain in MiceAlejandro Redondo, Pablo Aníbal Ferreira Chamorro, Gabriela Riego, Sergi Leánez and Olga PolJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 293-302; DOI: https://doi.org/10.1124/jpet.117.244376
Chapman, Richard W.
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Chen, Kuan-Ju
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Choksi, Riya
- You have accessActivation of Focal Adhesion Kinase and Src Mediates Acquired Sorafenib Resistance in A549 Human Lung Adenocarcinoma XenograftsQingyu Zhou, Xiaofang Guo and Riya ChoksiJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 428-443; DOI: https://doi.org/10.1124/jpet.117.240507
Collier, Justin B.
- You have accessExtracellular Signal–Regulated Kinase 1/2 Regulates Mouse Kidney Injury Molecule-1 Expression Physiologically and Following Ischemic and Septic Renal InjuryJustin B. Collier and Rick G. SchnellmannJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 419-427; DOI: https://doi.org/10.1124/jpet.117.244152
Corboz, Michel R.
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Cravatt, Benjamin F.
- You have accessInvestigation of Diacylglycerol Lipase Alpha Inhibition in the Mouse Lipopolysaccharide Inflammatory Pain ModelJenny L. Wilkerson, Giulia Donvito, Travis W. Grim, Rehab A. Abdullah, Daisuke Ogasawara, Benjamin F. Cravatt and Aron H. LichtmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 394-401; DOI: https://doi.org/10.1124/jpet.117.243808
Curran, Aidan
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
D
DiFilippo, Erin Hugger
- You have accessDiscovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor–Prolyl Hydroxylase Inhibitor for AnemiaJennifer L. Ariazi, Kevin J. Duffy, David F. Adams, Duke M. Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-MillerJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 336-347; DOI: https://doi.org/10.1124/jpet.117.242503
Doi, Takefumi
- You have accessCreation of a Claudin-2 Binder and Its Tight Junction–Modulating Activity in a Human Intestinal ModelMutsumi Takigawa, Manami Iida, Shotaro Nagase, Hidehiko Suzuki, Akihiro Watari, Minoru Tada, Yoshiaki Okada, Takefumi Doi, Masayoshi Fukasawa, Kiyohito Yagi, Jun Kunisawa and Masuo KondohJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 444-451; DOI: https://doi.org/10.1124/jpet.117.242214
Donvito, Giulia
- You have accessInvestigation of Diacylglycerol Lipase Alpha Inhibition in the Mouse Lipopolysaccharide Inflammatory Pain ModelJenny L. Wilkerson, Giulia Donvito, Travis W. Grim, Rehab A. Abdullah, Daisuke Ogasawara, Benjamin F. Cravatt and Aron H. LichtmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 394-401; DOI: https://doi.org/10.1124/jpet.117.243808
Duffy, Kevin J.
- You have accessDiscovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor–Prolyl Hydroxylase Inhibitor for AnemiaJennifer L. Ariazi, Kevin J. Duffy, David F. Adams, Duke M. Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-MillerJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 336-347; DOI: https://doi.org/10.1124/jpet.117.242503
E
Erickson-Miller, Connie
- You have accessDiscovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor–Prolyl Hydroxylase Inhibitor for AnemiaJennifer L. Ariazi, Kevin J. Duffy, David F. Adams, Duke M. Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-MillerJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 336-347; DOI: https://doi.org/10.1124/jpet.117.242503
F
Falck, John R.
- You have accessThe Blood Pressure–Lowering Effect of 20-HETE Blockade in Cyp4a14(−/−) Mice Is Associated with NatriuresisVarunkumar Pandey, Victor Garcia, Ankit Gilani, Priyanka Mishra, Frank Fan Zhang, Mahesh P. Paudyal, John R. Falck, Alberto Nasjletti, Wen-Hui Wang and Michal Laniado SchwartzmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 412-418; DOI: https://doi.org/10.1124/jpet.117.243618
Fernandes, Alda
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Fitch, Duke M.
