pIC50u | pIC50 | Imax | Emax | E0 | Cell Density | Number of Observations | |
---|---|---|---|---|---|---|---|
% | pg/ml | pg/ml | 105/ml | ||||
AM in vitro | 9.0 ± 0.1 | 9.0 ± 0.1 | 62 ± 5 | 469.9 ± 92.7 | 244.7 ± 44.0 | 3.125 | 4 |
PBMC in vitro | 8.4 ± 0.1 | 8.4 ± 0.1 | 100 | 3909.0 ± 351.0 | 175.0 ± 28.5 | 9.6 | 14 |
Whole blood in vitro | 8.7 ± 0.1 | 8.1 ± 0.1 | 100 | 544.1 ± 140.5 | 0.0 ± 0.0 | N/A | 11 |
Whole blood ex vivo | 8.8 ± 0.1 | 8.2 ± 0.1 | 95 ± 7 | 2021.2 ± 124.9 | 11 ± 1.0 | N/A | 36 |
AM, alveolar macrophages.