TABLE 1
IC
50
values for compounds against PI3K
δ
and BTK in kinase inhibition assay
PI3K
δ
BTK
nM
nM
Idelalisib
1.2
>100,000
Ibrutinib
640
0.142
MDVN1001
149
0.9
MDVN1002
25.9
695
MDVN1003
16.9
32.3