Comparison of the NOP affinity and antagonistic potency of BTRX-246040 and SB-612111
Receptor-binding and stimulated GTPγS-binding data are taken from Statnick et al. (2016) for BTRX-246040 and from Spagnolo et al. (2007) for SB-612111. Receptor-binding data are expressed as pKi, GTPγS-binding and BRET data are expressed as pKB, and other data are expressed as pA2.