Tissue | Compound | c (h × µM) | S.E. (h × µM) | 95% t-CI (h × µM) | AUC0–12 (h × µM) | Ratio of AUC0–12 Tissue vs. Plasma |
---|---|---|---|---|---|---|
LV myocardium | cDEXs | 632 | 38 | 546–719 | 632 | 0.75 |
cADR-925 | 111 | 13 | 80–142 | 111 | 0.46 | |
Liver | cDEX | 589 | 31 | 521–657 | 589 | 0.70 |
cADR-925 | 123 | 12 | 94–152 | 123 | 0.51 | |
Soleus | cDEX | 531 | 38 | 440–622 | 531 | 0.63 |
cADR-925 | 153 | 15 | 116–189 | 153 | 0.63 |