Research ArticleCardiovascular
Discovery and Preclinical Characterization of GSK1278863 (daprodustat), A Small Molecule Hypoxia Inducible Factor (HIF)-Prolyl Hydroxylase Inhibitor for Anemia
Jennifer L Ariazi, Kevin J Duffy, David F Adams, Duke M Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-Miller
Journal of Pharmacology and Experimental Therapeutics September 19, 2017, jpet.117.242503; DOI: https://doi.org/10.1124/jpet.117.242503
Jennifer L Ariazi
1 GlaxoSmithKline;
Kevin J Duffy
1 GlaxoSmithKline;
David F Adams
1 GlaxoSmithKline;
Duke M Fitch
1 GlaxoSmithKline;
Lusong Luo
2 Beigene;
Melissa Pappalardi
1 GlaxoSmithKline;
Mangatt Biju
1 GlaxoSmithKline;
Erin Hugger DiFilippo
3 formerly at GSK;
Tony Shaw
1 GlaxoSmithKline;
Ken Wiggall
1 GlaxoSmithKline;
Connie Erickson-Miller
4 Adaptimmune
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Research ArticleCardiovascular
Discovery and Preclinical Characterization of GSK1278863 (daprodustat), A Small Molecule Hypoxia Inducible Factor (HIF)-Prolyl Hydroxylase Inhibitor for Anemia
Jennifer L Ariazi, Kevin J Duffy, David F Adams, Duke M Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-Miller
Journal of Pharmacology and Experimental Therapeutics September 19, 2017, jpet.117.242503; DOI: https://doi.org/10.1124/jpet.117.242503
Research ArticleCardiovascular
Discovery and Preclinical Characterization of GSK1278863 (daprodustat), A Small Molecule Hypoxia Inducible Factor (HIF)-Prolyl Hydroxylase Inhibitor for Anemia
Jennifer L Ariazi, Kevin J Duffy, David F Adams, Duke M Fitch, Lusong Luo, Melissa Pappalardi, Mangatt Biju, Erin Hugger DiFilippo, Tony Shaw, Ken Wiggall and Connie Erickson-Miller
Journal of Pharmacology and Experimental Therapeutics September 19, 2017, jpet.117.242503; DOI: https://doi.org/10.1124/jpet.117.242503
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