Index by author
March 01, 2021; Volume 376,Issue 3
A
Ahlschwede, Kristen M.
- You have accessDistinct Uptake Kinetics of Alzheimer Disease Amyloid-β 40 and 42 at the Blood-Brain Barrier EndotheliumNidhi Sharda, Kristen M. Ahlschwede, Geoffry L. Curran, Val J. Lowe and Karunya K. KandimallaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 482-490; DOI: https://doi.org/10.1124/jpet.120.000086
Ahmed-Belkacem, Abdelhakim
- You have accessA Phenyl-Pyrrolidine Derivative Reveals a Dual Inhibition Mechanism of Myocardial Mitochondrial Permeability Transition Pore, Which Is Limited by Its Myocardial DistributionMathieu Panel, Abdelhakim Ahmed-Belkacem, Isaac Ruiz, Jean-François Guichou, Jean-Michel Pawlotsky, Bijan Ghaleh and Didier MorinJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 348-357; DOI: https://doi.org/10.1124/jpet.120.000359
Anderson, Mitchell
- Open AccessNovel Tocolytic Strategy: Modulating Cx43 Activity by S-NitrosationScott D. Barnett, Hazik Asif, Mitchell Anderson and Iain L. O. BuxtonJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 444-453; DOI: https://doi.org/10.1124/jpet.120.000427
Asai, Kuniya
- You have accessβ3-Adrenergic Receptor Agonist Prevents Diastolic Dysfunction in an Angiotensin II–Induced Cardiomyopathy Mouse ModelMasataka Kamiya, Kuniya Asai, Yasuhiro Maejima, Akihiro Shirakabe, Koji Murai, Satsuki Noma, Hidenori Komiyama, Naoki Sato, Kyoichi Mizuno and Wataru ShimizuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 473-481; DOI: https://doi.org/10.1124/jpet.120.000140
Asif, Hazik
- Open AccessNovel Tocolytic Strategy: Modulating Cx43 Activity by S-NitrosationScott D. Barnett, Hazik Asif, Mitchell Anderson and Iain L. O. BuxtonJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 444-453; DOI: https://doi.org/10.1124/jpet.120.000427
B
Bai, Dongdong
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
Banks, M.L.
- You have accessManipulating Pharmacodynamic Efficacy with Agonist + Antagonist Mixtures: In Vitro and In Vivo Studies with Opioids and CannabinoidsD.E. Selley, M.L. Banks, C.M. Diester, A.M. Jali, L.P. Legakis, E.J. Santos and S.S. NegusJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 374-384; DOI: https://doi.org/10.1124/jpet.120.000349
Barnett, Scott D.
- Open AccessNovel Tocolytic Strategy: Modulating Cx43 Activity by S-NitrosationScott D. Barnett, Hazik Asif, Mitchell Anderson and Iain L. O. BuxtonJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 444-453; DOI: https://doi.org/10.1124/jpet.120.000427
Behm, David J.
- You have accessIdentification of a Human Whole Blood–Based Endothelial Cell Impedance Assay for Assessing Clinical Transient Receptor Potential Vanilloid 4 Target Engagement Ex VivoXiaoping Xu, Navin Goyal, Melissa H. Costell, Theresa Roethke, Christian H. James, Kevin S. Thorneloe, Jaclyn Patterson, Patrick Stoy, Krista Goodman, Dennis L. Sprecher and David J. BehmJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 436-443; DOI: https://doi.org/10.1124/jpet.120.000307
Bender, Andrew T.
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
Borhegyi, Zsolt
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Braun, Tobias
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Buxton, Iain L. O.
- Open AccessNovel Tocolytic Strategy: Modulating Cx43 Activity by S-NitrosationScott D. Barnett, Hazik Asif, Mitchell Anderson and Iain L. O. BuxtonJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 444-453; DOI: https://doi.org/10.1124/jpet.120.000427
C
Cantrill, Carina
- You have accessCalculation of an Apical Efflux Ratio from P-Glycoprotein (P-gp) In Vitro Transport Experiments Shows an Improved Correlation with In Vivo Cerebrospinal Fluid Measurements in Rats: Impact on P-gp Screening and Compound OptimizationHolger Fischer, Claudia Senn, Mohammed Ullah, Carina Cantrill, Franz Schuler and Li YuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 322-329; DOI: https://doi.org/10.1124/jpet.120.000158
Cao, Pingfeng
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
Chen, Dapeng
- You have accessPhytochemical Regulation of RNA in Treating Inflammatory Bowel Disease and Colon Cancer: Inspirations from Cell and Animal StudiesGuolin Zhang, Chi Zhang, Jia’ao Sun, Yongjian Xiong, Liang Wang and Dapeng ChenJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 464-472; DOI: https://doi.org/10.1124/jpet.120.000354
Chen, Lei
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
Costell, Melissa H.
- You have accessIdentification of a Human Whole Blood–Based Endothelial Cell Impedance Assay for Assessing Clinical Transient Receptor Potential Vanilloid 4 Target Engagement Ex VivoXiaoping Xu, Navin Goyal, Melissa H. Costell, Theresa Roethke, Christian H. James, Kevin S. Thorneloe, Jaclyn Patterson, Patrick Stoy, Krista Goodman, Dennis L. Sprecher and David J. BehmJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 436-443; DOI: https://doi.org/10.1124/jpet.120.000307
Crowley, Morgan L.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Curran, Geoffry L.
- You have accessDistinct Uptake Kinetics of Alzheimer Disease Amyloid-β 40 and 42 at the Blood-Brain Barrier EndotheliumNidhi Sharda, Kristen M. Ahlschwede, Geoffry L. Curran, Val J. Lowe and Karunya K. KandimallaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 482-490; DOI: https://doi.org/10.1124/jpet.120.000086
D
Déri, Máté T.
