Overcoming roadblocks in lead optimization: a thermodynamic perspective
Chem Biol Drug Des
.
2006 Jan;67(1):2-4.
doi: 10.1111/j.1747-0285.2005.00314.x.
Authors
Adam J Ruben
1
,
Yoshiaki Kiso
,
Ernesto Freire
Affiliation
1
Department of Biology, Johns Hopkins University, Baltimore, MD 21218, USA.
PMID:
16492143
DOI:
10.1111/j.1747-0285.2005.00314.x
No abstract available
Publication types
Research Support, N.I.H., Extramural
Research Support, U.S. Gov't, Non-P.H.S.
MeSH terms
Animals
Drug Design*
Drug Interactions
Humans
Kinetics
Protein Binding
Thermodynamics*
Grants and funding
GM 56550/GM/NIGMS NIH HHS/United States
GM 57144/GM/NIGMS NIH HHS/United States