Research ArticleDrug Discovery and Translational Medicine
A novel G protein-biased agonist at the δ opioid receptor with analgesic efficacy in models of chronic pain
Alexandra E Conibear, Junaid Asghar, Rob Hill, Graeme Henderson, Eva Borbely, Valeria Tekus, Zsuzsanna Helyes, Jo Palandri, Chris P Bailey, Ingemar Starke, Bengt von Mentzer, David Kendall and Eamonn Kelly
Journal of Pharmacology and Experimental Therapeutics October 8, 2019, jpet.119.258640; DOI: https://doi.org/10.1124/jpet.119.258640
Alexandra E Conibear
1 University of Bristol, UK;
Junaid Asghar
2 Gomal University, Pakistan;
Rob Hill
1 University of Bristol, UK;
Graeme Henderson
1 University of Bristol, UK;
Eva Borbely
3 PharmInVivo Ltd, University of Pecs, Hungary;
Valeria Tekus
3 PharmInVivo Ltd, University of Pecs, Hungary;
Zsuzsanna Helyes
3 PharmInVivo Ltd, University of Pecs, Hungary;
Jo Palandri
4 Department of Pharmacy & Pharmacology, University of Bath, UK;
Chris P Bailey
5 University of Bath;
Ingemar Starke
6 PharmNovo AB, Tangenvagen 7, 456 32 Kungshamn, Sweden
Bengt von Mentzer
6 PharmNovo AB, Tangenvagen 7, 456 32 Kungshamn, Sweden
David Kendall
6 PharmNovo AB, Tangenvagen 7, 456 32 Kungshamn, Sweden
Eamonn Kelly
1 University of Bristol, UK;
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Research ArticleDrug Discovery and Translational Medicine
A novel G protein-biased agonist at the δ opioid receptor with analgesic efficacy in models of chronic pain
Alexandra E Conibear, Junaid Asghar, Rob Hill, Graeme Henderson, Eva Borbely, Valeria Tekus, Zsuzsanna Helyes, Jo Palandri, Chris P Bailey, Ingemar Starke, Bengt von Mentzer, David Kendall and Eamonn Kelly
Journal of Pharmacology and Experimental Therapeutics October 8, 2019, jpet.119.258640; DOI: https://doi.org/10.1124/jpet.119.258640
Research ArticleDrug Discovery and Translational Medicine
A novel G protein-biased agonist at the δ opioid receptor with analgesic efficacy in models of chronic pain
Alexandra E Conibear, Junaid Asghar, Rob Hill, Graeme Henderson, Eva Borbely, Valeria Tekus, Zsuzsanna Helyes, Jo Palandri, Chris P Bailey, Ingemar Starke, Bengt von Mentzer, David Kendall and Eamonn Kelly
Journal of Pharmacology and Experimental Therapeutics October 8, 2019, jpet.119.258640; DOI: https://doi.org/10.1124/jpet.119.258640
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