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Deshpande, Aditee
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
Diester, C.M.
- You have accessManipulating Pharmacodynamic Efficacy with Agonist + Antagonist Mixtures: In Vitro and In Vivo Studies with Opioids and CannabinoidsD.E. Selley, M.L. Banks, C.M. Diester, A.M. Jali, L.P. Legakis, E.J. Santos and S.S. NegusJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 374-384; DOI: https://doi.org/10.1124/jpet.120.000349
Ding, Zheng-Ming
- You have accessSelf-Administration of Cotinine in Wistar Rats: Comparisons to NicotineZheng-Ming Ding, Yong Gao, Alena M. Sentir and Xiaoying TanJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 338-347; DOI: https://doi.org/10.1124/jpet.120.000367
F
Farahanchi, Nazli
- You have accessRNA Interference Targeting Liver Angiopoietin-Like Protein 3 Protects from Nephrotic Syndrome in a Rat Model Via Amelioration of Pathologic HypertriglyceridemiaYitong Zhao, Masaki Goto, Nosratola D. Vaziri, Mahyar Khazaeli, Han Liu, Nazli Farahanchi, Elham Khanifar, Ted Farzaneh, Patrick A. Haslett, Hamid Moradi and Mangala M. SoundarapandianJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 428-435; DOI: https://doi.org/10.1124/jpet.120.000257
Farzaneh, Ted
- You have accessRNA Interference Targeting Liver Angiopoietin-Like Protein 3 Protects from Nephrotic Syndrome in a Rat Model Via Amelioration of Pathologic HypertriglyceridemiaYitong Zhao, Masaki Goto, Nosratola D. Vaziri, Mahyar Khazaeli, Han Liu, Nazli Farahanchi, Elham Khanifar, Ted Farzaneh, Patrick A. Haslett, Hamid Moradi and Mangala M. SoundarapandianJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 428-435; DOI: https://doi.org/10.1124/jpet.120.000257
Fischer, Holger
- You have accessCalculation of an Apical Efflux Ratio from P-Glycoprotein (P-gp) In Vitro Transport Experiments Shows an Improved Correlation with In Vivo Cerebrospinal Fluid Measurements in Rats: Impact on P-gp Screening and Compound OptimizationHolger Fischer, Claudia Senn, Mohammed Ullah, Carina Cantrill, Franz Schuler and Li YuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 322-329; DOI: https://doi.org/10.1124/jpet.120.000158
Fortner, John D.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
G
Gamez-Jimenez, Lea R.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Gao, Yong
- You have accessSelf-Administration of Cotinine in Wistar Rats: Comparisons to NicotineZheng-Ming Ding, Yong Gao, Alena M. Sentir and Xiaoying TanJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 338-347; DOI: https://doi.org/10.1124/jpet.120.000367
Ghaleh, Bijan
- You have accessA Phenyl-Pyrrolidine Derivative Reveals a Dual Inhibition Mechanism of Myocardial Mitochondrial Permeability Transition Pore, Which Is Limited by Its Myocardial DistributionMathieu Panel, Abdelhakim Ahmed-Belkacem, Isaac Ruiz, Jean-François Guichou, Jean-Michel Pawlotsky, Bijan Ghaleh and Didier MorinJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 348-357; DOI: https://doi.org/10.1124/jpet.120.000359
Goodman, Krista
- You have accessIdentification of a Human Whole Blood–Based Endothelial Cell Impedance Assay for Assessing Clinical Transient Receptor Potential Vanilloid 4 Target Engagement Ex VivoXiaoping Xu, Navin Goyal, Melissa H. Costell, Theresa Roethke, Christian H. James, Kevin S. Thorneloe, Jaclyn Patterson, Patrick Stoy, Krista Goodman, Dennis L. Sprecher and David J. BehmJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 436-443; DOI: https://doi.org/10.1124/jpet.120.000307
Goto, Masaki
- You have accessRNA Interference Targeting Liver Angiopoietin-Like Protein 3 Protects from Nephrotic Syndrome in a Rat Model Via Amelioration of Pathologic HypertriglyceridemiaYitong Zhao, Masaki Goto, Nosratola D. Vaziri, Mahyar Khazaeli, Han Liu, Nazli Farahanchi, Elham Khanifar, Ted Farzaneh, Patrick A. Haslett, Hamid Moradi and Mangala M. SoundarapandianJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 428-435; DOI: https://doi.org/10.1124/jpet.120.000257
Gou, Xiaoli
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
Goyal, Navin
- You have accessIdentification of a Human Whole Blood–Based Endothelial Cell Impedance Assay for Assessing Clinical Transient Receptor Potential Vanilloid 4 Target Engagement Ex VivoXiaoping Xu, Navin Goyal, Melissa H. Costell, Theresa Roethke, Christian H. James, Kevin S. Thorneloe, Jaclyn Patterson, Patrick Stoy, Krista Goodman, Dennis L. Sprecher and David J. BehmJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 436-443; DOI: https://doi.org/10.1124/jpet.120.000307
Guichou, Jean-François
- You have accessA Phenyl-Pyrrolidine Derivative Reveals a Dual Inhibition Mechanism of Myocardial Mitochondrial Permeability Transition Pore, Which Is Limited by Its Myocardial DistributionMathieu Panel, Abdelhakim Ahmed-Belkacem, Isaac Ruiz, Jean-François Guichou, Jean-Michel Pawlotsky, Bijan Ghaleh and Didier MorinJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 348-357; DOI: https://doi.org/10.1124/jpet.120.000359
Gyimesi, Máté
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
H
Hamada, Hiroki
- You have accessDifferent Antioxidative and Antiapoptotic Effects of Piceatannol and ResveratrolRyusuke Hosoda, Hiroki Hamada, Daisuke Uesugi, Naotoshi Iwahara, Iyori Nojima, Yoshiyuki Horio and Atsushi KunoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 385-396; DOI: https://doi.org/10.1124/jpet.120.000096
Hamow, Kamirán Á.
