Receptor Subtype | Tissue | Radioligand | IC50/Ki(nM) |
---|---|---|---|
Serotonergic | |||
h5-HT1A | CHO cell line | [3H]-8-OH-DPAT | 540 |
5-HT1A | rat hippocampus | [3H]-8-OH-DPAT | >1000 |
5-HT1B | rat cortex | [125I]-cyanopindolol | >10000 |
5-HT1D | guinea pig striatum | [3H]-5-HT | >10000 |
5-HT2A | rat cortex | [3H]-ketanserin | >1000 |
5-HT2C | pig choroid plexus | [3H]-mesulergine | >1000 |
5-HT3 | rat cortex | [3H]-BRL 43694 | >10000 |
5-HT4 | guinea-pig striatum | [3H]-GR 113808 | >10000 |
r5-HT6 | HEK 293 cell line | [3H]-LSD | >10000 |
r5-HT7 | HEK 293 cell line | [3H]-LSD | >1000 |
Adrenergic | |||
α1 | rat cortex | [3H]-prazosin | 967 |
α2 | rat cortex | [3H]-RX 821002 | >1000 |
hα2A | CHO cell line | [3H]-RX 821002 | 249 |
hα2B | CHO cell line | [3H]-RX 821002 | >1000 |
hα2C | CHO cell line | [3H]-RX 821002 | 336 |
hβ1 | Sf9 cell line | [3H]-CGP 12177 | >1000 |
hβ2 | Sf9 cell line | [3H]-CGP 12177 | >1000 |
Histaminic | |||
H1 | guinea pig cerebellum | [3H]-pyrilamine | >1000 |
H2 | guinea pig brain | [3H]-tiotidine | >10000 |
Muscarinic | |||
hM1 | CHO cell line | [3H]-pirenzepine | >1000 |
hM2 | CHO cell line | [3H]-AF-DX 384 | >1000 |
hM3 | CHO cell line | [3H]-NMS | >10000 |
hM4 | CHO cell line | [3H]-NMS | >10000 |
All data are IC50 values except for Kivalues at h5-HT1A, α1, hα2A and hα2C receptors.