Diterpene | Cardiac AC EC50 | Cardiac AC Efficacy | AC5 EC50 | AC5 Efficacy | ||
---|---|---|---|---|---|---|
μM | % | μM | % | |||
FS | 3.0 ± 0.2 | 100 | 4.0 ± 0.6 | 100 | ||
6A7DA-FS | 3.6 ± 0.5 | 76 ± 10 | 7.4 ± 2.8b | 103 ± 11b | ||
BODIPY-FS | 1.4 ± 0.5 | 54 ± 6 | 2.3 ± 1.1b | 48 ± 2b | ||
7DA-FS | 30.2 ± 10.2a | 83 ± 5a | 63.3 ± 10.6b | 63 ± 4b | ||
9d-FS | 38.6 ± 19.2a | 90 ± 12a | 65.3 ± 9.0b | 79 ± 10b | ||
DMB-FS | 17.4 ± 2.0a | 118 ± 4a | 48.0 ± 9.6b | 95 ± 1b | ||
1d-FS | Ineffective | Ineffectiveb |