| | nM |
Bantag-1 | Boc-Phe-His-4-amino-5-cyclohexyl-2,4,5-trideoxypentonyl-Leu-(3-dimethylamino) benzylamide N-methylammonium trifluoroacetate | 0.40 ± 0.25 | 0.27 ± 0.01 |
1 | [D-Tyr6, β-Ala11, Phe13, Nle14]Bn-(6-14) | 1.58 ± 0.09 | 0.68 ± 0.02 |
2 | [D-Phe6, β-Ala11, Phe13, Nle14]Bn-(6-14) | 5.50 ± 0.29 | 7.94 ± 0.38 |
6 | [D-Tyr6(S), Apa11-4Cl, Phe13, Nle14]Bn-(6-14) | 110 ± 6 | 31.6 ± 0.6 |
7 | [D-Tyr6(R), Apa11-4Cl, Phe13, Nle14]Bn-(6-14) | 2.52 ± 0.13 | 2.04 ± 0.06 |
15 | [D-Tyr6(S), Apa11, Phe13, Nle14]Bn-(6-14) | 20.0 ± 1.1 | 31.5 ± 1.1 |
34 | Ac-Phe, Trp, Ala, His (t-Bzl), Nip, Gly,Arg-NH2 | 162 ± 8 | 74 ± 3 |
54 | H-D-Phe, Gln, D-Trp, Phe-NH2 | >1000 | >1000 |
68 | 3-phenyl-propionyl-Ala, D-Trp, NH (CH2) C6H5 | >1000 | 467 ± 11 |
NMB | Neuromedin B | >1000 | >1000 |
GRP | Gastrin-releasing peptide | >1000 | >1000 |