TABLE 1

Ki values of phlorizin and canagliflozin

InhibitorKi for SGLT1 (nM)Ki for SGLT2 (nM)
Phlorizin545.7 ± 56.89 (n = 3)102.3 ± 27.41 (n = 3)
Canagliflozin770.5 ± 85.19 (n = 5)4.0 ± 0.77 (n = 3)
  • Values are presented as the mean ± S.E.M.