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Haselmayer, Philipp
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
Haslett, Patrick A.
- You have accessRNA Interference Targeting Liver Angiopoietin-Like Protein 3 Protects from Nephrotic Syndrome in a Rat Model Via Amelioration of Pathologic HypertriglyceridemiaYitong Zhao, Masaki Goto, Nosratola D. Vaziri, Mahyar Khazaeli, Han Liu, Nazli Farahanchi, Elham Khanifar, Ted Farzaneh, Patrick A. Haslett, Hamid Moradi and Mangala M. SoundarapandianJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 428-435; DOI: https://doi.org/10.1124/jpet.120.000257
Hibi, Chihiro
- You have accessOpening of Intermediate Conductance Ca2+-Activated K+ Channels in C2C12 Skeletal Muscle Cells Increases the Myotube Diameter via the Akt/Mammalian Target of Rapamycin PathwayYuzo Iseki, Yuko Ono, Chihiro Hibi, Shoko Tanaka, Shunya Takeshita, Yuko Maejima, Junko Kurokawa, Masahiro Murakawa, Kenju Shimomura and Kazuho SakamotoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 454-462; DOI: https://doi.org/10.1124/jpet.120.000290
Hiranita, Takato
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Ho, Nicholas P.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Horio, Yoshiyuki
- You have accessDifferent Antioxidative and Antiapoptotic Effects of Piceatannol and ResveratrolRyusuke Hosoda, Hiroki Hamada, Daisuke Uesugi, Naotoshi Iwahara, Iyori Nojima, Yoshiyuki Horio and Atsushi KunoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 385-396; DOI: https://doi.org/10.1124/jpet.120.000096
Hosoda, Ryusuke
- You have accessDifferent Antioxidative and Antiapoptotic Effects of Piceatannol and ResveratrolRyusuke Hosoda, Hiroki Hamada, Daisuke Uesugi, Naotoshi Iwahara, Iyori Nojima, Yoshiyuki Horio and Atsushi KunoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 385-396; DOI: https://doi.org/10.1124/jpet.120.000096
I
Iseki, Yuzo
- You have accessOpening of Intermediate Conductance Ca2+-Activated K+ Channels in C2C12 Skeletal Muscle Cells Increases the Myotube Diameter via the Akt/Mammalian Target of Rapamycin PathwayYuzo Iseki, Yuko Ono, Chihiro Hibi, Shoko Tanaka, Shunya Takeshita, Yuko Maejima, Junko Kurokawa, Masahiro Murakawa, Kenju Shimomura and Kazuho SakamotoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 454-462; DOI: https://doi.org/10.1124/jpet.120.000290
Iwahara, Naotoshi
- You have accessDifferent Antioxidative and Antiapoptotic Effects of Piceatannol and ResveratrolRyusuke Hosoda, Hiroki Hamada, Daisuke Uesugi, Naotoshi Iwahara, Iyori Nojima, Yoshiyuki Horio and Atsushi KunoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 385-396; DOI: https://doi.org/10.1124/jpet.120.000096
J
Jali, A.M.
- You have accessManipulating Pharmacodynamic Efficacy with Agonist + Antagonist Mixtures: In Vitro and In Vivo Studies with Opioids and CannabinoidsD.E. Selley, M.L. Banks, C.M. Diester, A.M. Jali, L.P. Legakis, E.J. Santos and S.S. NegusJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 374-384; DOI: https://doi.org/10.1124/jpet.120.000349
James, Christian H.
- You have accessIdentification of a Human Whole Blood–Based Endothelial Cell Impedance Assay for Assessing Clinical Transient Receptor Potential Vanilloid 4 Target Engagement Ex VivoXiaoping Xu, Navin Goyal, Melissa H. Costell, Theresa Roethke, Christian H. James, Kevin S. Thorneloe, Jaclyn Patterson, Patrick Stoy, Krista Goodman, Dennis L. Sprecher and David J. BehmJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 436-443; DOI: https://doi.org/10.1124/jpet.120.000307
Johnson, Theresa L.
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
K
Kamiya, Masataka
- You have accessβ3-Adrenergic Receptor Agonist Prevents Diastolic Dysfunction in an Angiotensin II–Induced Cardiomyopathy Mouse ModelMasataka Kamiya, Kuniya Asai, Yasuhiro Maejima, Akihiro Shirakabe, Koji Murai, Satsuki Noma, Hidenori Komiyama, Naoki Sato, Kyoichi Mizuno and Wataru ShimizuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 473-481; DOI: https://doi.org/10.1124/jpet.120.000140
Kandimalla, Karunya K.
