Index by author
October 01, 2016; Volume 359,Issue 1
A
Aaltonen, Niina
- You have accessIn Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor {4-[bis-(benzo[d][1,3]dioxol-5-yl)methyl]-piperidin-1-yl}(1H-1,2,4-triazol-1-yl)methanone (JJKK-048)Niina Aaltonen, Ewa Kedzierska, Jolanta Orzelska-Górka, Marko Lehtonen, Dina Navia-Paldanius, Hermina Jakupovic, Juha R. Savinainen, Tapio Nevalainen, Jarmo T. Laitinen, Teija Parkkari and Mikko GyntherJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 62-72; DOI: https://doi.org/10.1124/jpet.116.233114
Abagyan, Ruben
- You have accessMolecular Properties of Drugs Interacting with SLC22 Transporters OAT1, OAT3, OCT1, and OCT2: A Machine-Learning ApproachHenry C. Liu, Anne Goldenberg, Yuchen Chen, Christina Lun, Wei Wu, Kevin T. Bush, Natasha Balac, Paul Rodriguez, Ruben Abagyan and Sanjay K. NigamJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 215-229; DOI: https://doi.org/10.1124/jpet.116.232660
Abbott, Megan
- You have accessDiscriminative Stimulus Effects of Binary Drug Mixtures: Studies with Cocaine, MDPV, and CaffeineGregory T. Collins, Megan Abbott, Kayla Galindo, Elise L. Rush, Kenner C. Rice and Charles P. FranceJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 1-10; DOI: https://doi.org/10.1124/jpet.116.234252
Adili, Reheman
- You have accessDevelopment of Poly Unsaturated Fatty Acid Derivatives of Aspirin for Inhibition of Platelet FunctionJahnabi Roy, Reheman Adili, Richard Kulmacz, Michael Holinstat and Aditi DasJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 134-141; DOI: https://doi.org/10.1124/jpet.116.234781
Ai, Jing
- You have accessThe Marine-Derived Oligosaccharide Sulfate MS80, a Novel Transforming Growth Factor β1 Inhibitor, Reverses Epithelial Mesenchymal Transition Induced by Transforming Growth Factor-β1 and Suppresses Tumor MetastasisJi Zhou, Wenjie You, Guangqiang Sun, Yixuan Li, Bi Chen, Jing Ai and Handong JiangJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 54-61; DOI: https://doi.org/10.1124/jpet.116.234799
Al-Khrasani, Mahmoud
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Alonso-Galicia, Magdalena
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Alston, Laurie
- You have accessPregnane X Receptor Activation Attenuates Inflammation-Associated Intestinal Epithelial Barrier Dysfunction by Inhibiting Cytokine-Induced Myosin Light-Chain Kinase Expression and c-Jun N-Terminal Kinase 1/2 ActivationAditya Garg, Angela Zhao, Sarah L. Erickson, Subhajit Mukherjee, Aik Jiang Lau, Laurie Alston, Thomas K. H. Chang, Sridhar Mani and Simon A. HirotaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 91-101; DOI: https://doi.org/10.1124/jpet.116.234096
B
Balac, Natasha
- You have accessMolecular Properties of Drugs Interacting with SLC22 Transporters OAT1, OAT3, OCT1, and OCT2: A Machine-Learning ApproachHenry C. Liu, Anne Goldenberg, Yuchen Chen, Christina Lun, Wei Wu, Kevin T. Bush, Natasha Balac, Paul Rodriguez, Ruben Abagyan and Sanjay K. NigamJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 215-229; DOI: https://doi.org/10.1124/jpet.116.232660
Balogh, Mihály
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Banfor, Patricia
- You have accessSphingosine-1-Phosphate (S1P) Lyase Inhibition Causes Increased Cardiac S1P Levels and Bradycardia in RatsChristopher M. Harris, Scott Mittelstadt, Patricia Banfor, Peter Bousquet, David B. Duignan, Gary Gintant, Michelle Hart, Youngjae Kim and Jason SegretiJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 151-158; DOI: https://doi.org/10.1124/jpet.116.235002
Benetti, Elisa
- You have accessEmpagliflozin Protects against Diet-Induced NLRP-3 Inflammasome Activation and Lipid AccumulationElisa Benetti, Raffaella Mastrocola, Giovanna Vitarelli, Juan Carlos Cutrin, Debora Nigro, Fausto Chiazza, Eric Mayoux, Massimo Collino and Roberto FantozziJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 45-53; DOI: https://doi.org/10.1124/jpet.116.235069
Bousquet, Peter
- You have accessSphingosine-1-Phosphate (S1P) Lyase Inhibition Causes Increased Cardiac S1P Levels and Bradycardia in RatsChristopher M. Harris, Scott Mittelstadt, Patricia Banfor, Peter Bousquet, David B. Duignan, Gary Gintant, Michelle Hart, Youngjae Kim and Jason SegretiJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 151-158; DOI: https://doi.org/10.1124/jpet.116.235002
Brodeur, Scott R.
- You have accessUnexpected Potency Differences between B-Cell–Activating Factor (BAFF) Antagonist Antibodies against Various Forms of BAFF: Trimer, 60-Mer, and Membrane-BoundAmy M. Nicoletti, Cynthia Hess Kenny, Ashraf M. Khalil, Qi Pan, Kerry L. M. Ralph, Julie Ritchie, Sathyadevi Venkataramani, David H. Presky, Scott M. DeWire and Scott R. BrodeurJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 37-44; DOI: https://doi.org/10.1124/jpet.116.236075
Brown, Nicholas F.
- You have accessSelectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman PrimatesSteven M. Weldon, Matthew A. Cerny, Kristina Gueneva-Boucheva, Derek Cogan, Xin Guo, Neil Moss, Jean-Hugues Parmentier, Jeremy R. Richman, Glenn A. Reinhart and Nicholas F. BrownJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 142-150; DOI: https://doi.org/10.1124/jpet.116.236463
Bui, Hai H.
- You have accessPharmacological Characterization of a Potent Inhibitor of Autotaxin in Animal Models of Inflammatory Bowel Disease and Multiple SclerosisKannan Thirunavukkarasu, Bailin Tan, Craig A. Swearingen, Guilherme Rocha, Hai H. Bui, Denis J. McCann, Spencer B. Jones, Bryan H. Norman, Lance A. Pfeifer and Joy K. SahaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 207-214; DOI: https://doi.org/10.1124/jpet.116.234013
Bush, Kevin T.
- You have accessMolecular Properties of Drugs Interacting with SLC22 Transporters OAT1, OAT3, OCT1, and OCT2: A Machine-Learning ApproachHenry C. Liu, Anne Goldenberg, Yuchen Chen, Christina Lun, Wei Wu, Kevin T. Bush, Natasha Balac, Paul Rodriguez, Ruben Abagyan and Sanjay K. NigamJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 215-229; DOI: https://doi.org/10.1124/jpet.116.232660
C
Can, Adem
- You have accessEffects of Ketamine and Ketamine Metabolites on Evoked Striatal Dopamine Release, Dopamine Receptors, and Monoamine TransportersAdem Can, Panos Zanos, Ruin Moaddel, Hye Jin Kang, Katinia S. S. Dossou, Irving W. Wainer, Joseph F. Cheer, Douglas O. Frost, Xi-Ping Huang and Todd D. GouldJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 159-170; DOI: https://doi.org/10.1124/jpet.116.235838
Cerny, Matthew A.
- You have accessSelectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman PrimatesSteven M. Weldon, Matthew A. Cerny, Kristina Gueneva-Boucheva, Derek Cogan, Xin Guo, Neil Moss, Jean-Hugues Parmentier, Jeremy R. Richman, Glenn A. Reinhart and Nicholas F. BrownJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 142-150; DOI: https://doi.org/10.1124/jpet.116.236463
Chang, Thomas K. H.
