Affinity of α5IA for human recombinant and native rat brain GABAA receptors
Affinity at α1-, α2-, α3-, and α5-containing recombinant as well as native rat brain GABAA receptor was measured using a [3H]flumazenil binding assay, whereas affinity for receptors containing either an α4 or α6 subunit was measured using [3H]Ro 15-4513. Data are the mean ± S.E.M. (n = 3–6 separate determinations).
Human Recombinant GABAA Receptors Containing β3, γ2 Plus