NSAID | MRP2 | MRP4 | |
---|---|---|---|
μM | |||
Salicylate | 1760 ± 30 | 1500 ± 20 | |
Piroxicam | 257 ± 2 | 216 ± 2 | |
Ibuprofen | 930 ± 20 | 26.3 ± 0.3 | |
Naproxen | 609 ± 7 | 42.3 ± 0.3 | |
Sulindac | 38 ± 1 | 2.11 ± 0.02 | |
Tolmetin | 494 ± 5 | 20.5 ± 0.3 | |
Etodolac | 480 ± 2a | 120 ± 1 | |
Diclofenac | 97 ± 1 | 0.006 ± 0.001 (H) | |
326 ± 6 (L) | |||
Indomethacin | 0.06 ± 0.01 (H) | 6.1 ± 0.1 | |
46 ± 1 (L) | |||
Ketoprofen | 1.4 ± 0.1 (H) | 11.9 ± 0.1 | |
470 ± 20 (L) | |||
Celecoxib | 100 ± 2 | 35 ± 1b | |
Phenylbutazone | 605 ± 4b | 130 ± 2 |