- You have accessPregnane X Receptor Activation Attenuates Inflammation-Associated Intestinal Epithelial Barrier Dysfunction by Inhibiting Cytokine-Induced Myosin Light-Chain Kinase Expression and c-Jun N-Terminal Kinase 1/2 ActivationAditya Garg, Angela Zhao, Sarah L. Erickson, Subhajit Mukherjee, Aik Jiang Lau, Laurie Alston, Thomas K. H. Chang, Sridhar Mani and Simon A. HirotaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 91-101; DOI: https://doi.org/10.1124/jpet.116.234096
Cheer, Joseph F.
- You have accessEffects of Ketamine and Ketamine Metabolites on Evoked Striatal Dopamine Release, Dopamine Receptors, and Monoamine TransportersAdem Can, Panos Zanos, Ruin Moaddel, Hye Jin Kang, Katinia S. S. Dossou, Irving W. Wainer, Joseph F. Cheer, Douglas O. Frost, Xi-Ping Huang and Todd D. GouldJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 159-170; DOI: https://doi.org/10.1124/jpet.116.235838
Chen, Bi
- You have accessThe Marine-Derived Oligosaccharide Sulfate MS80, a Novel Transforming Growth Factor β1 Inhibitor, Reverses Epithelial Mesenchymal Transition Induced by Transforming Growth Factor-β1 and Suppresses Tumor MetastasisJi Zhou, Wenjie You, Guangqiang Sun, Yixuan Li, Bi Chen, Jing Ai and Handong JiangJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 54-61; DOI: https://doi.org/10.1124/jpet.116.234799
Chen, Gang
- You have accessRegulation of UGT2B Expression and Activity by miR-216b-5p in Liver Cancer Cell LinesDouglas F. Dluzen, Aimee K. Sutliff, Gang Chen, Christy J. W. Watson, Faoud T. Ishmael and Philip LazarusJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 182-193; DOI: https://doi.org/10.1124/jpet.116.235044
Chen, Y. Eugene
- You have accessSignificant Improvement of Antithrombotic Responses to Clopidogrel by Use of a Novel Conjugate as Revealed in an Arterial Model of ThrombosisHaoming Zhang, D. Adam Lauver, Hui Wang, Duxin Sun, Paul F. Hollenberg, Y. Eugene Chen, Yoichi Osawa and Daniel T. EitzmanJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 11-17; DOI: https://doi.org/10.1124/jpet.116.236034
Chen, Yuchen
- You have accessMolecular Properties of Drugs Interacting with SLC22 Transporters OAT1, OAT3, OCT1, and OCT2: A Machine-Learning ApproachHenry C. Liu, Anne Goldenberg, Yuchen Chen, Christina Lun, Wei Wu, Kevin T. Bush, Natasha Balac, Paul Rodriguez, Ruben Abagyan and Sanjay K. NigamJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 215-229; DOI: https://doi.org/10.1124/jpet.116.232660
Chiazza, Fausto
- You have accessEmpagliflozin Protects against Diet-Induced NLRP-3 Inflammasome Activation and Lipid AccumulationElisa Benetti, Raffaella Mastrocola, Giovanna Vitarelli, Juan Carlos Cutrin, Debora Nigro, Fausto Chiazza, Eric Mayoux, Massimo Collino and Roberto FantozziJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 45-53; DOI: https://doi.org/10.1124/jpet.116.235069
Chiu, Weihsueh A.
- You have accessTarget Organ Metabolism, Toxicity, and Mechanisms of Trichloroethylene and Perchloroethylene: Key Similarities, Differences, and Data GapsJoseph A. Cichocki, Kathryn Z. Guyton, Neela Guha, Weihsueh A. Chiu, Ivan Rusyn and Lawrence H. LashJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 110-123; DOI: https://doi.org/10.1124/jpet.116.232629
Cichocki, Joseph A.
- You have accessTarget Organ Metabolism, Toxicity, and Mechanisms of Trichloroethylene and Perchloroethylene: Key Similarities, Differences, and Data GapsJoseph A. Cichocki, Kathryn Z. Guyton, Neela Guha, Weihsueh A. Chiu, Ivan Rusyn and Lawrence H. LashJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 110-123; DOI: https://doi.org/10.1124/jpet.116.232629
Cogan, Derek
- You have accessSelectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman PrimatesSteven M. Weldon, Matthew A. Cerny, Kristina Gueneva-Boucheva, Derek Cogan, Xin Guo, Neil Moss, Jean-Hugues Parmentier, Jeremy R. Richman, Glenn A. Reinhart and Nicholas F. BrownJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 142-150; DOI: https://doi.org/10.1124/jpet.116.236463
Collino, Massimo
- You have accessEmpagliflozin Protects against Diet-Induced NLRP-3 Inflammasome Activation and Lipid AccumulationElisa Benetti, Raffaella Mastrocola, Giovanna Vitarelli, Juan Carlos Cutrin, Debora Nigro, Fausto Chiazza, Eric Mayoux, Massimo Collino and Roberto FantozziJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 45-53; DOI: https://doi.org/10.1124/jpet.116.235069
Collins, Gregory T.
- You have accessDiscriminative Stimulus Effects of Binary Drug Mixtures: Studies with Cocaine, MDPV, and CaffeineGregory T. Collins, Megan Abbott, Kayla Galindo, Elise L. Rush, Kenner C. Rice and Charles P. FranceJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 1-10; DOI: https://doi.org/10.1124/jpet.116.234252
Cornic, Laura
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Corona, Aaron
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Csekő, Kata
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Cutrin, Juan Carlos
- You have accessEmpagliflozin Protects against Diet-Induced NLRP-3 Inflammasome Activation and Lipid AccumulationElisa Benetti, Raffaella Mastrocola, Giovanna Vitarelli, Juan Carlos Cutrin, Debora Nigro, Fausto Chiazza, Eric Mayoux, Massimo Collino and Roberto FantozziJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 45-53; DOI: https://doi.org/10.1124/jpet.116.235069
D
Das, Aditi
- You have accessDevelopment of Poly Unsaturated Fatty Acid Derivatives of Aspirin for Inhibition of Platelet FunctionJahnabi Roy, Reheman Adili, Richard Kulmacz, Michael Holinstat and Aditi DasJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 134-141; DOI: https://doi.org/10.1124/jpet.116.234781
DeWire, Scott M.
- You have accessUnexpected Potency Differences between B-Cell–Activating Factor (BAFF) Antagonist Antibodies against Various Forms of BAFF: Trimer, 60-Mer, and Membrane-BoundAmy M. Nicoletti, Cynthia Hess Kenny, Ashraf M. Khalil, Qi Pan, Kerry L. M. Ralph, Julie Ritchie, Sathyadevi Venkataramani, David H. Presky, Scott M. DeWire and Scott R. BrodeurJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 37-44; DOI: https://doi.org/10.1124/jpet.116.236075
Dluzen, Douglas F.
- You have accessRegulation of UGT2B Expression and Activity by miR-216b-5p in Liver Cancer Cell LinesDouglas F. Dluzen, Aimee K. Sutliff, Gang Chen, Christy J. W. Watson, Faoud T. Ishmael and Philip LazarusJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 182-193; DOI: https://doi.org/10.1124/jpet.116.235044
Dossou, Katinia S. S.
- You have accessEffects of Ketamine and Ketamine Metabolites on Evoked Striatal Dopamine Release, Dopamine Receptors, and Monoamine TransportersAdem Can, Panos Zanos, Ruin Moaddel, Hye Jin Kang, Katinia S. S. Dossou, Irving W. Wainer, Joseph F. Cheer, Douglas O. Frost, Xi-Ping Huang and Todd D. GouldJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 159-170; DOI: https://doi.org/10.1124/jpet.116.235838
Duignan, David B.
