TABLE 1

Selectivity profile of BAY 61-3606 in six tyrosine kinase assays Ki values were shown as mean ± S.E. of two independent experiments.


Enzymes

Ki
nM
Syk 7.5 ± 2.5
Lyn >5,400
Fyn >12,500
Src >6,250
Itk >4,700
Btk
>5,000