- You have accessDiscovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor–Prolyl Hydroxylase Inhibitor for AnemiaJennifer L. Ariazi, Kevin J. Duffy, David F. Adams, Duke M. Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-MillerJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 336-347; DOI: https://doi.org/10.1124/jpet.117.242503
Fujio, Yasushi
- You have accessSustained Activation of Guanylate Cyclase-A with TDT, a Natriuretic Peptide Derivative, Exhibits Cardiorenal Protection in Dahl Salt-Sensitive Hypertensive RatsShohei Oishi, Naoko Suzuki, Yuri Hasui, Tsuyoshi Homma, Masanori Obana, Takahiro Nagayama and Yasushi FujioJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 402-410; DOI: https://doi.org/10.1124/jpet.117.244459
Fukasawa, Masayoshi
- You have accessCreation of a Claudin-2 Binder and Its Tight Junction–Modulating Activity in a Human Intestinal ModelMutsumi Takigawa, Manami Iida, Shotaro Nagase, Hidehiko Suzuki, Akihiro Watari, Minoru Tada, Yoshiaki Okada, Takefumi Doi, Masayoshi Fukasawa, Kiyohito Yagi, Jun Kunisawa and Masuo KondohJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 444-451; DOI: https://doi.org/10.1124/jpet.117.242214
G
Garcia, Victor
- You have accessThe Blood Pressure–Lowering Effect of 20-HETE Blockade in Cyp4a14(−/−) Mice Is Associated with NatriuresisVarunkumar Pandey, Victor Garcia, Ankit Gilani, Priyanka Mishra, Frank Fan Zhang, Mahesh P. Paudyal, John R. Falck, Alberto Nasjletti, Wen-Hui Wang and Michal Laniado SchwartzmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 412-418; DOI: https://doi.org/10.1124/jpet.117.243618
Gilani, Ankit
- You have accessThe Blood Pressure–Lowering Effect of 20-HETE Blockade in Cyp4a14(−/−) Mice Is Associated with NatriuresisVarunkumar Pandey, Victor Garcia, Ankit Gilani, Priyanka Mishra, Frank Fan Zhang, Mahesh P. Paudyal, John R. Falck, Alberto Nasjletti, Wen-Hui Wang and Michal Laniado SchwartzmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 412-418; DOI: https://doi.org/10.1124/jpet.117.243618
Graef, John D.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Granneman, James G.
- You have accessNovel Pharmacological Probes Reveal ABHD5 as a Locus of Lipolysis Control in White and Brown AdipocytesElizabeth A. Rondini, Ljiljana Mladenovic-Lucas, William R. Roush, Geoff T. Halvorsen, Alex E. Green and James G. GrannemanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 367-376; DOI: https://doi.org/10.1124/jpet.117.243253
Green, Alex E.
- You have accessNovel Pharmacological Probes Reveal ABHD5 as a Locus of Lipolysis Control in White and Brown AdipocytesElizabeth A. Rondini, Ljiljana Mladenovic-Lucas, William R. Roush, Geoff T. Halvorsen, Alex E. Green and James G. GrannemanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 367-376; DOI: https://doi.org/10.1124/jpet.117.243253
Grim, Travis W.
- You have accessInvestigation of Diacylglycerol Lipase Alpha Inhibition in the Mouse Lipopolysaccharide Inflammatory Pain ModelJenny L. Wilkerson, Giulia Donvito, Travis W. Grim, Rehab A. Abdullah, Daisuke Ogasawara, Benjamin F. Cravatt and Aron H. LichtmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 394-401; DOI: https://doi.org/10.1124/jpet.117.243808
Gulia, Jyoti
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Guo, Xiaofang
- You have accessActivation of Focal Adhesion Kinase and Src Mediates Acquired Sorafenib Resistance in A549 Human Lung Adenocarcinoma XenograftsQingyu Zhou, Xiaofang Guo and Riya ChoksiJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 428-443; DOI: https://doi.org/10.1124/jpet.117.240507
H
Halvorsen, Geoff T.