- You have accessDistinct Uptake Kinetics of Alzheimer Disease Amyloid-β 40 and 42 at the Blood-Brain Barrier EndotheliumNidhi Sharda, Kristen M. Ahlschwede, Geoffry L. Curran, Val J. Lowe and Karunya K. KandimallaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 482-490; DOI: https://doi.org/10.1124/jpet.120.000086
Khanifar, Elham
- You have accessRNA Interference Targeting Liver Angiopoietin-Like Protein 3 Protects from Nephrotic Syndrome in a Rat Model Via Amelioration of Pathologic HypertriglyceridemiaYitong Zhao, Masaki Goto, Nosratola D. Vaziri, Mahyar Khazaeli, Han Liu, Nazli Farahanchi, Elham Khanifar, Ted Farzaneh, Patrick A. Haslett, Hamid Moradi and Mangala M. SoundarapandianJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 428-435; DOI: https://doi.org/10.1124/jpet.120.000257
Khazaeli, Mahyar
- You have accessRNA Interference Targeting Liver Angiopoietin-Like Protein 3 Protects from Nephrotic Syndrome in a Rat Model Via Amelioration of Pathologic HypertriglyceridemiaYitong Zhao, Masaki Goto, Nosratola D. Vaziri, Mahyar Khazaeli, Han Liu, Nazli Farahanchi, Elham Khanifar, Ted Farzaneh, Patrick A. Haslett, Hamid Moradi and Mangala M. SoundarapandianJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 428-435; DOI: https://doi.org/10.1124/jpet.120.000257
Kiss, Ádám F.
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Komiyama, Hidenori
- You have accessβ3-Adrenergic Receptor Agonist Prevents Diastolic Dysfunction in an Angiotensin II–Induced Cardiomyopathy Mouse ModelMasataka Kamiya, Kuniya Asai, Yasuhiro Maejima, Akihiro Shirakabe, Koji Murai, Satsuki Noma, Hidenori Komiyama, Naoki Sato, Kyoichi Mizuno and Wataru ShimizuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 473-481; DOI: https://doi.org/10.1124/jpet.120.000140
Kornya, László
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Kovács, Mihály
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Krans, Jacob
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Kuno, Atsushi
- You have accessDifferent Antioxidative and Antiapoptotic Effects of Piceatannol and ResveratrolRyusuke Hosoda, Hiroki Hamada, Daisuke Uesugi, Naotoshi Iwahara, Iyori Nojima, Yoshiyuki Horio and Atsushi KunoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 385-396; DOI: https://doi.org/10.1124/jpet.120.000096
Kurokawa, Junko
- You have accessOpening of Intermediate Conductance Ca2+-Activated K+ Channels in C2C12 Skeletal Muscle Cells Increases the Myotube Diameter via the Akt/Mammalian Target of Rapamycin PathwayYuzo Iseki, Yuko Ono, Chihiro Hibi, Shoko Tanaka, Shunya Takeshita, Yuko Maejima, Junko Kurokawa, Masahiro Murakawa, Kenju Shimomura and Kazuho SakamotoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 454-462; DOI: https://doi.org/10.1124/jpet.120.000290
L
Legakis, L.P.
- You have accessManipulating Pharmacodynamic Efficacy with Agonist + Antagonist Mixtures: In Vitro and In Vivo Studies with Opioids and CannabinoidsD.E. Selley, M.L. Banks, C.M. Diester, A.M. Jali, L.P. Legakis, E.J. Santos and S.S. NegusJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 374-384; DOI: https://doi.org/10.1124/jpet.120.000349
León, Francisco
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Li, Yao
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
Liang, Yong
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
Liu, Han
- You have accessRNA Interference Targeting Liver Angiopoietin-Like Protein 3 Protects from Nephrotic Syndrome in a Rat Model Via Amelioration of Pathologic HypertriglyceridemiaYitong Zhao, Masaki Goto, Nosratola D. Vaziri, Mahyar Khazaeli, Han Liu, Nazli Farahanchi, Elham Khanifar, Ted Farzaneh, Patrick A. Haslett, Hamid Moradi and Mangala M. SoundarapandianJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 428-435; DOI: https://doi.org/10.1124/jpet.120.000257
Lopera-Londoño, Carolina
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Lőrincz, István
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Lowe, Val J.
- You have accessDistinct Uptake Kinetics of Alzheimer Disease Amyloid-β 40 and 42 at the Blood-Brain Barrier EndotheliumNidhi Sharda, Kristen M. Ahlschwede, Geoffry L. Curran, Val J. Lowe and Karunya K. KandimallaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 482-490; DOI: https://doi.org/10.1124/jpet.120.000086
M
Maejima, Yasuhiro
- You have accessβ3-Adrenergic Receptor Agonist Prevents Diastolic Dysfunction in an Angiotensin II–Induced Cardiomyopathy Mouse ModelMasataka Kamiya, Kuniya Asai, Yasuhiro Maejima, Akihiro Shirakabe, Koji Murai, Satsuki Noma, Hidenori Komiyama, Naoki Sato, Kyoichi Mizuno and Wataru ShimizuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 473-481; DOI: https://doi.org/10.1124/jpet.120.000140
Maejima, Yuko
- You have accessOpening of Intermediate Conductance Ca2+-Activated K+ Channels in C2C12 Skeletal Muscle Cells Increases the Myotube Diameter via the Akt/Mammalian Target of Rapamycin PathwayYuzo Iseki, Yuko Ono, Chihiro Hibi, Shoko Tanaka, Shunya Takeshita, Yuko Maejima, Junko Kurokawa, Masahiro Murakawa, Kenju Shimomura and Kazuho SakamotoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 454-462; DOI: https://doi.org/10.1124/jpet.120.000290
Málnási-Csizmadia, András
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
McCurdy, Christopher R.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
McMahon, Lance R.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Mizuno, Kyoichi
- You have accessβ3-Adrenergic Receptor Agonist Prevents Diastolic Dysfunction in an Angiotensin II–Induced Cardiomyopathy Mouse ModelMasataka Kamiya, Kuniya Asai, Yasuhiro Maejima, Akihiro Shirakabe, Koji Murai, Satsuki Noma, Hidenori Komiyama, Naoki Sato, Kyoichi Mizuno and Wataru ShimizuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 473-481; DOI: https://doi.org/10.1124/jpet.120.000140
