TABLE 3

Competition binding data (24-well plate method) showing pKi values for each tested peptide at RXFP1, RXFP2, RXFP1-BP, and RXFP2-BP

Values are expressed as means ± the standard error of the mean of three to four experiments.




H2 Relaxin

H3 Relaxin

INSL3

Rhesus Monkey Relaxin
RXFP1 10.18 ± 0.23 8.01 ± 0.19 5.38 ± 0.83 U.T.
RXFP2 9.21 ± 0.13 U.T. 9.69 ± 0.20 7.86 ± 0.20
RXFP1-BP 9.53 ± 0.25* 8.28 ± 0.17 7.67 ± 0.22* U.T.
RXFP2-BP
9.46 ± 0.12
U.T.
9.69 ± 0.19
7.48 ± 0.10
  • U.T., untested.

  • * p < 0.05 versus RXFP1 (unpaired t test).