- You have accessNovel Pharmacological Probes Reveal ABHD5 as a Locus of Lipolysis Control in White and Brown AdipocytesElizabeth A. Rondini, Ljiljana Mladenovic-Lucas, William R. Roush, Geoff T. Halvorsen, Alex E. Green and James G. GrannemanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 367-376; DOI: https://doi.org/10.1124/jpet.117.243253
Hasui, Yuri
- You have accessSustained Activation of Guanylate Cyclase-A with TDT, a Natriuretic Peptide Derivative, Exhibits Cardiorenal Protection in Dahl Salt-Sensitive Hypertensive RatsShohei Oishi, Naoko Suzuki, Yuri Hasui, Tsuyoshi Homma, Masanori Obana, Takahiro Nagayama and Yasushi FujioJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 402-410; DOI: https://doi.org/10.1124/jpet.117.244459
Homma, Tsuyoshi
- You have accessSustained Activation of Guanylate Cyclase-A with TDT, a Natriuretic Peptide Derivative, Exhibits Cardiorenal Protection in Dahl Salt-Sensitive Hypertensive RatsShohei Oishi, Naoko Suzuki, Yuri Hasui, Tsuyoshi Homma, Masanori Obana, Takahiro Nagayama and Yasushi FujioJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 402-410; DOI: https://doi.org/10.1124/jpet.117.244459
Hoque, Md Tozammel
- You have accessXenobiotic Nuclear Receptors Pregnane X Receptor and Constitutive Androstane Receptor Regulate Antiretroviral Drug Efflux Transporters at the Blood-Testis BarrierSana-Kay Whyte-Allman, Md Tozammel Hoque, Mohammad-Ali Jenabian, Jean-Pierre Routy and Reina BendayanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 324-335; DOI: https://doi.org/10.1124/jpet.117.243584
I
Iida, Manami
- You have accessCreation of a Claudin-2 Binder and Its Tight Junction–Modulating Activity in a Human Intestinal ModelMutsumi Takigawa, Manami Iida, Shotaro Nagase, Hidehiko Suzuki, Akihiro Watari, Minoru Tada, Yoshiaki Okada, Takefumi Doi, Masayoshi Fukasawa, Kiyohito Yagi, Jun Kunisawa and Masuo KondohJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 444-451; DOI: https://doi.org/10.1124/jpet.117.242214
Islam, Imadul
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
J
Jackson, Edwin K.
- You have access8-Aminoguanosine Exerts Diuretic, Natriuretic, and Glucosuric Activity via Conversion to 8-Aminoguanine, Yet Has Direct Antikaliuretic EffectsEdwin K. Jackson and Zaichuan MiJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 358-366; DOI: https://doi.org/10.1124/jpet.117.243758
Jenabian, Mohammad-Ali
- You have accessXenobiotic Nuclear Receptors Pregnane X Receptor and Constitutive Androstane Receptor Regulate Antiretroviral Drug Efflux Transporters at the Blood-Testis BarrierSana-Kay Whyte-Allman, Md Tozammel Hoque, Mohammad-Ali Jenabian, Jean-Pierre Routy and Reina BendayanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 324-335; DOI: https://doi.org/10.1124/jpet.117.243584
Ji, Lipin
- You have accessCannabinoid CB1 Discrimination: Effects of Endocannabinoids and Catabolic Enzyme InhibitorsMichael Z. Leonard, Shakiru O. Alapafuja, Lipin Ji, Vidyanand G. Shukla, Yingpeng Liu, Spyros P. Nikas, Alexandros Makriyannis, Jack Bergman and Brian D. KangasJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 314-323; DOI: https://doi.org/10.1124/jpet.117.244392
K
Kalidindi, Narasimharaju
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Kallem, Raja Reddy
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Kangas, Brian D.
- You have accessCannabinoid CB1 Discrimination: Effects of Endocannabinoids and Catabolic Enzyme InhibitorsMichael Z. Leonard, Shakiru O. Alapafuja, Lipin Ji, Vidyanand G. Shukla, Yingpeng Liu, Spyros P. Nikas, Alexandros Makriyannis, Jack Bergman and Brian D. KangasJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 314-323; DOI: https://doi.org/10.1124/jpet.117.244392
Keavy, Deborah
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Kempson, James
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
King, Dalton
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Kondoh, Masuo
- You have accessCreation of a Claudin-2 Binder and Its Tight Junction–Modulating Activity in a Human Intestinal ModelMutsumi Takigawa, Manami Iida, Shotaro Nagase, Hidehiko Suzuki, Akihiro Watari, Minoru Tada, Yoshiaki Okada, Takefumi Doi, Masayoshi Fukasawa, Kiyohito Yagi, Jun Kunisawa and Masuo KondohJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 444-451; DOI: https://doi.org/10.1124/jpet.117.242214
Konicek, Donna M.
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Kumar, Kuchibhotla Vijaya
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Kunisawa, Jun
- You have accessCreation of a Claudin-2 Binder and Its Tight Junction–Modulating Activity in a Human Intestinal ModelMutsumi Takigawa, Manami Iida, Shotaro Nagase, Hidehiko Suzuki, Akihiro Watari, Minoru Tada, Yoshiaki Okada, Takefumi Doi, Masayoshi Fukasawa, Kiyohito Yagi, Jun Kunisawa and Masuo KondohJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 444-451; DOI: https://doi.org/10.1124/jpet.117.242214
L
Laurent, Charles E.
