Effects of β-funaltrexamine on radiolabeled opioid binding
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Reversibility of opioid receptor occupancy of buprenorphine in vivo
2006, European Journal of PharmacologyMechanisms involved in morphine-induced activation of synaptosomal Na<sup>+</sup>,K<sup>+</sup>-ATPase
2002, Brain ResearchCitation Excerpt :In particular two opioid receptor subtypes known as μ1 and μ2 have been described [31,32]. β-FNA blocks both μ1 and μ2 opioid receptors [34,36], whereas pretreatment of the animals 24 h before the experiment with 35 mg/kg of naloxonazine predominantly blocks the μ1-opioid receptor [13,34]. This led us to study the effect of naloxonazine on the morphine-induced increase in Na+,K+-ATPase activity.
Determination of the amino acid residue involved in [<sup>3</sup>H]β- funaltrexamine covalent binding in the cloned rat μ opioid receptor
1996, Journal of Biological Chemistry
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