Research ArticleDrug Discovery and Translational Medicine
Relative Selectivity of Covalent Inhibitors Requires Assessment of Inactivation Kinetics and Cellular Occupancy: A Case Study of Ibrutinib and Acalabrutinib
Melissa Hopper, Tarikere Gururaja, Taisei Kinoshita, James P Dean, Ronald J Hill and Ann Mongan
Journal of Pharmacology and Experimental Therapeutics December 23, 2019, jpet.119.262063; DOI: https://doi.org/10.1124/jpet.119.262063