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Leánez, Sergi
- You have accessTreatment with Sulforaphane Produces Antinociception and Improves Morphine Effects during Inflammatory Pain in MiceAlejandro Redondo, Pablo Aníbal Ferreira Chamorro, Gabriela Riego, Sergi Leánez and Olga PolJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 293-302; DOI: https://doi.org/10.1124/jpet.117.244376
Leifer, Franziska G.
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Leonard, Michael Z.
- You have accessCannabinoid CB1 Discrimination: Effects of Endocannabinoids and Catabolic Enzyme InhibitorsMichael Z. Leonard, Shakiru O. Alapafuja, Lipin Ji, Vidyanand G. Shukla, Yingpeng Liu, Spyros P. Nikas, Alexandros Makriyannis, Jack Bergman and Brian D. KangasJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 314-323; DOI: https://doi.org/10.1124/jpet.117.244392
Li, Jianqing
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Li, Yu-Wen
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Li, Zhili
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Lichtman, Aron H.
- You have accessInvestigation of Diacylglycerol Lipase Alpha Inhibition in the Mouse Lipopolysaccharide Inflammatory Pain ModelJenny L. Wilkerson, Giulia Donvito, Travis W. Grim, Rehab A. Abdullah, Daisuke Ogasawara, Benjamin F. Cravatt and Aron H. LichtmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 394-401; DOI: https://doi.org/10.1124/jpet.117.243808
Liu, Yingpeng
- You have accessCannabinoid CB1 Discrimination: Effects of Endocannabinoids and Catabolic Enzyme InhibitorsMichael Z. Leonard, Shakiru O. Alapafuja, Lipin Ji, Vidyanand G. Shukla, Yingpeng Liu, Spyros P. Nikas, Alexandros Makriyannis, Jack Bergman and Brian D. KangasJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 314-323; DOI: https://doi.org/10.1124/jpet.117.244392
Luo, Lusong
- You have accessDiscovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor–Prolyl Hydroxylase Inhibitor for AnemiaJennifer L. Ariazi, Kevin J. Duffy, David F. Adams, Duke M. Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-MillerJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 336-347; DOI: https://doi.org/10.1124/jpet.117.242503
M
Macor, John E.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Makriyannis, Alexandros
- You have accessCannabinoid CB1 Discrimination: Effects of Endocannabinoids and Catabolic Enzyme InhibitorsMichael Z. Leonard, Shakiru O. Alapafuja, Lipin Ji, Vidyanand G. Shukla, Yingpeng Liu, Spyros P. Nikas, Alexandros Makriyannis, Jack Bergman and Brian D. KangasJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 314-323; DOI: https://doi.org/10.1124/jpet.117.244392
Malinin, Vladimir
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Marcin, Lawrence R.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Mathur, Arvind
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Mi, Zaichuan
- You have access8-Aminoguanosine Exerts Diuretic, Natriuretic, and Glucosuric Activity via Conversion to 8-Aminoguanine, Yet Has Direct Antikaliuretic EffectsEdwin K. Jackson and Zaichuan MiJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 358-366; DOI: https://doi.org/10.1124/jpet.117.243758
Mishra, Priyanka
- You have accessThe Blood Pressure–Lowering Effect of 20-HETE Blockade in Cyp4a14(−/−) Mice Is Associated with NatriuresisVarunkumar Pandey, Victor Garcia, Ankit Gilani, Priyanka Mishra, Frank Fan Zhang, Mahesh P. Paudyal, John R. Falck, Alberto Nasjletti, Wen-Hui Wang and Michal Laniado SchwartzmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 412-418; DOI: https://doi.org/10.1124/jpet.117.243618
Mladenovic-Lucas, Ljiljana
- You have accessNovel Pharmacological Probes Reveal ABHD5 as a Locus of Lipolysis Control in White and Brown AdipocytesElizabeth A. Rondini, Ljiljana Mladenovic-Lucas, William R. Roush, Geoff T. Halvorsen, Alex E. Green and James G. GrannemanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 367-376; DOI: https://doi.org/10.1124/jpet.117.243253
Molski, Thaddeus
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
N
Nagase, Shotaro
- You have accessCreation of a Claudin-2 Binder and Its Tight Junction–Modulating Activity in a Human Intestinal ModelMutsumi Takigawa, Manami Iida, Shotaro Nagase, Hidehiko Suzuki, Akihiro Watari, Minoru Tada, Yoshiaki Okada, Takefumi Doi, Masayoshi Fukasawa, Kiyohito Yagi, Jun Kunisawa and Masuo KondohJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 444-451; DOI: https://doi.org/10.1124/jpet.117.242214
Nagayama, Takahiro
- You have accessSustained Activation of Guanylate Cyclase-A with TDT, a Natriuretic Peptide Derivative, Exhibits Cardiorenal Protection in Dahl Salt-Sensitive Hypertensive RatsShohei Oishi, Naoko Suzuki, Yuri Hasui, Tsuyoshi Homma, Masanori Obana, Takahiro Nagayama and Yasushi FujioJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 402-410; DOI: https://doi.org/10.1124/jpet.117.244459
Naidu, Pattipati S.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Nasjletti, Alberto
- You have accessThe Blood Pressure–Lowering Effect of 20-HETE Blockade in Cyp4a14(−/−) Mice Is Associated with NatriuresisVarunkumar Pandey, Victor Garcia, Ankit Gilani, Priyanka Mishra, Frank Fan Zhang, Mahesh P. Paudyal, John R. Falck, Alberto Nasjletti, Wen-Hui Wang and Michal Laniado SchwartzmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 412-418; DOI: https://doi.org/10.1124/jpet.117.243618
Newberry, Kimberly
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Newton, Amy
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Nikas, Spyros P.