- You have accessSphingosine-1-Phosphate (S1P) Lyase Inhibition Causes Increased Cardiac S1P Levels and Bradycardia in RatsChristopher M. Harris, Scott Mittelstadt, Patricia Banfor, Peter Bousquet, David B. Duignan, Gary Gintant, Michelle Hart, Youngjae Kim and Jason SegretiJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 151-158; DOI: https://doi.org/10.1124/jpet.116.235002
E
Eberhardt, Esther
- You have accessPropacetamol-Induced Injection Pain Is Associated with Activation of Transient Receptor Potential Vanilloid 1 ChannelsFlorian Schillers, Esther Eberhardt, Andreas Leffler and Mirjam EberhardtJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 18-25; DOI: https://doi.org/10.1124/jpet.116.233452
Eberhardt, Mirjam
- You have accessPropacetamol-Induced Injection Pain Is Associated with Activation of Transient Receptor Potential Vanilloid 1 ChannelsFlorian Schillers, Esther Eberhardt, Andreas Leffler and Mirjam EberhardtJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 18-25; DOI: https://doi.org/10.1124/jpet.116.233452
Eitzman, Daniel T.
- You have accessSignificant Improvement of Antithrombotic Responses to Clopidogrel by Use of a Novel Conjugate as Revealed in an Arterial Model of ThrombosisHaoming Zhang, D. Adam Lauver, Hui Wang, Duxin Sun, Paul F. Hollenberg, Y. Eugene Chen, Yoichi Osawa and Daniel T. EitzmanJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 11-17; DOI: https://doi.org/10.1124/jpet.116.236034
Erickson, Sarah L.
- You have accessPregnane X Receptor Activation Attenuates Inflammation-Associated Intestinal Epithelial Barrier Dysfunction by Inhibiting Cytokine-Induced Myosin Light-Chain Kinase Expression and c-Jun N-Terminal Kinase 1/2 ActivationAditya Garg, Angela Zhao, Sarah L. Erickson, Subhajit Mukherjee, Aik Jiang Lau, Laurie Alston, Thomas K. H. Chang, Sridhar Mani and Simon A. HirotaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 91-101; DOI: https://doi.org/10.1124/jpet.116.234096
F
Fantozzi, Roberto
- You have accessEmpagliflozin Protects against Diet-Induced NLRP-3 Inflammasome Activation and Lipid AccumulationElisa Benetti, Raffaella Mastrocola, Giovanna Vitarelli, Juan Carlos Cutrin, Debora Nigro, Fausto Chiazza, Eric Mayoux, Massimo Collino and Roberto FantozziJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 45-53; DOI: https://doi.org/10.1124/jpet.116.235069
Felix, John P.
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Ferdinandy, Péter
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
France, Charles P.
- You have accessDiscriminative Stimulus Effects of Binary Drug Mixtures: Studies with Cocaine, MDPV, and CaffeineGregory T. Collins, Megan Abbott, Kayla Galindo, Elise L. Rush, Kenner C. Rice and Charles P. FranceJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 1-10; DOI: https://doi.org/10.1124/jpet.116.234252
Freissmuth, Michael
- You have accessComparison of the β-Adrenergic Receptor Antagonists Landiolol and Esmolol: Receptor Selectivity, Partial Agonism, and Pharmacochaperoning ActionsShahrooz Nasrollahi-Shirazi, Sonja Sucic, Qiong Yang, Michael Freissmuth and Christian NanoffJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 73-81; DOI: https://doi.org/10.1124/jpet.116.232884
Frost, Douglas O.
- You have accessEffects of Ketamine and Ketamine Metabolites on Evoked Striatal Dopamine Release, Dopamine Receptors, and Monoamine TransportersAdem Can, Panos Zanos, Ruin Moaddel, Hye Jin Kang, Katinia S. S. Dossou, Irving W. Wainer, Joseph F. Cheer, Douglas O. Frost, Xi-Ping Huang and Todd D. GouldJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 159-170; DOI: https://doi.org/10.1124/jpet.116.235838
Funakoshi, Kodai
- You have accessActivation of p38 Mitogen-Activated Protein Kinase by Clotrimazole Induces Multidrug Resistance–Associated Protein 3 Activation through a Novel Transcriptional ElementTakamitsu Sasaki, Keita Inami, Yoshihiro Numata, Kodai Funakoshi, Midori Yoshida, Takeshi Kumagai, Shuichi Kanno, Satomi Matsui, Takayoshi Toriyabe, Yasushi Yamazoe, Kouichi Yoshinari and Kiyoshi NagataJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 102-109; DOI: https://doi.org/10.1124/jpet.115.231589
Fürst, Susanna
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
G
Galindo, Kayla
- You have accessDiscriminative Stimulus Effects of Binary Drug Mixtures: Studies with Cocaine, MDPV, and CaffeineGregory T. Collins, Megan Abbott, Kayla Galindo, Elise L. Rush, Kenner C. Rice and Charles P. FranceJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 1-10; DOI: https://doi.org/10.1124/jpet.116.234252
Garcia, Maria L.
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Garg, Aditya
- You have accessPregnane X Receptor Activation Attenuates Inflammation-Associated Intestinal Epithelial Barrier Dysfunction by Inhibiting Cytokine-Induced Myosin Light-Chain Kinase Expression and c-Jun N-Terminal Kinase 1/2 ActivationAditya Garg, Angela Zhao, Sarah L. Erickson, Subhajit Mukherjee, Aik Jiang Lau, Laurie Alston, Thomas K. H. Chang, Sridhar Mani and Simon A. HirotaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 91-101; DOI: https://doi.org/10.1124/jpet.116.234096
Gill, Charles
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Gintant, Gary
- You have accessSphingosine-1-Phosphate (S1P) Lyase Inhibition Causes Increased Cardiac S1P Levels and Bradycardia in RatsChristopher M. Harris, Scott Mittelstadt, Patricia Banfor, Peter Bousquet, David B. Duignan, Gary Gintant, Michelle Hart, Youngjae Kim and Jason SegretiJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 151-158; DOI: https://doi.org/10.1124/jpet.116.235002
Giricz, Zoltán
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Goldenberg, Anne
- You have accessMolecular Properties of Drugs Interacting with SLC22 Transporters OAT1, OAT3, OCT1, and OCT2: A Machine-Learning ApproachHenry C. Liu, Anne Goldenberg, Yuchen Chen, Christina Lun, Wei Wu, Kevin T. Bush, Natasha Balac, Paul Rodriguez, Ruben Abagyan and Sanjay K. NigamJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 215-229; DOI: https://doi.org/10.1124/jpet.116.232660
Gould, Todd D.
- You have accessEffects of Ketamine and Ketamine Metabolites on Evoked Striatal Dopamine Release, Dopamine Receptors, and Monoamine TransportersAdem Can, Panos Zanos, Ruin Moaddel, Hye Jin Kang, Katinia S. S. Dossou, Irving W. Wainer, Joseph F. Cheer, Douglas O. Frost, Xi-Ping Huang and Todd D. GouldJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 159-170; DOI: https://doi.org/10.1124/jpet.116.235838
Gueneva-Boucheva, Kristina
- You have accessSelectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman PrimatesSteven M. Weldon, Matthew A. Cerny, Kristina Gueneva-Boucheva, Derek Cogan, Xin Guo, Neil Moss, Jean-Hugues Parmentier, Jeremy R. Richman, Glenn A. Reinhart and Nicholas F. BrownJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 142-150; DOI: https://doi.org/10.1124/jpet.116.236463
Guha, Neela
- You have accessTarget Organ Metabolism, Toxicity, and Mechanisms of Trichloroethylene and Perchloroethylene: Key Similarities, Differences, and Data GapsJoseph A. Cichocki, Kathryn Z. Guyton, Neela Guha, Weihsueh A. Chiu, Ivan Rusyn and Lawrence H. LashJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 110-123; DOI: https://doi.org/10.1124/jpet.116.232629
Guo, Xin
- You have accessSelectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman PrimatesSteven M. Weldon, Matthew A. Cerny, Kristina Gueneva-Boucheva, Derek Cogan, Xin Guo, Neil Moss, Jean-Hugues Parmentier, Jeremy R. Richman, Glenn A. Reinhart and Nicholas F. BrownJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 142-150; DOI: https://doi.org/10.1124/jpet.116.236463
Guyton, Kathryn Z.
