Overcoming roadblocks in lead optimization: a thermodynamic perspective

Chem Biol Drug Des. 2006 Jan;67(1):2-4. doi: 10.1111/j.1747-0285.2005.00314.x.
No abstract available

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Drug Design*
  • Drug Interactions
  • Humans
  • Kinetics
  • Protein Binding
  • Thermodynamics*