Ki values of unlabeled compounds on the uptake of [14C]salicylate into rOat2-expressed LLC-PK1 cells
| Inhibitors | Ki Values |
|---|---|
| μM | |
| Indocyanine green | 1.15 ± 0.18 |
| Ketoprofen | 1.84 ± 1.84 |
| Glibenclamide | 12.3 ± 2.1 |
| Diclofenac | 49.3 ± 10.0 |
| Benzoate | 86.9 ± 12.7 |
| Verapamil | 142 ± 59 |
| Ibuprofen | 155 ± 23 |
| Tolbutamide | 176 ± 32 |
Data were taken from Fig. 5. The effects of unlabeled compounds on the uptake of [14C]salicylate into rOat2-expressed cells were examined. These Ki values were determined by nonlinear regression analysis.