Table 3

Equilibrium dissociation constants (Kd values) of SR141716A calculated in the presence of five cannabinoid receptor agonists

Agonist usedKd (95% limits)
nM
WIN 55,212-20.33  (0.22–0.78)
CP 55,9400.14  (0.01–0.20)
HU-2100.40  (0.08–1.22)
Deoxy-HU2100.06  (0.01–0.16)
Fluoro-methanandamide0.33  (0.08–0.90)