- You have accessTarget Organ Metabolism, Toxicity, and Mechanisms of Trichloroethylene and Perchloroethylene: Key Similarities, Differences, and Data GapsJoseph A. Cichocki, Kathryn Z. Guyton, Neela Guha, Weihsueh A. Chiu, Ivan Rusyn and Lawrence H. LashJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 110-123; DOI: https://doi.org/10.1124/jpet.116.232629
Gynther, Mikko
- You have accessIn Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor {4-[bis-(benzo[d][1,3]dioxol-5-yl)methyl]-piperidin-1-yl}(1H-1,2,4-triazol-1-yl)methanone (JJKK-048)Niina Aaltonen, Ewa Kedzierska, Jolanta Orzelska-Górka, Marko Lehtonen, Dina Navia-Paldanius, Hermina Jakupovic, Juha R. Savinainen, Tapio Nevalainen, Jarmo T. Laitinen, Teija Parkkari and Mikko GyntherJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 62-72; DOI: https://doi.org/10.1124/jpet.116.233114
H
Hampton, Caryn
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Harris, Christopher M.
- You have accessSphingosine-1-Phosphate (S1P) Lyase Inhibition Causes Increased Cardiac S1P Levels and Bradycardia in RatsChristopher M. Harris, Scott Mittelstadt, Patricia Banfor, Peter Bousquet, David B. Duignan, Gary Gintant, Michelle Hart, Youngjae Kim and Jason SegretiJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 151-158; DOI: https://doi.org/10.1124/jpet.116.235002
Hart, Michelle
- You have accessSphingosine-1-Phosphate (S1P) Lyase Inhibition Causes Increased Cardiac S1P Levels and Bradycardia in RatsChristopher M. Harris, Scott Mittelstadt, Patricia Banfor, Peter Bousquet, David B. Duignan, Gary Gintant, Michelle Hart, Youngjae Kim and Jason SegretiJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 151-158; DOI: https://doi.org/10.1124/jpet.116.235002
Helyes, Zsuzsanna
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Hirota, Simon A.
- You have accessPregnane X Receptor Activation Attenuates Inflammation-Associated Intestinal Epithelial Barrier Dysfunction by Inhibiting Cytokine-Induced Myosin Light-Chain Kinase Expression and c-Jun N-Terminal Kinase 1/2 ActivationAditya Garg, Angela Zhao, Sarah L. Erickson, Subhajit Mukherjee, Aik Jiang Lau, Laurie Alston, Thomas K. H. Chang, Sridhar Mani and Simon A. HirotaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 91-101; DOI: https://doi.org/10.1124/jpet.116.234096
Holinstat, Michael
- You have accessDevelopment of Poly Unsaturated Fatty Acid Derivatives of Aspirin for Inhibition of Platelet FunctionJahnabi Roy, Reheman Adili, Richard Kulmacz, Michael Holinstat and Aditi DasJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 134-141; DOI: https://doi.org/10.1124/jpet.116.234781
Hollenberg, Paul F.
- You have accessSignificant Improvement of Antithrombotic Responses to Clopidogrel by Use of a Novel Conjugate as Revealed in an Arterial Model of ThrombosisHaoming Zhang, D. Adam Lauver, Hui Wang, Duxin Sun, Paul F. Hollenberg, Y. Eugene Chen, Yoichi Osawa and Daniel T. EitzmanJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 11-17; DOI: https://doi.org/10.1124/jpet.116.236034
Hopkins, Mandi M.
- You have accessPositive and Negative Cross-Talk between Lysophosphatidic Acid Receptor 1, Free Fatty Acid Receptor 4, and Epidermal Growth Factor Receptor in Human Prostate Cancer CellsMandi M. Hopkins, Ze Liu and Kathryn E. MeierJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 124-133; DOI: https://doi.org/10.1124/jpet.116.233379
Hosztafi, Sándor
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Huang, Xi-Ping
- You have accessEffects of Ketamine and Ketamine Metabolites on Evoked Striatal Dopamine Release, Dopamine Receptors, and Monoamine TransportersAdem Can, Panos Zanos, Ruin Moaddel, Hye Jin Kang, Katinia S. S. Dossou, Irving W. Wainer, Joseph F. Cheer, Douglas O. Frost, Xi-Ping Huang and Todd D. GouldJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 159-170; DOI: https://doi.org/10.1124/jpet.116.235838
I
Inami, Keita
- You have accessActivation of p38 Mitogen-Activated Protein Kinase by Clotrimazole Induces Multidrug Resistance–Associated Protein 3 Activation through a Novel Transcriptional ElementTakamitsu Sasaki, Keita Inami, Yoshihiro Numata, Kodai Funakoshi, Midori Yoshida, Takeshi Kumagai, Shuichi Kanno, Satomi Matsui, Takayoshi Toriyabe, Yasushi Yamazoe, Kouichi Yoshinari and Kiyoshi NagataJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 102-109; DOI: https://doi.org/10.1124/jpet.115.231589
Ishmael, Faoud T.
- You have accessRegulation of UGT2B Expression and Activity by miR-216b-5p in Liver Cancer Cell LinesDouglas F. Dluzen, Aimee K. Sutliff, Gang Chen, Christy J. W. Watson, Faoud T. Ishmael and Philip LazarusJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 182-193; DOI: https://doi.org/10.1124/jpet.116.235044
J
Jakupovic, Hermina
- You have accessIn Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor {4-[bis-(benzo[d][1,3]dioxol-5-yl)methyl]-piperidin-1-yl}(1H-1,2,4-triazol-1-yl)methanone (JJKK-048)Niina Aaltonen, Ewa Kedzierska, Jolanta Orzelska-Górka, Marko Lehtonen, Dina Navia-Paldanius, Hermina Jakupovic, Juha R. Savinainen, Tapio Nevalainen, Jarmo T. Laitinen, Teija Parkkari and Mikko GyntherJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 62-72; DOI: https://doi.org/10.1124/jpet.116.233114
Jiang, Handong
- You have accessThe Marine-Derived Oligosaccharide Sulfate MS80, a Novel Transforming Growth Factor β1 Inhibitor, Reverses Epithelial Mesenchymal Transition Induced by Transforming Growth Factor-β1 and Suppresses Tumor MetastasisJi Zhou, Wenjie You, Guangqiang Sun, Yixuan Li, Bi Chen, Jing Ai and Handong JiangJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 54-61; DOI: https://doi.org/10.1124/jpet.116.234799
Jones, Spencer B.
- You have accessPharmacological Characterization of a Potent Inhibitor of Autotaxin in Animal Models of Inflammatory Bowel Disease and Multiple SclerosisKannan Thirunavukkarasu, Bailin Tan, Craig A. Swearingen, Guilherme Rocha, Hai H. Bui, Denis J. McCann, Spencer B. Jones, Bryan H. Norman, Lance A. Pfeifer and Joy K. SahaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 207-214; DOI: https://doi.org/10.1124/jpet.116.234013
K
Kaczorowski, Gregory J.