Monostory, Katalin
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Moradi, Hamid
- You have accessRNA Interference Targeting Liver Angiopoietin-Like Protein 3 Protects from Nephrotic Syndrome in a Rat Model Via Amelioration of Pathologic HypertriglyceridemiaYitong Zhao, Masaki Goto, Nosratola D. Vaziri, Mahyar Khazaeli, Han Liu, Nazli Farahanchi, Elham Khanifar, Ted Farzaneh, Patrick A. Haslett, Hamid Moradi and Mangala M. SoundarapandianJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 428-435; DOI: https://doi.org/10.1124/jpet.120.000257
Morin, Didier
- You have accessA Phenyl-Pyrrolidine Derivative Reveals a Dual Inhibition Mechanism of Myocardial Mitochondrial Permeability Transition Pore, Which Is Limited by Its Myocardial DistributionMathieu Panel, Abdelhakim Ahmed-Belkacem, Isaac Ruiz, Jean-François Guichou, Jean-Michel Pawlotsky, Bijan Ghaleh and Didier MorinJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 348-357; DOI: https://doi.org/10.1124/jpet.120.000359
Morse, Noune Tahmassian
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
Mottinelli, Marco
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Murai, Koji
- You have accessβ3-Adrenergic Receptor Agonist Prevents Diastolic Dysfunction in an Angiotensin II–Induced Cardiomyopathy Mouse ModelMasataka Kamiya, Kuniya Asai, Yasuhiro Maejima, Akihiro Shirakabe, Koji Murai, Satsuki Noma, Hidenori Komiyama, Naoki Sato, Kyoichi Mizuno and Wataru ShimizuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 473-481; DOI: https://doi.org/10.1124/jpet.120.000140
Murakawa, Masahiro
- You have accessOpening of Intermediate Conductance Ca2+-Activated K+ Channels in C2C12 Skeletal Muscle Cells Increases the Myotube Diameter via the Akt/Mammalian Target of Rapamycin PathwayYuzo Iseki, Yuko Ono, Chihiro Hibi, Shoko Tanaka, Shunya Takeshita, Yuko Maejima, Junko Kurokawa, Masahiro Murakawa, Kenju Shimomura and Kazuho SakamotoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 454-462; DOI: https://doi.org/10.1124/jpet.120.000290
Musil, Djordje
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
N
Nag, Suman
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Negus, S.S.
- You have accessManipulating Pharmacodynamic Efficacy with Agonist + Antagonist Mixtures: In Vitro and In Vivo Studies with Opioids and CannabinoidsD.E. Selley, M.L. Banks, C.M. Diester, A.M. Jali, L.P. Legakis, E.J. Santos and S.S. NegusJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 374-384; DOI: https://doi.org/10.1124/jpet.120.000349
Ni, Jia
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
Nojima, Iyori
- You have accessDifferent Antioxidative and Antiapoptotic Effects of Piceatannol and ResveratrolRyusuke Hosoda, Hiroki Hamada, Daisuke Uesugi, Naotoshi Iwahara, Iyori Nojima, Yoshiyuki Horio and Atsushi KunoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 385-396; DOI: https://doi.org/10.1124/jpet.120.000096
Noma, Satsuki
- You have accessβ3-Adrenergic Receptor Agonist Prevents Diastolic Dysfunction in an Angiotensin II–Induced Cardiomyopathy Mouse ModelMasataka Kamiya, Kuniya Asai, Yasuhiro Maejima, Akihiro Shirakabe, Koji Murai, Satsuki Noma, Hidenori Komiyama, Naoki Sato, Kyoichi Mizuno and Wataru ShimizuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 473-481; DOI: https://doi.org/10.1124/jpet.120.000140
O
Obeng, Samuel
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Okitsu, Shinji L.
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
Ono, Yuko
- You have accessOpening of Intermediate Conductance Ca2+-Activated K+ Channels in C2C12 Skeletal Muscle Cells Increases the Myotube Diameter via the Akt/Mammalian Target of Rapamycin PathwayYuzo Iseki, Yuko Ono, Chihiro Hibi, Shoko Tanaka, Shunya Takeshita, Yuko Maejima, Junko Kurokawa, Masahiro Murakawa, Kenju Shimomura and Kazuho SakamotoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 454-462; DOI: https://doi.org/10.1124/jpet.120.000290
Oravecz, Kinga
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
P
Pallares, Victoria L.C.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Panel, Mathieu
- You have accessA Phenyl-Pyrrolidine Derivative Reveals a Dual Inhibition Mechanism of Myocardial Mitochondrial Permeability Transition Pore, Which Is Limited by Its Myocardial DistributionMathieu Panel, Abdelhakim Ahmed-Belkacem, Isaac Ruiz, Jean-François Guichou, Jean-Michel Pawlotsky, Bijan Ghaleh and Didier MorinJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 348-357; DOI: https://doi.org/10.1124/jpet.120.000359
Patel, Avi
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Patterson, Jaclyn
- You have accessIdentification of a Human Whole Blood–Based Endothelial Cell Impedance Assay for Assessing Clinical Transient Receptor Potential Vanilloid 4 Target Engagement Ex VivoXiaoping Xu, Navin Goyal, Melissa H. Costell, Theresa Roethke, Christian H. James, Kevin S. Thorneloe, Jaclyn Patterson, Patrick Stoy, Krista Goodman, Dennis L. Sprecher and David J. BehmJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 436-443; DOI: https://doi.org/10.1124/jpet.120.000307
Pawlotsky, Jean-Michel
- You have accessA Phenyl-Pyrrolidine Derivative Reveals a Dual Inhibition Mechanism of Myocardial Mitochondrial Permeability Transition Pore, Which Is Limited by Its Myocardial DistributionMathieu Panel, Abdelhakim Ahmed-Belkacem, Isaac Ruiz, Jean-François Guichou, Jean-Michel Pawlotsky, Bijan Ghaleh and Didier MorinJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 348-357; DOI: https://doi.org/10.1124/jpet.120.000359
Pennington, Anna E.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Pereira, Albertina
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
Przetak, Melinda
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
Q
Qian, Meilin
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
R
Rauscher, Anna Á.
