pIC50 | α | |
---|---|---|
Antipsychotic | ||
Perlapine | 9.7 ± 0.1 | -1.01 ± 0.05 |
Clozapine | 9.4 ± 0.1 | -1.03 ± 0.03 |
Octoclothepin | 8.6 ± 0.1 | -1.01 ± 0.02 |
Clothiapine | 8.5 ± 0.1 | -0.95 ± 0.02 |
Loxapine | 8.3 ± 0.1 | -0.79 ± 0.06 |
Quetiapine | 8.3 ± 0.1 | -0.99 ± 0.01 |
JL-18 | 8.3 ± 0.1 | -0.97 ± 0.04 |
cis-Flupentixol | 8.1 ± 0.1 | -0.92 ± 0.05 |
Promazine | 7.9 ± 0.1 | -0.97 ± 0.02 |
Thiothixene | 7.9 ± 0.2 | -1.01 ± 0.04 |
Telfudazine | 7.8 ± 0.2 | -1.03 ± 0.01 |
Olanzapine | 7.8 ± 0.1 | -0.99 ± 0.02 |
Pimozide | 7.8 ± 0.2 | -1.03 ± 0.03 |
Mesioridazine | 7.7 ± 0.1 | -0.92 ± 0.07 |
trans-Flupentixol | 7.6 ± 0.1 | -0.96 ± 0.03 |
Prothypendyl | 7.6 ± 0.1 | -0.97 ± 0.04 |
Perazine | 7.5 ± 0.1 | -0.97 ± 0.02 |
Fluphenazine | 7.4 ± 0.1 | -0.97 ± 0.02 |
Amoxapine | 7.4 ± 0.1 | -0.94 ± 0.04 |
Chlorpromazine | 7.4 ± 0.1 | -0.94 ± 0.05 |
Thioridazine | 7.3 ± 0.1 | -0.91 ± 0.04 |
Thiospirone | 7.1 ± 0.1 | -0.98 ± 0.02 |
Chlorproethizene | 7.1 ± 0.2 | -0.91 ± 0.04 |
Fluspiriline | 6.8 ± 0.3 | -0.88 ± 0.09 |
Trifluoperazine | 6.5 ± 0.2 | -0.94 ± 0.06 |
MDL 10097 | 6.5 ± 0.1 | -0.74 ± 0.07 |
Amperozide | 6.4 ± 0.1 | -0.88 ± 0.03 |
Sertindole | 6.2 ± 0.3 | -0.93 ± 0.05 |
Moperone | 6.1 ± 0.2 | -0.83 ± 0.08 |
Spiperone | 5.9 ± 0.2 | -0.98 ± 0.08 |
Trifluperidol | 5.9 ± 0.2 | -0.85 ± 0.09 |
Haloperidol | 5.6 ± 0.1 | -0.55 ± 0.06 |
Butaclamol | 5.6 ± 0.3 | -0.89 ± 0.03 |
Risperidone | 5.5 ± 0.1 | -0.73 ± 0.06 |
Antidepressant | ||
Mirtazepine | 9.6 ± 0.1 | -0.90 ± 0.04 |
Doxepin | 9.2 ± 0.1 | -0.96 ± 0.03 |
Amitypriline | 8.9 ± 0.2 | -0.95 ± 0.05 |
Trimipramine | 8.7 ± 0.1 | -0.93 ± 0.01 |
Nortryptiline | 7.9 ± 0.2 | -1.05 ± 0.04 |
Imitramine | 7.5 ± 0.1 | -0.90 ± 0.05 |
Protrypriline | 7.3 ± 0.1 | -1.04 ± 0.05 |
Clomipramine | 6.9 ± 0.2 | -0.96 ± 0.02 |
Desipramine | 6.7 ± 0.1 | -0.92 ± 0.05 |
Trazodone | 6.3 ± 0.1 | -0.82 ± 0.05 |
Buspirone | 6.0 ± 0.2 | -0.80 ± 0.05 |
Flouxetine | 5.9 ± 0.2 | -0.62 ± 0.03 |
Zimelidine | 5.3 ± 0.1 | N.D. |
Serotonergic | ||
Cyproheptadine | 9.4 ± 0.1 | -0.81 ± 0.08 |
Mianserin | 9.0 ± 0.1 | -0.99 ± 0.01 |
Methiothepin | 8.8 ± 0.2 | -0.96 ± 0.03 |
Ritanserin | 7.0 ± 0.1 | -0.93 ± 0.02 |
Ketanserin | 6.6 ± 0.1 | -0.90 ± 0.01 |
Pirenpirone | 6.4 ± 0.1 | -0.74 ± 0.09 |
Cinanserin | 6.1 ± 0.4 | -0.98 ± 0.04 |
LY 53,857 | 5.9 ± 0.2 | -0.65 ± 0.04 |
Metergoline | 5.8 ± 0.2 | -0.79 ± 0.09 |
m-Chlorophenylpiperazine | 5.7 ± 0.2 | -0.74 ± 0.05 |
Dopaminergic | ||
Prochlorperazine | 6.7 ± 0.2 | -0.94 ± 0.05 |
Muscarinic | ||
Benztropine | 7.7 ± 0.2 | -0.91 ± 0.02 |
N.D., not determined.