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Kang, Hye Jin
- You have accessEffects of Ketamine and Ketamine Metabolites on Evoked Striatal Dopamine Release, Dopamine Receptors, and Monoamine TransportersAdem Can, Panos Zanos, Ruin Moaddel, Hye Jin Kang, Katinia S. S. Dossou, Irving W. Wainer, Joseph F. Cheer, Douglas O. Frost, Xi-Ping Huang and Todd D. GouldJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 159-170; DOI: https://doi.org/10.1124/jpet.116.235838
Kanno, Shuichi
- You have accessActivation of p38 Mitogen-Activated Protein Kinase by Clotrimazole Induces Multidrug Resistance–Associated Protein 3 Activation through a Novel Transcriptional ElementTakamitsu Sasaki, Keita Inami, Yoshihiro Numata, Kodai Funakoshi, Midori Yoshida, Takeshi Kumagai, Shuichi Kanno, Satomi Matsui, Takayoshi Toriyabe, Yasushi Yamazoe, Kouichi Yoshinari and Kiyoshi NagataJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 102-109; DOI: https://doi.org/10.1124/jpet.115.231589
Kedzierska, Ewa
- You have accessIn Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor {4-[bis-(benzo[d][1,3]dioxol-5-yl)methyl]-piperidin-1-yl}(1H-1,2,4-triazol-1-yl)methanone (JJKK-048)Niina Aaltonen, Ewa Kedzierska, Jolanta Orzelska-Górka, Marko Lehtonen, Dina Navia-Paldanius, Hermina Jakupovic, Juha R. Savinainen, Tapio Nevalainen, Jarmo T. Laitinen, Teija Parkkari and Mikko GyntherJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 62-72; DOI: https://doi.org/10.1124/jpet.116.233114
Kenny, Cynthia Hess
- You have accessUnexpected Potency Differences between B-Cell–Activating Factor (BAFF) Antagonist Antibodies against Various Forms of BAFF: Trimer, 60-Mer, and Membrane-BoundAmy M. Nicoletti, Cynthia Hess Kenny, Ashraf M. Khalil, Qi Pan, Kerry L. M. Ralph, Julie Ritchie, Sathyadevi Venkataramani, David H. Presky, Scott M. DeWire and Scott R. BrodeurJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 37-44; DOI: https://doi.org/10.1124/jpet.116.236075
Khalil, Ashraf M.
- You have accessUnexpected Potency Differences between B-Cell–Activating Factor (BAFF) Antagonist Antibodies against Various Forms of BAFF: Trimer, 60-Mer, and Membrane-BoundAmy M. Nicoletti, Cynthia Hess Kenny, Ashraf M. Khalil, Qi Pan, Kerry L. M. Ralph, Julie Ritchie, Sathyadevi Venkataramani, David H. Presky, Scott M. DeWire and Scott R. BrodeurJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 37-44; DOI: https://doi.org/10.1124/jpet.116.236075
Kim, Youngjae
- You have accessSphingosine-1-Phosphate (S1P) Lyase Inhibition Causes Increased Cardiac S1P Levels and Bradycardia in RatsChristopher M. Harris, Scott Mittelstadt, Patricia Banfor, Peter Bousquet, David B. Duignan, Gary Gintant, Michelle Hart, Youngjae Kim and Jason SegretiJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 151-158; DOI: https://doi.org/10.1124/jpet.116.235002
Király, Kornél
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Kohler, Martin
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Korzekwa, Kenneth
- You have accessIntracellular Unbound Atorvastatin Concentrations in the Presence of Metabolism and TransportPriyanka Kulkarni, Kenneth Korzekwa and Swati NagarJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 26-36; DOI: https://doi.org/10.1124/jpet.116.235689
Kulkarni, Priyanka
- You have accessIntracellular Unbound Atorvastatin Concentrations in the Presence of Metabolism and TransportPriyanka Kulkarni, Kenneth Korzekwa and Swati NagarJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 26-36; DOI: https://doi.org/10.1124/jpet.116.235689
Kulmacz, Richard
- You have accessDevelopment of Poly Unsaturated Fatty Acid Derivatives of Aspirin for Inhibition of Platelet FunctionJahnabi Roy, Reheman Adili, Richard Kulmacz, Michael Holinstat and Aditi DasJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 134-141; DOI: https://doi.org/10.1124/jpet.116.234781
Kumagai, Takeshi
- You have accessActivation of p38 Mitogen-Activated Protein Kinase by Clotrimazole Induces Multidrug Resistance–Associated Protein 3 Activation through a Novel Transcriptional ElementTakamitsu Sasaki, Keita Inami, Yoshihiro Numata, Kodai Funakoshi, Midori Yoshida, Takeshi Kumagai, Shuichi Kanno, Satomi Matsui, Takayoshi Toriyabe, Yasushi Yamazoe, Kouichi Yoshinari and Kiyoshi NagataJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 102-109; DOI: https://doi.org/10.1124/jpet.115.231589
L
Lackó, Erzsébet
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Laitinen, Jarmo T.
- You have accessIn Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor {4-[bis-(benzo[d][1,3]dioxol-5-yl)methyl]-piperidin-1-yl}(1H-1,2,4-triazol-1-yl)methanone (JJKK-048)Niina Aaltonen, Ewa Kedzierska, Jolanta Orzelska-Górka, Marko Lehtonen, Dina Navia-Paldanius, Hermina Jakupovic, Juha R. Savinainen, Tapio Nevalainen, Jarmo T. Laitinen, Teija Parkkari and Mikko GyntherJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 62-72; DOI: https://doi.org/10.1124/jpet.116.233114
Lash, Lawrence H.
- You have accessTarget Organ Metabolism, Toxicity, and Mechanisms of Trichloroethylene and Perchloroethylene: Key Similarities, Differences, and Data GapsJoseph A. Cichocki, Kathryn Z. Guyton, Neela Guha, Weihsueh A. Chiu, Ivan Rusyn and Lawrence H. LashJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 110-123; DOI: https://doi.org/10.1124/jpet.116.232629
Lau, Aik Jiang
- You have accessPregnane X Receptor Activation Attenuates Inflammation-Associated Intestinal Epithelial Barrier Dysfunction by Inhibiting Cytokine-Induced Myosin Light-Chain Kinase Expression and c-Jun N-Terminal Kinase 1/2 ActivationAditya Garg, Angela Zhao, Sarah L. Erickson, Subhajit Mukherjee, Aik Jiang Lau, Laurie Alston, Thomas K. H. Chang, Sridhar Mani and Simon A. HirotaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 91-101; DOI: https://doi.org/10.1124/jpet.116.234096
Lauver, D. Adam
- You have accessSignificant Improvement of Antithrombotic Responses to Clopidogrel by Use of a Novel Conjugate as Revealed in an Arterial Model of ThrombosisHaoming Zhang, D. Adam Lauver, Hui Wang, Duxin Sun, Paul F. Hollenberg, Y. Eugene Chen, Yoichi Osawa and Daniel T. EitzmanJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 11-17; DOI: https://doi.org/10.1124/jpet.116.236034
Lazarus, Philip
- You have accessRegulation of UGT2B Expression and Activity by miR-216b-5p in Liver Cancer Cell LinesDouglas F. Dluzen, Aimee K. Sutliff, Gang Chen, Christy J. W. Watson, Faoud T. Ishmael and Philip LazarusJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 182-193; DOI: https://doi.org/10.1124/jpet.116.235044
Leffler, Andreas
- You have accessPropacetamol-Induced Injection Pain Is Associated with Activation of Transient Receptor Potential Vanilloid 1 ChannelsFlorian Schillers, Esther Eberhardt, Andreas Leffler and Mirjam EberhardtJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 18-25; DOI: https://doi.org/10.1124/jpet.116.233452
Lehtonen, Marko
- You have accessIn Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor {4-[bis-(benzo[d][1,3]dioxol-5-yl)methyl]-piperidin-1-yl}(1H-1,2,4-triazol-1-yl)methanone (JJKK-048)Niina Aaltonen, Ewa Kedzierska, Jolanta Orzelska-Górka, Marko Lehtonen, Dina Navia-Paldanius, Hermina Jakupovic, Juha R. Savinainen, Tapio Nevalainen, Jarmo T. Laitinen, Teija Parkkari and Mikko GyntherJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 62-72; DOI: https://doi.org/10.1124/jpet.116.233114
Li, Chenhong
- You have accessInhibition of CaMKIIα in the Central Nucleus of Amygdala Attenuates Fentanyl-Induced Hyperalgesia in RatsZhen Li, Chenhong Li, Pingping Yin, Zaijie Jim Wang and Fang LuoJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 82-89; DOI: https://doi.org/10.1124/jpet.116.233817
Li, Yixuan
- You have accessThe Marine-Derived Oligosaccharide Sulfate MS80, a Novel Transforming Growth Factor β1 Inhibitor, Reverses Epithelial Mesenchymal Transition Induced by Transforming Growth Factor-β1 and Suppresses Tumor MetastasisJi Zhou, Wenjie You, Guangqiang Sun, Yixuan Li, Bi Chen, Jing Ai and Handong JiangJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 54-61; DOI: https://doi.org/10.1124/jpet.116.234799
Li, Zhen
- You have accessInhibition of CaMKIIα in the Central Nucleus of Amygdala Attenuates Fentanyl-Induced Hyperalgesia in RatsZhen Li, Chenhong Li, Pingping Yin, Zaijie Jim Wang and Fang LuoJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 82-89; DOI: https://doi.org/10.1124/jpet.116.233817
Liu, Henry C.