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Reeves, Morgan E.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Reissig, Sonja
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
Restrepo, Luis F.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Roethke, Theresa
- You have accessIdentification of a Human Whole Blood–Based Endothelial Cell Impedance Assay for Assessing Clinical Transient Receptor Potential Vanilloid 4 Target Engagement Ex VivoXiaoping Xu, Navin Goyal, Melissa H. Costell, Theresa Roethke, Christian H. James, Kevin S. Thorneloe, Jaclyn Patterson, Patrick Stoy, Krista Goodman, Dennis L. Sprecher and David J. BehmJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 436-443; DOI: https://doi.org/10.1124/jpet.120.000307
Ruiz, Isaac
- You have accessA Phenyl-Pyrrolidine Derivative Reveals a Dual Inhibition Mechanism of Myocardial Mitochondrial Permeability Transition Pore, Which Is Limited by Its Myocardial DistributionMathieu Panel, Abdelhakim Ahmed-Belkacem, Isaac Ruiz, Jean-François Guichou, Jean-Michel Pawlotsky, Bijan Ghaleh and Didier MorinJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 348-357; DOI: https://doi.org/10.1124/jpet.120.000359
S
Sakamoto, Kazuho
- You have accessOpening of Intermediate Conductance Ca2+-Activated K+ Channels in C2C12 Skeletal Muscle Cells Increases the Myotube Diameter via the Akt/Mammalian Target of Rapamycin PathwayYuzo Iseki, Yuko Ono, Chihiro Hibi, Shoko Tanaka, Shunya Takeshita, Yuko Maejima, Junko Kurokawa, Masahiro Murakawa, Kenju Shimomura and Kazuho SakamotoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 454-462; DOI: https://doi.org/10.1124/jpet.120.000290
Santos, E.J.
- You have accessManipulating Pharmacodynamic Efficacy with Agonist + Antagonist Mixtures: In Vitro and In Vivo Studies with Opioids and CannabinoidsD.E. Selley, M.L. Banks, C.M. Diester, A.M. Jali, L.P. Legakis, E.J. Santos and S.S. NegusJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 374-384; DOI: https://doi.org/10.1124/jpet.120.000349
Sato, Naoki
- You have accessβ3-Adrenergic Receptor Agonist Prevents Diastolic Dysfunction in an Angiotensin II–Induced Cardiomyopathy Mouse ModelMasataka Kamiya, Kuniya Asai, Yasuhiro Maejima, Akihiro Shirakabe, Koji Murai, Satsuki Noma, Hidenori Komiyama, Naoki Sato, Kyoichi Mizuno and Wataru ShimizuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 473-481; DOI: https://doi.org/10.1124/jpet.120.000140
Schuler, Franz
- You have accessCalculation of an Apical Efflux Ratio from P-Glycoprotein (P-gp) In Vitro Transport Experiments Shows an Improved Correlation with In Vivo Cerebrospinal Fluid Measurements in Rats: Impact on P-gp Screening and Compound OptimizationHolger Fischer, Claudia Senn, Mohammed Ullah, Carina Cantrill, Franz Schuler and Li YuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 322-329; DOI: https://doi.org/10.1124/jpet.120.000158
Selley, D.E.
- You have accessManipulating Pharmacodynamic Efficacy with Agonist + Antagonist Mixtures: In Vitro and In Vivo Studies with Opioids and CannabinoidsD.E. Selley, M.L. Banks, C.M. Diester, A.M. Jali, L.P. Legakis, E.J. Santos and S.S. NegusJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 374-384; DOI: https://doi.org/10.1124/jpet.120.000349
Senn, Claudia
- You have accessCalculation of an Apical Efflux Ratio from P-Glycoprotein (P-gp) In Vitro Transport Experiments Shows an Improved Correlation with In Vivo Cerebrospinal Fluid Measurements in Rats: Impact on P-gp Screening and Compound OptimizationHolger Fischer, Claudia Senn, Mohammed Ullah, Carina Cantrill, Franz Schuler and Li YuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 322-329; DOI: https://doi.org/10.1124/jpet.120.000158
Sentir, Alena M.