- You have accessCannabinoid CB1 Discrimination: Effects of Endocannabinoids and Catabolic Enzyme InhibitorsMichael Z. Leonard, Shakiru O. Alapafuja, Lipin Ji, Vidyanand G. Shukla, Yingpeng Liu, Spyros P. Nikas, Alexandros Makriyannis, Jack Bergman and Brian D. KangasJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 314-323; DOI: https://doi.org/10.1124/jpet.117.244392
O
Obana, Masanori
- You have accessSustained Activation of Guanylate Cyclase-A with TDT, a Natriuretic Peptide Derivative, Exhibits Cardiorenal Protection in Dahl Salt-Sensitive Hypertensive RatsShohei Oishi, Naoko Suzuki, Yuri Hasui, Tsuyoshi Homma, Masanori Obana, Takahiro Nagayama and Yasushi FujioJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 402-410; DOI: https://doi.org/10.1124/jpet.117.244459
Ogasawara, Daisuke
- You have accessInvestigation of Diacylglycerol Lipase Alpha Inhibition in the Mouse Lipopolysaccharide Inflammatory Pain ModelJenny L. Wilkerson, Giulia Donvito, Travis W. Grim, Rehab A. Abdullah, Daisuke Ogasawara, Benjamin F. Cravatt and Aron H. LichtmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 394-401; DOI: https://doi.org/10.1124/jpet.117.243808
Oishi, Shohei
- You have accessSustained Activation of Guanylate Cyclase-A with TDT, a Natriuretic Peptide Derivative, Exhibits Cardiorenal Protection in Dahl Salt-Sensitive Hypertensive RatsShohei Oishi, Naoko Suzuki, Yuri Hasui, Tsuyoshi Homma, Masanori Obana, Takahiro Nagayama and Yasushi FujioJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 402-410; DOI: https://doi.org/10.1124/jpet.117.244459
Okada, Yoshiaki
- You have accessCreation of a Claudin-2 Binder and Its Tight Junction–Modulating Activity in a Human Intestinal ModelMutsumi Takigawa, Manami Iida, Shotaro Nagase, Hidehiko Suzuki, Akihiro Watari, Minoru Tada, Yoshiaki Okada, Takefumi Doi, Masayoshi Fukasawa, Kiyohito Yagi, Jun Kunisawa and Masuo KondohJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 444-451; DOI: https://doi.org/10.1124/jpet.117.242214
Olson, Richard E.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
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Pandey, Varunkumar
- You have accessThe Blood Pressure–Lowering Effect of 20-HETE Blockade in Cyp4a14(−/−) Mice Is Associated with NatriuresisVarunkumar Pandey, Victor Garcia, Ankit Gilani, Priyanka Mishra, Frank Fan Zhang, Mahesh P. Paudyal, John R. Falck, Alberto Nasjletti, Wen-Hui Wang and Michal Laniado SchwartzmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 412-418; DOI: https://doi.org/10.1124/jpet.117.243618
Pappalardi, Melissa
- You have accessDiscovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor–Prolyl Hydroxylase Inhibitor for AnemiaJennifer L. Ariazi, Kevin J. Duffy, David F. Adams, Duke M. Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-MillerJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 336-347; DOI: https://doi.org/10.1124/jpet.117.242503
Paschapur, Mahesh
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Paudyal, Mahesh P.