- You have accessMolecular Properties of Drugs Interacting with SLC22 Transporters OAT1, OAT3, OCT1, and OCT2: A Machine-Learning ApproachHenry C. Liu, Anne Goldenberg, Yuchen Chen, Christina Lun, Wei Wu, Kevin T. Bush, Natasha Balac, Paul Rodriguez, Ruben Abagyan and Sanjay K. NigamJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 215-229; DOI: https://doi.org/10.1124/jpet.116.232660
Liu, Jessica
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Liu, Ze
- You have accessPositive and Negative Cross-Talk between Lysophosphatidic Acid Receptor 1, Free Fatty Acid Receptor 4, and Epidermal Growth Factor Receptor in Human Prostate Cancer CellsMandi M. Hopkins, Ze Liu and Kathryn E. MeierJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 124-133; DOI: https://doi.org/10.1124/jpet.116.233379
Lun, Christina
- You have accessMolecular Properties of Drugs Interacting with SLC22 Transporters OAT1, OAT3, OCT1, and OCT2: A Machine-Learning ApproachHenry C. Liu, Anne Goldenberg, Yuchen Chen, Christina Lun, Wei Wu, Kevin T. Bush, Natasha Balac, Paul Rodriguez, Ruben Abagyan and Sanjay K. NigamJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 215-229; DOI: https://doi.org/10.1124/jpet.116.232660
Luo, Fang
- You have accessInhibition of CaMKIIα in the Central Nucleus of Amygdala Attenuates Fentanyl-Induced Hyperalgesia in RatsZhen Li, Chenhong Li, Pingping Yin, Zaijie Jim Wang and Fang LuoJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 82-89; DOI: https://doi.org/10.1124/jpet.116.233817
M
Mani, Sridhar
- You have accessPregnane X Receptor Activation Attenuates Inflammation-Associated Intestinal Epithelial Barrier Dysfunction by Inhibiting Cytokine-Induced Myosin Light-Chain Kinase Expression and c-Jun N-Terminal Kinase 1/2 ActivationAditya Garg, Angela Zhao, Sarah L. Erickson, Subhajit Mukherjee, Aik Jiang Lau, Laurie Alston, Thomas K. H. Chang, Sridhar Mani and Simon A. HirotaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 91-101; DOI: https://doi.org/10.1124/jpet.116.234096
Mastrocola, Raffaella
- You have accessEmpagliflozin Protects against Diet-Induced NLRP-3 Inflammasome Activation and Lipid AccumulationElisa Benetti, Raffaella Mastrocola, Giovanna Vitarelli, Juan Carlos Cutrin, Debora Nigro, Fausto Chiazza, Eric Mayoux, Massimo Collino and Roberto FantozziJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 45-53; DOI: https://doi.org/10.1124/jpet.116.235069
Matsui, Satomi
- You have accessActivation of p38 Mitogen-Activated Protein Kinase by Clotrimazole Induces Multidrug Resistance–Associated Protein 3 Activation through a Novel Transcriptional ElementTakamitsu Sasaki, Keita Inami, Yoshihiro Numata, Kodai Funakoshi, Midori Yoshida, Takeshi Kumagai, Shuichi Kanno, Satomi Matsui, Takayoshi Toriyabe, Yasushi Yamazoe, Kouichi Yoshinari and Kiyoshi NagataJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 102-109; DOI: https://doi.org/10.1124/jpet.115.231589
Mayoux, Eric
- You have accessEmpagliflozin Protects against Diet-Induced NLRP-3 Inflammasome Activation and Lipid AccumulationElisa Benetti, Raffaella Mastrocola, Giovanna Vitarelli, Juan Carlos Cutrin, Debora Nigro, Fausto Chiazza, Eric Mayoux, Massimo Collino and Roberto FantozziJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 45-53; DOI: https://doi.org/10.1124/jpet.116.235069
McCann, Denis J.
- You have accessPharmacological Characterization of a Potent Inhibitor of Autotaxin in Animal Models of Inflammatory Bowel Disease and Multiple SclerosisKannan Thirunavukkarasu, Bailin Tan, Craig A. Swearingen, Guilherme Rocha, Hai H. Bui, Denis J. McCann, Spencer B. Jones, Bryan H. Norman, Lance A. Pfeifer and Joy K. SahaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 207-214; DOI: https://doi.org/10.1124/jpet.116.234013
Meier, Kathryn E.
- You have accessPositive and Negative Cross-Talk between Lysophosphatidic Acid Receptor 1, Free Fatty Acid Receptor 4, and Epidermal Growth Factor Receptor in Human Prostate Cancer CellsMandi M. Hopkins, Ze Liu and Kathryn E. MeierJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 124-133; DOI: https://doi.org/10.1124/jpet.116.233379
Metzger, Joseph M.
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Mittelstadt, Scott
- You have accessSphingosine-1-Phosphate (S1P) Lyase Inhibition Causes Increased Cardiac S1P Levels and Bradycardia in RatsChristopher M. Harris, Scott Mittelstadt, Patricia Banfor, Peter Bousquet, David B. Duignan, Gary Gintant, Michelle Hart, Youngjae Kim and Jason SegretiJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 151-158; DOI: https://doi.org/10.1124/jpet.116.235002
Moaddel, Ruin
- You have accessEffects of Ketamine and Ketamine Metabolites on Evoked Striatal Dopamine Release, Dopamine Receptors, and Monoamine TransportersAdem Can, Panos Zanos, Ruin Moaddel, Hye Jin Kang, Katinia S. S. Dossou, Irving W. Wainer, Joseph F. Cheer, Douglas O. Frost, Xi-Ping Huang and Todd D. GouldJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 159-170; DOI: https://doi.org/10.1124/jpet.116.235838
Moss, Neil
- You have accessSelectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman PrimatesSteven M. Weldon, Matthew A. Cerny, Kristina Gueneva-Boucheva, Derek Cogan, Xin Guo, Neil Moss, Jean-Hugues Parmentier, Jeremy R. Richman, Glenn A. Reinhart and Nicholas F. BrownJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 142-150; DOI: https://doi.org/10.1124/jpet.116.236463
Mousa, Shaaban A.
