Table 1

Percentage of dopamine transporter occupancy determined with PET following i.v. cocaine administration

SubjectCocaine Dose
0.1 mg/kg1.0 mg/kg
RMk-353.092.1
RLm-155.895.5
RL1–444.284.0
RLk-452.783.6
RSu-359.188.0
Avg. ± S.D.53  ±587  ± 5