- You have accessThe Blood Pressure–Lowering Effect of 20-HETE Blockade in Cyp4a14(−/−) Mice Is Associated with NatriuresisVarunkumar Pandey, Victor Garcia, Ankit Gilani, Priyanka Mishra, Frank Fan Zhang, Mahesh P. Paudyal, John R. Falck, Alberto Nasjletti, Wen-Hui Wang and Michal Laniado SchwartzmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 412-418; DOI: https://doi.org/10.1124/jpet.117.243618
Perkins, Walter R.
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Pieschl, Rick
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Plaunt, Adam J.
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Pol, Olga
- You have accessTreatment with Sulforaphane Produces Antinociception and Improves Morphine Effects during Inflammatory Pain in MiceAlejandro Redondo, Pablo Aníbal Ferreira Chamorro, Gabriela Riego, Sergi Leánez and Olga PolJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 293-302; DOI: https://doi.org/10.1124/jpet.117.244376
Polino, Joseph
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
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Ramarao, Manjunath
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Redondo, Alejandro
- You have accessTreatment with Sulforaphane Produces Antinociception and Improves Morphine Effects during Inflammatory Pain in MiceAlejandro Redondo, Pablo Aníbal Ferreira Chamorro, Gabriela Riego, Sergi Leánez and Olga PolJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 293-302; DOI: https://doi.org/10.1124/jpet.117.244376
Riego, Gabriela
- You have accessTreatment with Sulforaphane Produces Antinociception and Improves Morphine Effects during Inflammatory Pain in MiceAlejandro Redondo, Pablo Aníbal Ferreira Chamorro, Gabriela Riego, Sergi Leánez and Olga PolJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 293-302; DOI: https://doi.org/10.1124/jpet.117.244376
Rondini, Elizabeth A.
- You have accessNovel Pharmacological Probes Reveal ABHD5 as a Locus of Lipolysis Control in White and Brown AdipocytesElizabeth A. Rondini, Ljiljana Mladenovic-Lucas, William R. Roush, Geoff T. Halvorsen, Alex E. Green and James G. GrannemanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 367-376; DOI: https://doi.org/10.1124/jpet.117.243253
Roush, William R.
- You have accessNovel Pharmacological Probes Reveal ABHD5 as a Locus of Lipolysis Control in White and Brown AdipocytesElizabeth A. Rondini, Ljiljana Mladenovic-Lucas, William R. Roush, Geoff T. Halvorsen, Alex E. Green and James G. GrannemanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 367-376; DOI: https://doi.org/10.1124/jpet.117.243253
Routy, Jean-Pierre
- You have accessXenobiotic Nuclear Receptors Pregnane X Receptor and Constitutive Androstane Receptor Regulate Antiretroviral Drug Efflux Transporters at the Blood-Testis BarrierSana-Kay Whyte-Allman, Md Tozammel Hoque, Mohammad-Ali Jenabian, Jean-Pierre Routy and Reina BendayanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 324-335; DOI: https://doi.org/10.1124/jpet.117.243584
S
Salvail, Dany
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Sanmathi, Charulatha
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Schnellmann, Rick G.
- You have accessMitochondrial-Based Therapeutics for the Treatment of Spinal Cord Injury: Mitochondrial Biogenesis as a Potential Pharmacological TargetNatalie E. Scholpa and Rick G. SchnellmannJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 303-313; DOI: https://doi.org/10.1124/jpet.117.244806
- You have accessExtracellular Signal–Regulated Kinase 1/2 Regulates Mouse Kidney Injury Molecule-1 Expression Physiologically and Following Ischemic and Septic Renal InjuryJustin B. Collier and Rick G. SchnellmannJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 419-427; DOI: https://doi.org/10.1124/jpet.117.244152
Scholpa, Natalie E.
- You have accessMitochondrial-Based Therapeutics for the Treatment of Spinal Cord Injury: Mitochondrial Biogenesis as a Potential Pharmacological TargetNatalie E. Scholpa and Rick G. SchnellmannJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 303-313; DOI: https://doi.org/10.1124/jpet.117.244806
Schwartzman, Michal Laniado
- You have accessThe Blood Pressure–Lowering Effect of 20-HETE Blockade in Cyp4a14(−/−) Mice Is Associated with NatriuresisVarunkumar Pandey, Victor Garcia, Ankit Gilani, Priyanka Mishra, Frank Fan Zhang, Mahesh P. Paudyal, John R. Falck, Alberto Nasjletti, Wen-Hui Wang and Michal Laniado SchwartzmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 412-418; DOI: https://doi.org/10.1124/jpet.117.243618
Shaw, Tony
- You have accessDiscovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor–Prolyl Hydroxylase Inhibitor for AnemiaJennifer L. Ariazi, Kevin J. Duffy, David F. Adams, Duke M. Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-MillerJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 336-347; DOI: https://doi.org/10.1124/jpet.117.242503
Shields, Eric
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Shukla, Vidyanand G.
