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Journal of Pharmacology and Experimental Therapeutics

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OtherNeuropharmacology

A Novel Potent and Selective Histamine H3 Receptor Antagonist Enerisant: In Vitro Profiles, In Vivo Receptor Occupancy, Wake-Promoting and Pro-cognitive Effects in Rodents

Noriko Hino, Toshiyuki Marumo, Makiko Kotani, Toshiharu Shimazaki, Ayaka Kaku-Fukumoto, Hirohiko Hikichi, Jun-ichi Karasawa, Yasumitsu Tomishima, Hiroko Komiyama, Emi Tatsuda, Dai Nozawa, Toshio Nakamura and Shigeyuki Chaki
Journal of Pharmacology and Experimental Therapeutics August 29, 2020, JPET-AR-2020-000185; DOI: https://doi.org/10.1124/jpet.120.000185
Noriko Hino
1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
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Toshiyuki Marumo
1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
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Makiko Kotani
1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
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Toshiharu Shimazaki
1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
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Ayaka Kaku-Fukumoto
1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
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Hirohiko Hikichi
1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
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Jun-ichi Karasawa
1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
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Yasumitsu Tomishima
1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
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Hiroko Komiyama
1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
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Emi Tatsuda
1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
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Dai Nozawa
1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
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Toshio Nakamura
2Taisho Pharmaceutical Co., Ltd., Japan
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Shigeyuki Chaki
1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
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  • For correspondence: s-chaki@taisho.co.jp
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Article Information

JPET-AR-2020-000185
DOI 
https://doi.org/10.1124/jpet.120.000185
PubMed 
32862143

Published By 
American Society for Pharmacology and Experimental Therapeutics
Print ISSN 
0022-3565
Online ISSN 
1521-0103
History 
  • Published online August 29, 2020.

Article Versions

  • You are currently viewing an Earlier version of this article (August 29, 2020 - 05:17).
  • View the most recent version of this article
Copyright & Usage 
Copyright © 2020 American Society for Pharmacology and Experimental Therapeutics

Author Information

  1. Noriko Hino1,
  2. Toshiyuki Marumo1,
  3. Makiko Kotani1,
  4. Toshiharu Shimazaki1,
  5. Ayaka Kaku-Fukumoto1,
  6. Hirohiko Hikichi1,
  7. Jun-ichi Karasawa1,
  8. Yasumitsu Tomishima1,
  9. Hiroko Komiyama1,
  10. Emi Tatsuda1,
  11. Dai Nozawa1,
  12. Toshio Nakamura2, and
  13. Shigeyuki Chaki1,*
  1. 1Research Headquarters, Taisho Pharmaceutical Co., Ltd., Japan
  2. 2Taisho Pharmaceutical Co., Ltd., Japan
  1. ↵* Corresponding Author:
    Shigeyuki Chaki, Research Headquarters, Taisho Pharmaceutical Co., Ltd., 1-403 Yoshino-cho, Kita-ku, Saitama, N/A, 331-9530, Japan. E-mail: s-chaki{at}taisho.co.jp

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Article usage: August 2020 to February 2021

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Aug 2020110045
Sep 20201800125
Oct 20203182787
Nov 20202004884
Dec 20201122244
Jan 2021801738
Feb 2021841237

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Journal of Pharmacology and Experimental Therapeutics: 376 (3)
Journal of Pharmacology and Experimental Therapeutics
Vol. 376, Issue 3
1 Mar 2021
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OtherNeuropharmacology

Pharmacological profiles of enelisant

Noriko Hino, Toshiyuki Marumo, Makiko Kotani, Toshiharu Shimazaki, Ayaka Kaku-Fukumoto, Hirohiko Hikichi, Jun-ichi Karasawa, Yasumitsu Tomishima, Hiroko Komiyama, Emi Tatsuda, Dai Nozawa, Toshio Nakamura and Shigeyuki Chaki
Journal of Pharmacology and Experimental Therapeutics August 29, 2020, JPET-AR-2020-000185; DOI: https://doi.org/10.1124/jpet.120.000185

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OtherNeuropharmacology

Pharmacological profiles of enelisant

Noriko Hino, Toshiyuki Marumo, Makiko Kotani, Toshiharu Shimazaki, Ayaka Kaku-Fukumoto, Hirohiko Hikichi, Jun-ichi Karasawa, Yasumitsu Tomishima, Hiroko Komiyama, Emi Tatsuda, Dai Nozawa, Toshio Nakamura and Shigeyuki Chaki
Journal of Pharmacology and Experimental Therapeutics August 29, 2020, JPET-AR-2020-000185; DOI: https://doi.org/10.1124/jpet.120.000185
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