How should values of pA2 and affinity constants for pharmacological competitive antagonists be estimated?

J Pharm Pharmacol. 1978 May;30(5):312-3. doi: 10.1111/j.2042-7158.1978.tb13237.x.
No abstract available

MeSH terms

  • Binding, Competitive
  • Drug Antagonism*
  • Mathematics
  • Models, Biological
  • Pharmaceutical Preparations / metabolism*
  • Receptors, Drug / metabolism*

Substances

  • Pharmaceutical Preparations
  • Receptors, Drug