Described herein is a synthetic strategy for the total synthesis of (±)‐phomoidride D. This
highly efficient and stereoselective approach provides rapid assembly of the carbocyclic core …

The treatment of a,| 3-unsaturated esters having a ketone function at an appropriate position
with either TBDMSOTf in the presence of Et3N or TMSI in the presence of (TMS) 2NH …

Brain-derived neurotrophic factor (BDNF) is reported to enhance synaptic transmission and
to play a role in long-term potentiation in hippocampus and neocortex. If so, a shortage or …

The enantioselective construction of a qua-ternary asymmetric carbon center was developed
through reaction of the dianions derived from the chiral half esters of monosubstituted …

A series of compounds structually related to 4'-[(4, 4-difluoro-5-methylidene-2, 3, 4, 5-tetrahydro-1H-1-benzoazepin-1-yl)
carbonyl]-2-phenylbenzanilide were synthesized and evaluated …

A series of compounds structurally related to 2-phenyl-4’-(2, 3, 4, 5—tetrahydro-lH-l, 5-benzodiazepine—l-carbonyl)
benzanilide was synthesized and demonstrated to have arginine …

Solutions of 4 are stable for weeks when stored at-20 C, but the UV-vis absorption features [Xmal
(e): 356 (1870), 490 (940) nm] at room temperature bleached upon brief application of …

A novel series of trans-N-aryl-2,5-dimethylpiperazine-1-carboxamide derivatives was
synthesized and their androgen receptor (AR) antagonist activities and in vivo antiandrogenic …

The radical cyclizations of (±)-f£)-3-((2-(bromomethyl) butoxy) carbonyl) prop-2-enoates 11
and 12 and (±)-ethyl (£)-3-{/V-[2-(bromomethyl) butyl]-/V-[2-(3-indolyl) ethyl] carbamoyl} prop-…

Arginine vasopressin (AVP) has a dual action mainly in the periphery, ie, vasoconstriction and
water reabsorption via V 1A and V 2 receptors; it may play a role in a number of diseases, …