Receptor | Racemic Mecamylamine | R-(−)-Mecamylamine | S-(+)-Mecamylamine |
---|---|---|---|
α3β4 | 640–90 nM | 420–50 nM | 640–200 nM |
α4β2 | 2.5–0.6 μM | 1.7–0.5 μM | 3.2–0.5 μM |
α3β2 | 3.6–1.2 μM | 3.2–0.6 μM | 3.7–0.8 μM |
α7 | 6.9–1.6 μM | 5.8–2.2 μM | 4.6–1.2 μM |
α1β1δε | N.A. | 1.1–0.3 μM | 2.2–0.6 μM |
N.A., not available.