-Log KD values determined from inhibition of [3H]CGP 12177 binding to intact C2C12 cells Values represent mean ± S.E.M. of -log KD values obtained from inhibition of the specific binding of [3H]CGP12177 (1 nM). Nonspecific binding was determined with 1 μM ICI 118551. n gives the number of separate experiments.
Ligand | –log KD | n |
|---|---|---|
| Terbutaline | 5.9 ± 0.1 | 7 |
| Salbutamol | 6.4 ± 0.1 | 8 |
| Noradrenaline | 5.5 ± 0.0 | 8 |
| Isoprenaline | 7.0 ± 0.1 | 8 |
| Adrenaline | 7.2 ± 0.1 | 8 |
| Salmeterol | 8.7 ± 0.0 | 4 |