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Mukherjee, Subhajit
- You have accessPregnane X Receptor Activation Attenuates Inflammation-Associated Intestinal Epithelial Barrier Dysfunction by Inhibiting Cytokine-Induced Myosin Light-Chain Kinase Expression and c-Jun N-Terminal Kinase 1/2 ActivationAditya Garg, Angela Zhao, Sarah L. Erickson, Subhajit Mukherjee, Aik Jiang Lau, Laurie Alston, Thomas K. H. Chang, Sridhar Mani and Simon A. HirotaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 91-101; DOI: https://doi.org/10.1124/jpet.116.234096
N
Nagar, Swati
- You have accessIntracellular Unbound Atorvastatin Concentrations in the Presence of Metabolism and TransportPriyanka Kulkarni, Kenneth Korzekwa and Swati NagarJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 26-36; DOI: https://doi.org/10.1124/jpet.116.235689
Nagata, Kiyoshi
- You have accessActivation of p38 Mitogen-Activated Protein Kinase by Clotrimazole Induces Multidrug Resistance–Associated Protein 3 Activation through a Novel Transcriptional ElementTakamitsu Sasaki, Keita Inami, Yoshihiro Numata, Kodai Funakoshi, Midori Yoshida, Takeshi Kumagai, Shuichi Kanno, Satomi Matsui, Takayoshi Toriyabe, Yasushi Yamazoe, Kouichi Yoshinari and Kiyoshi NagataJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 102-109; DOI: https://doi.org/10.1124/jpet.115.231589
Nanoff, Christian
- You have accessComparison of the β-Adrenergic Receptor Antagonists Landiolol and Esmolol: Receptor Selectivity, Partial Agonism, and Pharmacochaperoning ActionsShahrooz Nasrollahi-Shirazi, Sonja Sucic, Qiong Yang, Michael Freissmuth and Christian NanoffJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 73-81; DOI: https://doi.org/10.1124/jpet.116.232884
Nasrollahi-Shirazi, Shahrooz
- You have accessComparison of the β-Adrenergic Receptor Antagonists Landiolol and Esmolol: Receptor Selectivity, Partial Agonism, and Pharmacochaperoning ActionsShahrooz Nasrollahi-Shirazi, Sonja Sucic, Qiong Yang, Michael Freissmuth and Christian NanoffJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 73-81; DOI: https://doi.org/10.1124/jpet.116.232884
Navia-Paldanius, Dina
- You have accessIn Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor {4-[bis-(benzo[d][1,3]dioxol-5-yl)methyl]-piperidin-1-yl}(1H-1,2,4-triazol-1-yl)methanone (JJKK-048)Niina Aaltonen, Ewa Kedzierska, Jolanta Orzelska-Górka, Marko Lehtonen, Dina Navia-Paldanius, Hermina Jakupovic, Juha R. Savinainen, Tapio Nevalainen, Jarmo T. Laitinen, Teija Parkkari and Mikko GyntherJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 62-72; DOI: https://doi.org/10.1124/jpet.116.233114
Nevalainen, Tapio
- You have accessIn Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor {4-[bis-(benzo[d][1,3]dioxol-5-yl)methyl]-piperidin-1-yl}(1H-1,2,4-triazol-1-yl)methanone (JJKK-048)Niina Aaltonen, Ewa Kedzierska, Jolanta Orzelska-Górka, Marko Lehtonen, Dina Navia-Paldanius, Hermina Jakupovic, Juha R. Savinainen, Tapio Nevalainen, Jarmo T. Laitinen, Teija Parkkari and Mikko GyntherJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 62-72; DOI: https://doi.org/10.1124/jpet.116.233114
Nicoletti, Amy M.
- You have accessUnexpected Potency Differences between B-Cell–Activating Factor (BAFF) Antagonist Antibodies against Various Forms of BAFF: Trimer, 60-Mer, and Membrane-BoundAmy M. Nicoletti, Cynthia Hess Kenny, Ashraf M. Khalil, Qi Pan, Kerry L. M. Ralph, Julie Ritchie, Sathyadevi Venkataramani, David H. Presky, Scott M. DeWire and Scott R. BrodeurJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 37-44; DOI: https://doi.org/10.1124/jpet.116.236075
Nigam, Sanjay K.
- You have accessMolecular Properties of Drugs Interacting with SLC22 Transporters OAT1, OAT3, OCT1, and OCT2: A Machine-Learning ApproachHenry C. Liu, Anne Goldenberg, Yuchen Chen, Christina Lun, Wei Wu, Kevin T. Bush, Natasha Balac, Paul Rodriguez, Ruben Abagyan and Sanjay K. NigamJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 215-229; DOI: https://doi.org/10.1124/jpet.116.232660
Nigro, Debora
- You have accessEmpagliflozin Protects against Diet-Induced NLRP-3 Inflammasome Activation and Lipid AccumulationElisa Benetti, Raffaella Mastrocola, Giovanna Vitarelli, Juan Carlos Cutrin, Debora Nigro, Fausto Chiazza, Eric Mayoux, Massimo Collino and Roberto FantozziJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 45-53; DOI: https://doi.org/10.1124/jpet.116.235069
Norman, Bryan H.
- You have accessPharmacological Characterization of a Potent Inhibitor of Autotaxin in Animal Models of Inflammatory Bowel Disease and Multiple SclerosisKannan Thirunavukkarasu, Bailin Tan, Craig A. Swearingen, Guilherme Rocha, Hai H. Bui, Denis J. McCann, Spencer B. Jones, Bryan H. Norman, Lance A. Pfeifer and Joy K. SahaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 207-214; DOI: https://doi.org/10.1124/jpet.116.234013
Numata, Yoshihiro
- You have accessActivation of p38 Mitogen-Activated Protein Kinase by Clotrimazole Induces Multidrug Resistance–Associated Protein 3 Activation through a Novel Transcriptional ElementTakamitsu Sasaki, Keita Inami, Yoshihiro Numata, Kodai Funakoshi, Midori Yoshida, Takeshi Kumagai, Shuichi Kanno, Satomi Matsui, Takayoshi Toriyabe, Yasushi Yamazoe, Kouichi Yoshinari and Kiyoshi NagataJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 102-109; DOI: https://doi.org/10.1124/jpet.115.231589
O
Ormes, James
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Orzelska-Górka, Jolanta
- You have accessIn Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor {4-[bis-(benzo[d][1,3]dioxol-5-yl)methyl]-piperidin-1-yl}(1H-1,2,4-triazol-1-yl)methanone (JJKK-048)Niina Aaltonen, Ewa Kedzierska, Jolanta Orzelska-Górka, Marko Lehtonen, Dina Navia-Paldanius, Hermina Jakupovic, Juha R. Savinainen, Tapio Nevalainen, Jarmo T. Laitinen, Teija Parkkari and Mikko GyntherJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 62-72; DOI: https://doi.org/10.1124/jpet.116.233114
Osawa, Yoichi
- You have accessSignificant Improvement of Antithrombotic Responses to Clopidogrel by Use of a Novel Conjugate as Revealed in an Arterial Model of ThrombosisHaoming Zhang, D. Adam Lauver, Hui Wang, Duxin Sun, Paul F. Hollenberg, Y. Eugene Chen, Yoichi Osawa and Daniel T. EitzmanJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 11-17; DOI: https://doi.org/10.1124/jpet.116.236034
Owens, Karen
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
P
Pai, Lee-Yuh
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Pan, Qi
- You have accessUnexpected Potency Differences between B-Cell–Activating Factor (BAFF) Antagonist Antibodies against Various Forms of BAFF: Trimer, 60-Mer, and Membrane-BoundAmy M. Nicoletti, Cynthia Hess Kenny, Ashraf M. Khalil, Qi Pan, Kerry L. M. Ralph, Julie Ritchie, Sathyadevi Venkataramani, David H. Presky, Scott M. DeWire and Scott R. BrodeurJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 37-44; DOI: https://doi.org/10.1124/jpet.116.236075
Parkkari, Teija
- You have accessIn Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor {4-[bis-(benzo[d][1,3]dioxol-5-yl)methyl]-piperidin-1-yl}(1H-1,2,4-triazol-1-yl)methanone (JJKK-048)Niina Aaltonen, Ewa Kedzierska, Jolanta Orzelska-Górka, Marko Lehtonen, Dina Navia-Paldanius, Hermina Jakupovic, Juha R. Savinainen, Tapio Nevalainen, Jarmo T. Laitinen, Teija Parkkari and Mikko GyntherJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 62-72; DOI: https://doi.org/10.1124/jpet.116.233114
Parmentier, Jean-Hugues
- You have accessSelectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman PrimatesSteven M. Weldon, Matthew A. Cerny, Kristina Gueneva-Boucheva, Derek Cogan, Xin Guo, Neil Moss, Jean-Hugues Parmentier, Jeremy R. Richman, Glenn A. Reinhart and Nicholas F. BrownJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 142-150; DOI: https://doi.org/10.1124/jpet.116.236463
Pasternak, Alexander
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Pfeifer, Lance A.
- You have accessPharmacological Characterization of a Potent Inhibitor of Autotaxin in Animal Models of Inflammatory Bowel Disease and Multiple SclerosisKannan Thirunavukkarasu, Bailin Tan, Craig A. Swearingen, Guilherme Rocha, Hai H. Bui, Denis J. McCann, Spencer B. Jones, Bryan H. Norman, Lance A. Pfeifer and Joy K. SahaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 207-214; DOI: https://doi.org/10.1124/jpet.116.234013
Presky, David H.
