OtherDrug Discovery and Translational Medicine
A novel selective PKR inhibitor restores cognitive deficits and neurodegeneration in Alzheimer's disease experimental model
Matilde Lopez-Grancha, Patrick Bernardelli, Nicolas Moindrot, Elisabeth Genet, Carine Vincent, Valerie Roudieres, Alain Krick, Jean-Francois Sabuco, David Machnik, Delphine Ibghi, Laurent Pradier and Veronique Taupin
Journal of Pharmacology and Experimental Therapeutics June 16, 2021, JPET-AR-2021-000590; DOI: https://doi.org/10.1124/jpet.121.000590
Matilde Lopez-Grancha
1Neurodegeneration Cluster, Rare and Neurologic Disease Research TA, Sanofi R&D, France
Patrick Bernardelli
2Integrated Drug Discovery, Sanofi R&D, France
Nicolas Moindrot
1Neurodegeneration Cluster, Rare and Neurologic Disease Research TA, Sanofi R&D, France
Elisabeth Genet
1Neurodegeneration Cluster, Rare and Neurologic Disease Research TA, Sanofi R&D, France
Carine Vincent
1Neurodegeneration Cluster, Rare and Neurologic Disease Research TA, Sanofi R&D, France
Valerie Roudieres
1Neurodegeneration Cluster, Rare and Neurologic Disease Research TA, Sanofi R&D, France
Alain Krick
3DMPK, Sanofi R&D, France
Jean-Francois Sabuco
4medicinal chemistry, evotec Id, France
David Machnik
5Integrated drug discovery, Sanofi R&D, France
Delphine Ibghi
1Neurodegeneration Cluster, Rare and Neurologic Disease Research TA, Sanofi R&D, France
Laurent Pradier
1Neurodegeneration Cluster, Rare and Neurologic Disease Research TA, Sanofi R&D, France
Veronique Taupin
6PreClinicalSafety, Sanofi R&D, France
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In this issue
OtherDrug Discovery and Translational Medicine
New potent PKR inhibitor for Alzheimer's disease
Matilde Lopez-Grancha, Patrick Bernardelli, Nicolas Moindrot, Elisabeth Genet, Carine Vincent, Valerie Roudieres, Alain Krick, Jean-Francois Sabuco, David Machnik, Delphine Ibghi, Laurent Pradier and Veronique Taupin
Journal of Pharmacology and Experimental Therapeutics June 16, 2021, JPET-AR-2021-000590; DOI: https://doi.org/10.1124/jpet.121.000590
OtherDrug Discovery and Translational Medicine
New potent PKR inhibitor for Alzheimer's disease
Matilde Lopez-Grancha, Patrick Bernardelli, Nicolas Moindrot, Elisabeth Genet, Carine Vincent, Valerie Roudieres, Alain Krick, Jean-Francois Sabuco, David Machnik, Delphine Ibghi, Laurent Pradier and Veronique Taupin
Journal of Pharmacology and Experimental Therapeutics June 16, 2021, JPET-AR-2021-000590; DOI: https://doi.org/10.1124/jpet.121.000590
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