- You have accessCannabinoid CB1 Discrimination: Effects of Endocannabinoids and Catabolic Enzyme InhibitorsMichael Z. Leonard, Shakiru O. Alapafuja, Lipin Ji, Vidyanand G. Shukla, Yingpeng Liu, Spyros P. Nikas, Alexandros Makriyannis, Jack Bergman and Brian D. KangasJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 314-323; DOI: https://doi.org/10.1124/jpet.117.244392
Simmermacher, Jean
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Sinha, Meenakshee
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Sinz, Michael
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Sivarao, Digavalli V.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Srikumar, Bettadapura N.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Suzuki, Hidehiko
- You have accessCreation of a Claudin-2 Binder and Its Tight Junction–Modulating Activity in a Human Intestinal ModelMutsumi Takigawa, Manami Iida, Shotaro Nagase, Hidehiko Suzuki, Akihiro Watari, Minoru Tada, Yoshiaki Okada, Takefumi Doi, Masayoshi Fukasawa, Kiyohito Yagi, Jun Kunisawa and Masuo KondohJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 444-451; DOI: https://doi.org/10.1124/jpet.117.242214
Suzuki, Naoko
- You have accessSustained Activation of Guanylate Cyclase-A with TDT, a Natriuretic Peptide Derivative, Exhibits Cardiorenal Protection in Dahl Salt-Sensitive Hypertensive RatsShohei Oishi, Naoko Suzuki, Yuri Hasui, Tsuyoshi Homma, Masanori Obana, Takahiro Nagayama and Yasushi FujioJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 402-410; DOI: https://doi.org/10.1124/jpet.117.244459
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Tada, Minoru
- You have accessCreation of a Claudin-2 Binder and Its Tight Junction–Modulating Activity in a Human Intestinal ModelMutsumi Takigawa, Manami Iida, Shotaro Nagase, Hidehiko Suzuki, Akihiro Watari, Minoru Tada, Yoshiaki Okada, Takefumi Doi, Masayoshi Fukasawa, Kiyohito Yagi, Jun Kunisawa and Masuo KondohJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 444-451; DOI: https://doi.org/10.1124/jpet.117.242214
Takigawa, Mutsumi
- You have accessCreation of a Claudin-2 Binder and Its Tight Junction–Modulating Activity in a Human Intestinal ModelMutsumi Takigawa, Manami Iida, Shotaro Nagase, Hidehiko Suzuki, Akihiro Watari, Minoru Tada, Yoshiaki Okada, Takefumi Doi, Masayoshi Fukasawa, Kiyohito Yagi, Jun Kunisawa and Masuo KondohJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 444-451; DOI: https://doi.org/10.1124/jpet.117.242214
Thangathirupathy, Srinivasan
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Thompson, Lorin A.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
V
Vikramadithyan, Reeba K.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
W
Wang, Wen-Hui
- You have accessThe Blood Pressure–Lowering Effect of 20-HETE Blockade in Cyp4a14(−/−) Mice Is Associated with NatriuresisVarunkumar Pandey, Victor Garcia, Ankit Gilani, Priyanka Mishra, Frank Fan Zhang, Mahesh P. Paudyal, John R. Falck, Alberto Nasjletti, Wen-Hui Wang and Michal Laniado SchwartzmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 412-418; DOI: https://doi.org/10.1124/jpet.117.243618
Warrier, Jayakumar
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Watari, Akihiro
- You have accessCreation of a Claudin-2 Binder and Its Tight Junction–Modulating Activity in a Human Intestinal ModelMutsumi Takigawa, Manami Iida, Shotaro Nagase, Hidehiko Suzuki, Akihiro Watari, Minoru Tada, Yoshiaki Okada, Takefumi Doi, Masayoshi Fukasawa, Kiyohito Yagi, Jun Kunisawa and Masuo KondohJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 444-451; DOI: https://doi.org/10.1124/jpet.117.242214
Weed, Michael R.
