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Research ArticleINFLAMMATION AND IMMUNOPHARMACOLOGY

SSR240612 [(2R)-2-[((3R)-3-(1,3-Benzodioxol-5-yl)-3-{[(6-methoxy-2-naphthyl)sulfonyl]amino}propanoyl)amino]-3-(4-{[2R,6S)-2,6-dimethylpiperidinyl]methyl}phenyl)-N-isopropyl-N-methylpropanamide Hydrochloride], a New Nonpeptide Antagonist of the Bradykinin B1 Receptor: Biochemical and Pharmacological Characterization

Jean Gougat, Bernard Ferrari, Lionel Sarran, Claudine Planchenault, Martine Poncelet, Jeanne Maruani, Richard Alonso, Annie Cudennec, Tiziano Croci, Fabio Guagnini, Katalin Urban-Szabo, Jean-Pierre Martinolle, Philippe Soubrié, Olivier Finance and Gérard Le Fur
Journal of Pharmacology and Experimental Therapeutics May 2004, 309 (2) 661-669; DOI: https://doi.org/10.1124/jpet.103.059527

Article Information

vol. 309 no. 2 661-669
DOI 
https://doi.org/10.1124/jpet.103.059527
PubMed 
14747609
Published By 
American Society for Pharmacology and Experimental Therapeutics
Print ISSN 
0022-3565
Online ISSN 
1521-0103
History 
  • Received September 4, 2003
  • Accepted January 21, 2004
  • Published online April 21, 2004.

Article Versions

Copyright & Usage 
The American Society for Pharmacology and Experimental Therapeutics

Author Information

  1. Jean Gougat,
  2. Bernard Ferrari,
  3. Lionel Sarran,
  4. Claudine Planchenault,
  5. Martine Poncelet,
  6. Jeanne Maruani,
  7. Richard Alonso,
  8. Annie Cudennec,
  9. Tiziano Croci,
  10. Fabio Guagnini,
  11. Katalin Urban-Szabo,
  12. Jean-Pierre Martinolle,
  13. Philippe Soubrié,
  14. Olivier Finance and
  15. Gérard Le Fur
  1. Sanofi-Synthelabo Recherche, Montpellier, France
  1. Address correspondence to:
    Jean Gougat, Sanofi-Synthelabo Recherche, 371 rue du Prof. J. Blayac, Cedex 04, 34184 Montpellier, France. E-mail: jean.gougat{at}sanofi-synthelabo.com
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Research ArticleINFLAMMATION AND IMMUNOPHARMACOLOGY

SSR240612 [(2R)-2-[((3R)-3-(1,3-Benzodioxol-5-yl)-3-{[(6-methoxy-2-naphthyl)sulfonyl]amino}propanoyl)amino]-3-(4-{[2R,6S)-2,6-dimethylpiperidinyl]methyl}phenyl)-N-isopropyl-N-methylpropanamide Hydrochloride], a New Nonpeptide Antagonist of the Bradykinin B1 Receptor: Biochemical and Pharmacological Characterization

Jean Gougat, Bernard Ferrari, Lionel Sarran, Claudine Planchenault, Martine Poncelet, Jeanne Maruani, Richard Alonso, Annie Cudennec, Tiziano Croci, Fabio Guagnini, Katalin Urban-Szabo, Jean-Pierre Martinolle, Philippe Soubrié, Olivier Finance and Gérard Le Fur
Journal of Pharmacology and Experimental Therapeutics May 1, 2004, 309 (2) 661-669; DOI: https://doi.org/10.1124/jpet.103.059527
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