- You have accessSelf-Administration of Cotinine in Wistar Rats: Comparisons to NicotineZheng-Ming Ding, Yong Gao, Alena M. Sentir and Xiaoying TanJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 338-347; DOI: https://doi.org/10.1124/jpet.120.000367
Sharda, Nidhi
- You have accessDistinct Uptake Kinetics of Alzheimer Disease Amyloid-β 40 and 42 at the Blood-Brain Barrier EndotheliumNidhi Sharda, Kristen M. Ahlschwede, Geoffry L. Curran, Val J. Lowe and Karunya K. KandimallaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 482-490; DOI: https://doi.org/10.1124/jpet.120.000086
Sherer, Brian
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
Shi, Zongjun
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
Shimizu, Wataru
- You have accessβ3-Adrenergic Receptor Agonist Prevents Diastolic Dysfunction in an Angiotensin II–Induced Cardiomyopathy Mouse ModelMasataka Kamiya, Kuniya Asai, Yasuhiro Maejima, Akihiro Shirakabe, Koji Murai, Satsuki Noma, Hidenori Komiyama, Naoki Sato, Kyoichi Mizuno and Wataru ShimizuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 473-481; DOI: https://doi.org/10.1124/jpet.120.000140
Shimomura, Kenju
- You have accessOpening of Intermediate Conductance Ca2+-Activated K+ Channels in C2C12 Skeletal Muscle Cells Increases the Myotube Diameter via the Akt/Mammalian Target of Rapamycin PathwayYuzo Iseki, Yuko Ono, Chihiro Hibi, Shoko Tanaka, Shunya Takeshita, Yuko Maejima, Junko Kurokawa, Masahiro Murakawa, Kenju Shimomura and Kazuho SakamotoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 454-462; DOI: https://doi.org/10.1124/jpet.120.000290
Shirakabe, Akihiro
- You have accessβ3-Adrenergic Receptor Agonist Prevents Diastolic Dysfunction in an Angiotensin II–Induced Cardiomyopathy Mouse ModelMasataka Kamiya, Kuniya Asai, Yasuhiro Maejima, Akihiro Shirakabe, Koji Murai, Satsuki Noma, Hidenori Komiyama, Naoki Sato, Kyoichi Mizuno and Wataru ShimizuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 473-481; DOI: https://doi.org/10.1124/jpet.120.000140
Soundarapandian, Mangala M.
- You have accessRNA Interference Targeting Liver Angiopoietin-Like Protein 3 Protects from Nephrotic Syndrome in a Rat Model Via Amelioration of Pathologic HypertriglyceridemiaYitong Zhao, Masaki Goto, Nosratola D. Vaziri, Mahyar Khazaeli, Han Liu, Nazli Farahanchi, Elham Khanifar, Ted Farzaneh, Patrick A. Haslett, Hamid Moradi and Mangala M. SoundarapandianJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 428-435; DOI: https://doi.org/10.1124/jpet.120.000257
Sprecher, Dennis L.
- You have accessIdentification of a Human Whole Blood–Based Endothelial Cell Impedance Assay for Assessing Clinical Transient Receptor Potential Vanilloid 4 Target Engagement Ex VivoXiaoping Xu, Navin Goyal, Melissa H. Costell, Theresa Roethke, Christian H. James, Kevin S. Thorneloe, Jaclyn Patterson, Patrick Stoy, Krista Goodman, Dennis L. Sprecher and David J. BehmJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 436-443; DOI: https://doi.org/10.1124/jpet.120.000307
Stoy, Patrick
- You have accessIdentification of a Human Whole Blood–Based Endothelial Cell Impedance Assay for Assessing Clinical Transient Receptor Potential Vanilloid 4 Target Engagement Ex VivoXiaoping Xu, Navin Goyal, Melissa H. Costell, Theresa Roethke, Christian H. James, Kevin S. Thorneloe, Jaclyn Patterson, Patrick Stoy, Krista Goodman, Dennis L. Sprecher and David J. BehmJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 436-443; DOI: https://doi.org/10.1124/jpet.120.000307
Sun, Jia’ao
- You have accessPhytochemical Regulation of RNA in Treating Inflammatory Bowel Disease and Colon Cancer: Inspirations from Cell and Animal StudiesGuolin Zhang, Chi Zhang, Jia’ao Sun, Yongjian Xiong, Liang Wang and Dapeng ChenJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 464-472; DOI: https://doi.org/10.1124/jpet.120.000354
Suthar, Sharad Kumar
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Szabó, Pál Tamás
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
T
Takeshita, Shunya
- You have accessOpening of Intermediate Conductance Ca2+-Activated K+ Channels in C2C12 Skeletal Muscle Cells Increases the Myotube Diameter via the Akt/Mammalian Target of Rapamycin PathwayYuzo Iseki, Yuko Ono, Chihiro Hibi, Shoko Tanaka, Shunya Takeshita, Yuko Maejima, Junko Kurokawa, Masahiro Murakawa, Kenju Shimomura and Kazuho SakamotoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 454-462; DOI: https://doi.org/10.1124/jpet.120.000290
Tan, Bowei
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
Tan, Xiaoying
- You have accessSelf-Administration of Cotinine in Wistar Rats: Comparisons to NicotineZheng-Ming Ding, Yong Gao, Alena M. Sentir and Xiaoying TanJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 338-347; DOI: https://doi.org/10.1124/jpet.120.000367
Tanaka, Shoko
- You have accessOpening of Intermediate Conductance Ca2+-Activated K+ Channels in C2C12 Skeletal Muscle Cells Increases the Myotube Diameter via the Akt/Mammalian Target of Rapamycin PathwayYuzo Iseki, Yuko Ono, Chihiro Hibi, Shoko Tanaka, Shunya Takeshita, Yuko Maejima, Junko Kurokawa, Masahiro Murakawa, Kenju Shimomura and Kazuho SakamotoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 454-462; DOI: https://doi.org/10.1124/jpet.120.000290
Taylor, Victoria A.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Thorneloe, Kevin S.
- You have accessIdentification of a Human Whole Blood–Based Endothelial Cell Impedance Assay for Assessing Clinical Transient Receptor Potential Vanilloid 4 Target Engagement Ex VivoXiaoping Xu, Navin Goyal, Melissa H. Costell, Theresa Roethke, Christian H. James, Kevin S. Thorneloe, Jaclyn Patterson, Patrick Stoy, Krista Goodman, Dennis L. Sprecher and David J. BehmJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 436-443; DOI: https://doi.org/10.1124/jpet.120.000307
Tierney, Patrick J.