- You have accessPreclinical Characterization of (R)-3-((3S,4S)-3-fluoro-4-(4-hydroxyphenyl)piperidin-1-yl)-1-(4-methylbenzyl)pyrrolidin-2-one (BMS-986169), a Novel, Intravenous, Glutamate N-Methyl-d-Aspartate 2B Receptor Negative Allosteric Modulator with Potential in Major Depressive DisorderLinda J. Bristow, Jyoti Gulia, Michael R. Weed, Bettadapura N. Srikumar, Yu-Wen Li, John D. Graef, Pattipati S. Naidu, Charulatha Sanmathi, Jayant Aher, Tanmaya Bastia, Mahesh Paschapur, Narasimharaju Kalidindi, Kuchibhotla Vijaya Kumar, Thaddeus Molski, Rick Pieschl, Alda Fernandes, Jeffrey M. Brown, Digavalli V. Sivarao, Kimberly Newberry, Mark Bookbinder, Joseph Polino, Deborah Keavy, Amy Newton, Eric Shields, Jean Simmermacher, James Kempson, Jianqing Li, Huiping Zhang, Arvind Mathur, Raja Reddy Kallem, Meenakshee Sinha, Manjunath Ramarao, Reeba K. Vikramadithyan, Srinivasan Thangathirupathy, Jayakumar Warrier, Imadul Islam, Joanne J. Bronson, Richard E. Olson, John E. Macor, Charlie F. Albright, Dalton King, Lorin A. Thompson, Lawrence R. Marcin and Michael SinzJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 377-393; DOI: https://doi.org/10.1124/jpet.117.242784
Whyte-Allman, Sana-Kay
- You have accessXenobiotic Nuclear Receptors Pregnane X Receptor and Constitutive Androstane Receptor Regulate Antiretroviral Drug Efflux Transporters at the Blood-Testis BarrierSana-Kay Whyte-Allman, Md Tozammel Hoque, Mohammad-Ali Jenabian, Jean-Pierre Routy and Reina BendayanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 324-335; DOI: https://doi.org/10.1124/jpet.117.243584
Wiggall, Ken
- You have accessDiscovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor–Prolyl Hydroxylase Inhibitor for AnemiaJennifer L. Ariazi, Kevin J. Duffy, David F. Adams, Duke M. Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-MillerJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 336-347; DOI: https://doi.org/10.1124/jpet.117.242503
Wilkerson, Jenny L.
- You have accessInvestigation of Diacylglycerol Lipase Alpha Inhibition in the Mouse Lipopolysaccharide Inflammatory Pain ModelJenny L. Wilkerson, Giulia Donvito, Travis W. Grim, Rehab A. Abdullah, Daisuke Ogasawara, Benjamin F. Cravatt and Aron H. LichtmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 394-401; DOI: https://doi.org/10.1124/jpet.117.243808
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Xu, Fadi
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
Y
Yagi, Kiyohito
- You have accessCreation of a Claudin-2 Binder and Its Tight Junction–Modulating Activity in a Human Intestinal ModelMutsumi Takigawa, Manami Iida, Shotaro Nagase, Hidehiko Suzuki, Akihiro Watari, Minoru Tada, Yoshiaki Okada, Takefumi Doi, Masayoshi Fukasawa, Kiyohito Yagi, Jun Kunisawa and Masuo KondohJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 444-451; DOI: https://doi.org/10.1124/jpet.117.242214
Yin, Han
- Open AccessPreclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator ProdrugMichel R. Corboz, Zhili Li, Vladimir Malinin, Adam J. Plaunt, Donna M. Konicek, Franziska G. Leifer, Kuan-Ju Chen, Charles E. Laurent, Han Yin, Marzena C. Biernat, Dany Salvail, Jianguo Zhuang, Fadi Xu, Aidan Curran, Walter R. Perkins and Richard W. ChapmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 348-357; DOI: https://doi.org/10.1124/jpet.117.242099
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Zhang, Frank Fan
- You have accessThe Blood Pressure–Lowering Effect of 20-HETE Blockade in Cyp4a14(−/−) Mice Is Associated with NatriuresisVarunkumar Pandey, Victor Garcia, Ankit Gilani, Priyanka Mishra, Frank Fan Zhang, Mahesh P. Paudyal, John R. Falck, Alberto Nasjletti, Wen-Hui Wang and Michal Laniado SchwartzmanJournal of Pharmacology and Experimental Therapeutics December 2017, 363 (3) 412-418; DOI: https://doi.org/10.1124/jpet.117.243618
Zhang, Huiping
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