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Journal of Pharmacology and Experimental Therapeutics

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Table of Contents

July 01, 2017; Volume 362,Issue 1

Behavioral Pharmacology

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    σ Receptor Effects of N-Substituted Benztropine Analogs: Implications for Antagonism of Cocaine Self-Administration
    Takato Hiranita, Weimin C. Hong, Theresa Kopajtic and Jonathan L. Katz
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 2-13; DOI: https://doi.org/10.1124/jpet.117.241109
  • You have access
    Relief of Pain-Depressed Behavior in Rats by Activation of D1-Like Dopamine Receptors
    Matthew F. Lazenka, Kelen C. Freitas, Sydney Henck and S. Stevens Negus
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 14-23; DOI: https://doi.org/10.1124/jpet.117.240796
  • You have access
    Preference for an Opioid/Benzodiazepine Mixture over an Opioid Alone Using a Concurrent Choice Procedure in Rhesus Monkeys
    Peter F. Weed, Charles P. France and Lisa R. Gerak
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 59-66; DOI: https://doi.org/10.1124/jpet.117.240200
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    Effects of Acute and Chronic Treatments with Dopamine D2 and D3 Receptor Ligands on Cocaine versus Food Choice in Rats
    Morgane Thomsen, Andrew C. Barrett, Paul Butler, S. Stevens Negus and S. Barak Caine
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 161-176; DOI: https://doi.org/10.1124/jpet.117.241141
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    Apparent CB1 Receptor Rimonabant Affinity Estimates: Combination with THC and Synthetic Cannabinoids in the Mouse In Vivo Triad Model
    T. W. Grim, A. J. Morales, B. F. Thomas, J. L. Wiley, G. W. Endres, S. S. Negus and A. H. Lichtman
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 210-218; DOI: https://doi.org/10.1124/jpet.117.240192

Cardiovascular

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    Treatment with Standard and Low Dose of Conjugated Equine Estrogen Differentially Modulates Estrogen Receptor Expression and Response to Angiotensin II in Mesenteric Venular Bed of Surgically Postmenopausal Hypertensive Rats
    Priscila Xavier Araujo, Tiago Januário Costa, Cinthya Echem, Maria Aparecida de Oliveira, Rosangela Aparecida Santos-Eichler, Lucas Giglio Colli, Francesc Jiménez-Altayó, Elisabet Vila, Eliana Hiromi Akamine, Ana Paula Dantas, Graziela Scalianti Ceravolo and Maria Helena Catelli de Carvalho
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 98-107; DOI: https://doi.org/10.1124/jpet.117.240465
  • Open Access
    Selexipag Active Metabolite ACT-333679 Displays Strong Anticontractile and Antiremodeling Effects but Low β-Arrestin Recruitment and Desensitization Potential
    John Gatfield, Katalin Menyhart, Daniel Wanner, Carmela Gnerre, Lucile Monnier, Keith Morrison, Patrick Hess, Marc Iglarz, Martine Clozel and Oliver Nayler
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 186-199; DOI: https://doi.org/10.1124/jpet.116.239665

Cellular and Molecular

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    XE991 and Linopirdine Are State-Dependent Inhibitors for Kv7/KCNQ Channels that Favor Activated Single Subunits
    Derek L Greene, Seungwoo Kang and Naoto Hoshi
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 177-185; DOI: https://doi.org/10.1124/jpet.117.241679
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    Regulation of δ Opioid Receptor-Mediated Signaling and Antinociception in Peripheral Sensory Neurons by Arachidonic Acid–Dependent 12/15-Lipoxygenase Metabolites
    Laura C. Sullivan, Teresa A. Chavera, Xiaoli Gao, Miryam M. Pando and Kelly A. Berg
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 200-209; DOI: https://doi.org/10.1124/jpet.117.241604

Drug Discovery and Translational Medicine

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    Identification of 4-Aminopyrazolopyrimidine Metabolite That May Contribute to the Hypolipidemic Effects of LY2584702 in Long Evans Diet–Induced Obese Rats
    Thomas B. Estridge, Asim B. Dey, Charles Reidy, Xiaohong Yu, Yuke Zhang, Maryalice Hartley, Paul L. Milligan, Najia Jin, Mark C. Kowala, Jennifer K. Leohr, Adrian J. Fretland, Thomas E. Mabry, Debra Luffer-Atlas and M. Jane Luo
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 108-118; DOI: https://doi.org/10.1124/jpet.117.240242
  • Rational Tuning of Visual Cycle Modulator Pharmacodynamics
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    Rational Tuning of Visual Cycle Modulator Pharmacodynamics
    Philip D. Kiser, Jianye Zhang, Mohsen Badiee, Junzo Kinoshita, Neal S. Peachey, Gregory P. Tochtrop and Krzysztof Palczewski
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 131-145; DOI: https://doi.org/10.1124/jpet.117.240721

Endocrine and Diabetes

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    The Dual Amylin- and Calcitonin-Receptor Agonist KBP-042 Works as Adjunct to Metformin on Fasting Hyperglycemia and HbA1c in a Rat Model of Type 2 Diabetes
    Sara T. Hjuler, Sofie Gydesen, Kim V. Andreassen, Morten A. Karsdal and Kim Henriksen
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 24-30; DOI: https://doi.org/10.1124/jpet.117.241281
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    LX2761, a Sodium/Glucose Cotransporter 1 Inhibitor Restricted to the Intestine, Improves Glycemic Control in Mice
    David R. Powell, Melinda G. Smith, Deon D. Doree, Angela L. Harris, Jennifer Greer, Christopher M. DaCosta, Andrea Thompson, Sabrina Jeter-Jones, Wendy Xiong, Kenneth G. Carson, Nicole C. Goodwin, Bryce A. Harrison, David B. Rawlins, Eric D. Strobel, Suma Gopinathan, Alan Wilson, Faika Mseeh, Brian Zambrowicz and Zhi-Ming Ding
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 85-97; DOI: https://doi.org/10.1124/jpet.117.240820

