Research ArticleMetabolism, Transport, and Pharmacogenomics
Blood-Brain Barrier (BBB) Pharmacoproteomics (PPx): Reconstruction of In Vivo Brain Distribution of 11 P-glycoprotein Substrates based on the BBB Transporter Protein Concentration, In Vitro Intrinsic Transport Activity, and Unbound Fraction in Plasma and Brain in Mice
Yasuo Uchida, Sumio Ohtsuki, Junichi Kamiie and Tetsuya Terasaki
Journal of Pharmacology and Experimental Therapeutics August 9, 2011, jpet.111.184200; DOI: https://doi.org/10.1124/jpet.111.184200