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Tomasic, Ivan
- Open AccessImproved Inhibitory and Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) Properties of Blebbistatin Derivatives Indicate That Blebbistatin Scaffold Is Ideal for drug Development Targeting Myosin-2Máté Gyimesi, Anna Á. Rauscher, Sharad Kumar Suthar, Kamirán Á. Hamow, Kinga Oravecz, István Lőrincz, Zsolt Borhegyi, Máté T. Déri, Ádám F. Kiss, Katalin Monostory, Pál Tamás Szabó, Suman Nag, Ivan Tomasic, Jacob Krans, Patrick J. Tierney, Mihály Kovács, László Kornya and András Málnási-CsizmadiaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 358-373; DOI: https://doi.org/10.1124/jpet.120.000167
Tzvetkov, Evgeni
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
U
Uesugi, Daisuke
- You have accessDifferent Antioxidative and Antiapoptotic Effects of Piceatannol and ResveratrolRyusuke Hosoda, Hiroki Hamada, Daisuke Uesugi, Naotoshi Iwahara, Iyori Nojima, Yoshiyuki Horio and Atsushi KunoJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 385-396; DOI: https://doi.org/10.1124/jpet.120.000096
Ullah, Mohammed
- You have accessCalculation of an Apical Efflux Ratio from P-Glycoprotein (P-gp) In Vitro Transport Experiments Shows an Improved Correlation with In Vivo Cerebrospinal Fluid Measurements in Rats: Impact on P-gp Screening and Compound OptimizationHolger Fischer, Claudia Senn, Mohammed Ullah, Carina Cantrill, Franz Schuler and Li YuJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 322-329; DOI: https://doi.org/10.1124/jpet.120.000158
V
Vaziri, Nosratola D.
- You have accessRNA Interference Targeting Liver Angiopoietin-Like Protein 3 Protects from Nephrotic Syndrome in a Rat Model Via Amelioration of Pathologic HypertriglyceridemiaYitong Zhao, Masaki Goto, Nosratola D. Vaziri, Mahyar Khazaeli, Han Liu, Nazli Farahanchi, Elham Khanifar, Ted Farzaneh, Patrick A. Haslett, Hamid Moradi and Mangala M. SoundarapandianJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 428-435; DOI: https://doi.org/10.1124/jpet.120.000257
Vlach, Jaromir
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
W
Walsky, Robert L.
- Open AccessDiscovery of M5049: A Novel Selective Toll-Like Receptor 7/8 Inhibitor for Treatment of AutoimmunityJaromir Vlach, Andrew T. Bender, Melinda Przetak, Albertina Pereira, Aditee Deshpande, Theresa L. Johnson, Sonja Reissig, Evgeni Tzvetkov, Djordje Musil, Noune Tahmassian Morse, Philipp Haselmayer, Simone C. Zimmerli, Shinji L. Okitsu, Robert L. Walsky and Brian ShererJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 397-409; DOI: https://doi.org/10.1124/jpet.120.000275
Wang, Liang
- You have accessPhytochemical Regulation of RNA in Treating Inflammatory Bowel Disease and Colon Cancer: Inspirations from Cell and Animal StudiesGuolin Zhang, Chi Zhang, Jia’ao Sun, Yongjian Xiong, Liang Wang and Dapeng ChenJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 464-472; DOI: https://doi.org/10.1124/jpet.120.000354
Wilkerson, Jenny L.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
Williamson, Morgan R.
- You have accessPharmacological Comparison of Mitragynine and 7-Hydroxymitragynine: In Vitro Affinity and Efficacy for μ-Opioid Receptor and Opioid-Like Behavioral Effects in RatsSamuel Obeng, Jenny L. Wilkerson, Francisco León, Morgan E. Reeves, Luis F. Restrepo, Lea R. Gamez-Jimenez, Avi Patel, Anna E. Pennington, Victoria A. Taylor, Nicholas P. Ho, Tobias Braun, John D. Fortner, Morgan L. Crowley, Morgan R. Williamson, Victoria L.C. Pallares, Marco Mottinelli, Carolina Lopera-Londoño, Christopher R. McCurdy, Lance R. McMahon and Takato HiranitaJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 410-427; DOI: https://doi.org/10.1124/jpet.120.000189
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Xiong, Yongjian
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Xu, Xiaoping
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Ye, Fei
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
Yu, Li
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Yu, Xiaojuan
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
Z
Zhang, Chi
- You have accessPhytochemical Regulation of RNA in Treating Inflammatory Bowel Disease and Colon Cancer: Inspirations from Cell and Animal StudiesGuolin Zhang, Chi Zhang, Jia’ao Sun, Yongjian Xiong, Liang Wang and Dapeng ChenJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 464-472; DOI: https://doi.org/10.1124/jpet.120.000354
Zhang, Guolin
- You have accessPhytochemical Regulation of RNA in Treating Inflammatory Bowel Disease and Colon Cancer: Inspirations from Cell and Animal StudiesGuolin Zhang, Chi Zhang, Jia’ao Sun, Yongjian Xiong, Liang Wang and Dapeng ChenJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 464-472; DOI: https://doi.org/10.1124/jpet.120.000354
Zhao, Yitong
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Zheng, Xiaoxiao
- You have accessPharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α2δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic PainXiaoli Gou, Xiaojuan Yu, Dongdong Bai, Bowei Tan, Pingfeng Cao, Meilin Qian, Xiaoxiao Zheng, Lei Chen, Zongjun Shi, Yao Li, Fei Ye, Yong Liang and Jia NiJournal of Pharmacology and Experimental Therapeutics March 2021, 376 (3) 330-337; DOI: https://doi.org/10.1124/jpet.120.000315
Zimmerli, Simone C.
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