Gastrointestinal, Hepatic, Pulmonary, and Renal

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    Glutamatergic Mechanisms Involved in Bladder Overactivity and Pudendal Neuromodulation in Cats
    Jamie Uy, Michelle Yu, Xuewen Jiang, Cameron Jones, Bing Shen, Jicheng Wang, James R. Roppolo, William C. de Groat and Changfeng Tai
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 53-58; DOI: https://doi.org/10.1124/jpet.117.240895
  • Open Access
    Mashiningan Improves Opioid-Induced Constipation in Rats by Activating Cystic Fibrosis Transmembrane Conductance Regulator Chloride Channel
    Yumi Harada, Seiichi Iizuka, Yayoi Saegusa, Sachiko Mogami, Naoki Fujitsuka and Tomohisa Hattori
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 78-84; DOI: https://doi.org/10.1124/jpet.117.240630

Neuropharmacology

  • Open Access
    Pharmacological and Toxicological Properties of the Potent Oral γ-Secretase Modulator BPN-15606
    Steven L. Wagner, Kevin D. Rynearson, Steven K. Duddy, Can Zhang, Phuong D. Nguyen, Ann Becker, Uyen Vo, Deborah Masliah, Louise Monte, Justin B. Klee, Corinne M. Echmalian, Weiming Xia, Luisa Quinti, Graham Johnson, Jiunn H. Lin, Doo Y. Kim, William C. Mobley, Robert A. Rissman and Rudolph E. Tanzi
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 31-44; DOI: https://doi.org/10.1124/jpet.117.240861
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    Ethanol Reversal of Tolerance to the Antinociceptive Effects of Oxycodone and Hydrocodone
    Joanna C. Jacob, Justin L. Poklis, Hamid I. Akbarali, Graeme Henderson and William L. Dewey
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 45-52; DOI: https://doi.org/10.1124/jpet.117.241083
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    Novel Phosphodiesterase 4 Inhibitor FCPR03 Alleviates Lipopolysaccharide-Induced Neuroinflammation by Regulation of the cAMP/PKA/CREB Signaling Pathway and NF-κB Inhibition
    Zheng-Qiang Zou, Jia-Jia Chen, Hong-Fang Feng, Yu-Fang Cheng, Hai-Tao Wang, Zhong-Zhen Zhou, Hai-Biao Guo, Wenhua Zheng and Jiang-Ping Xu
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 67-77; DOI: https://doi.org/10.1124/jpet.116.239608
  • Open Access
    Glutaminyl Cyclase Inhibitor PQ912 Improves Cognition in Mouse Models of Alzheimer’s Disease—Studies on Relation to Effective Target Occupancy
    Torsten Hoffmann, Antje Meyer, Ulrich Heiser, Stephan Kurat, Livia Böhme, Martin Kleinschmidt, Karl-Ulrich Bühring, Birgit Hutter-Paier, Martina Farcher, Hans-Ulrich Demuth, Inge Lues and Stephan Schilling
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 119-130; DOI: https://doi.org/10.1124/jpet.117.240614
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    Pharmacologic Characterization of AMG8379, a Potent and Selective Small Molecule Sulfonamide Antagonist of the Voltage-Gated Sodium Channel NaV1.7
    Thomas J. Kornecook, Ruoyuan Yin, Stephen Altmann, Xuhai Be, Virginia Berry, Christopher P. Ilch, Michael Jarosh, Danielle Johnson, Josie H. Lee, Sonya G. Lehto, Joseph Ligutti, Dong Liu, Jason Luther, David Matson, Danny Ortuno, John Roberts, Kristin Taborn, Jinti Wang, Matthew M. Weiss, Violeta Yu, Dawn X. D. Zhu, Robert T. Fremeau and Bryan D. Moyer
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 146-160; DOI: https://doi.org/10.1124/jpet.116.239590

Erratum

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    Correction to “Antidepressant Potential of (R)-Ketamine in Rodent Models: Comparison with (S)-Ketamine”
    Journal of Pharmacology and Experimental Therapeutics July 2017, 362 (1) 1; DOI: https://doi.org/10.1124/jpet.116.239228err
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In this issue

Journal of Pharmacology and Experimental Therapeutics: 362 (1)
Journal of Pharmacology and Experimental Therapeutics
Vol. 362, Issue 1
1 Jul 2017
  • Table of Contents
  • Table of Contents (PDF)
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  • Editorial Board (PDF)
  • Front Matter (PDF)
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  • Behavioral Pharmacology
  • Cardiovascular
  • Cellular and Molecular
  • Drug Discovery and Translational Medicine
  • Endocrine and Diabetes
  • Gastrointestinal, Hepatic, Pulmonary, and Renal
  • Neuropharmacology
  • Erratum
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  • Interindividual variations in human liver cytochrome P-450 enzymes involved in the oxidation of drugs, carcinogens and toxic chemicals: studies with liver microsomes of 30 Japanese and 30 Caucasians.
  • Functional Selectivity and Classical Concepts of Quantitative Pharmacology
  • Abl Protein-Tyrosine Kinase Inhibitor STI571 Inhibits In Vitro Signal Transduction Mediated by c-Kit and Platelet-Derived Growth Factor Receptors
  • The Prediction of Human Pharmacokinetic Parameters from Preclinical and In Vitro Metabolism Data
  • A METHOD FOR DETERMINING LOSS OF PAIN SENSATION
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