- You have accessUnexpected Potency Differences between B-Cell–Activating Factor (BAFF) Antagonist Antibodies against Various Forms of BAFF: Trimer, 60-Mer, and Membrane-BoundAmy M. Nicoletti, Cynthia Hess Kenny, Ashraf M. Khalil, Qi Pan, Kerry L. M. Ralph, Julie Ritchie, Sathyadevi Venkataramani, David H. Presky, Scott M. DeWire and Scott R. BrodeurJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 37-44; DOI: https://doi.org/10.1124/jpet.116.236075
Price, Olga
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Priest, Birgit T.
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
R
Ralph, Kerry L. M.
- You have accessUnexpected Potency Differences between B-Cell–Activating Factor (BAFF) Antagonist Antibodies against Various Forms of BAFF: Trimer, 60-Mer, and Membrane-BoundAmy M. Nicoletti, Cynthia Hess Kenny, Ashraf M. Khalil, Qi Pan, Kerry L. M. Ralph, Julie Ritchie, Sathyadevi Venkataramani, David H. Presky, Scott M. DeWire and Scott R. BrodeurJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 37-44; DOI: https://doi.org/10.1124/jpet.116.236075
Rasa, Cordelia
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Reinhart, Glenn A.
- You have accessSelectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman PrimatesSteven M. Weldon, Matthew A. Cerny, Kristina Gueneva-Boucheva, Derek Cogan, Xin Guo, Neil Moss, Jean-Hugues Parmentier, Jeremy R. Richman, Glenn A. Reinhart and Nicholas F. BrownJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 142-150; DOI: https://doi.org/10.1124/jpet.116.236463
Riba, Pál
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Rice, Kenner C.
- You have accessDiscriminative Stimulus Effects of Binary Drug Mixtures: Studies with Cocaine, MDPV, and CaffeineGregory T. Collins, Megan Abbott, Kayla Galindo, Elise L. Rush, Kenner C. Rice and Charles P. FranceJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 1-10; DOI: https://doi.org/10.1124/jpet.116.234252
Richman, Jeremy R.
- You have accessSelectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman PrimatesSteven M. Weldon, Matthew A. Cerny, Kristina Gueneva-Boucheva, Derek Cogan, Xin Guo, Neil Moss, Jean-Hugues Parmentier, Jeremy R. Richman, Glenn A. Reinhart and Nicholas F. BrownJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 142-150; DOI: https://doi.org/10.1124/jpet.116.236463
Ritchie, Julie
- You have accessUnexpected Potency Differences between B-Cell–Activating Factor (BAFF) Antagonist Antibodies against Various Forms of BAFF: Trimer, 60-Mer, and Membrane-BoundAmy M. Nicoletti, Cynthia Hess Kenny, Ashraf M. Khalil, Qi Pan, Kerry L. M. Ralph, Julie Ritchie, Sathyadevi Venkataramani, David H. Presky, Scott M. DeWire and Scott R. BrodeurJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 37-44; DOI: https://doi.org/10.1124/jpet.116.236075
Rocha, Guilherme
- You have accessPharmacological Characterization of a Potent Inhibitor of Autotaxin in Animal Models of Inflammatory Bowel Disease and Multiple SclerosisKannan Thirunavukkarasu, Bailin Tan, Craig A. Swearingen, Guilherme Rocha, Hai H. Bui, Denis J. McCann, Spencer B. Jones, Bryan H. Norman, Lance A. Pfeifer and Joy K. SahaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 207-214; DOI: https://doi.org/10.1124/jpet.116.234013
Rodriguez, Paul
- You have accessMolecular Properties of Drugs Interacting with SLC22 Transporters OAT1, OAT3, OCT1, and OCT2: A Machine-Learning ApproachHenry C. Liu, Anne Goldenberg, Yuchen Chen, Christina Lun, Wei Wu, Kevin T. Bush, Natasha Balac, Paul Rodriguez, Ruben Abagyan and Sanjay K. NigamJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 215-229; DOI: https://doi.org/10.1124/jpet.116.232660
Roy, Jahnabi
- You have accessDevelopment of Poly Unsaturated Fatty Acid Derivatives of Aspirin for Inhibition of Platelet FunctionJahnabi Roy, Reheman Adili, Richard Kulmacz, Michael Holinstat and Aditi DasJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 134-141; DOI: https://doi.org/10.1124/jpet.116.234781
Roy, Sophie
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Rush, Elise L.
- You have accessDiscriminative Stimulus Effects of Binary Drug Mixtures: Studies with Cocaine, MDPV, and CaffeineGregory T. Collins, Megan Abbott, Kayla Galindo, Elise L. Rush, Kenner C. Rice and Charles P. FranceJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 1-10; DOI: https://doi.org/10.1124/jpet.116.234252
Rusyn, Ivan
- You have accessTarget Organ Metabolism, Toxicity, and Mechanisms of Trichloroethylene and Perchloroethylene: Key Similarities, Differences, and Data GapsJoseph A. Cichocki, Kathryn Z. Guyton, Neela Guha, Weihsueh A. Chiu, Ivan Rusyn and Lawrence H. LashJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 110-123; DOI: https://doi.org/10.1124/jpet.116.232629
S
Saha, Joy K.
- You have accessPharmacological Characterization of a Potent Inhibitor of Autotaxin in Animal Models of Inflammatory Bowel Disease and Multiple SclerosisKannan Thirunavukkarasu, Bailin Tan, Craig A. Swearingen, Guilherme Rocha, Hai H. Bui, Denis J. McCann, Spencer B. Jones, Bryan H. Norman, Lance A. Pfeifer and Joy K. SahaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 207-214; DOI: https://doi.org/10.1124/jpet.116.234013
Sasaki, Takamitsu
- You have accessActivation of p38 Mitogen-Activated Protein Kinase by Clotrimazole Induces Multidrug Resistance–Associated Protein 3 Activation through a Novel Transcriptional ElementTakamitsu Sasaki, Keita Inami, Yoshihiro Numata, Kodai Funakoshi, Midori Yoshida, Takeshi Kumagai, Shuichi Kanno, Satomi Matsui, Takayoshi Toriyabe, Yasushi Yamazoe, Kouichi Yoshinari and Kiyoshi NagataJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 102-109; DOI: https://doi.org/10.1124/jpet.115.231589
Savinainen, Juha R.
- You have accessIn Vivo Characterization of the Ultrapotent Monoacylglycerol Lipase Inhibitor {4-[bis-(benzo[d][1,3]dioxol-5-yl)methyl]-piperidin-1-yl}(1H-1,2,4-triazol-1-yl)methanone (JJKK-048)Niina Aaltonen, Ewa Kedzierska, Jolanta Orzelska-Górka, Marko Lehtonen, Dina Navia-Paldanius, Hermina Jakupovic, Juha R. Savinainen, Tapio Nevalainen, Jarmo T. Laitinen, Teija Parkkari and Mikko GyntherJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 62-72; DOI: https://doi.org/10.1124/jpet.116.233114
Schäfer, Michael
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Schillers, Florian
- You have accessPropacetamol-Induced Injection Pain Is Associated with Activation of Transient Receptor Potential Vanilloid 1 ChannelsFlorian Schillers, Esther Eberhardt, Andreas Leffler and Mirjam EberhardtJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 18-25; DOI: https://doi.org/10.1124/jpet.116.233452
Segreti, Jason
- You have accessSphingosine-1-Phosphate (S1P) Lyase Inhibition Causes Increased Cardiac S1P Levels and Bradycardia in RatsChristopher M. Harris, Scott Mittelstadt, Patricia Banfor, Peter Bousquet, David B. Duignan, Gary Gintant, Michelle Hart, Youngjae Kim and Jason SegretiJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 151-158; DOI: https://doi.org/10.1124/jpet.116.235002
Shah, Kashmira
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Sucic, Sonja
- You have accessComparison of the β-Adrenergic Receptor Antagonists Landiolol and Esmolol: Receptor Selectivity, Partial Agonism, and Pharmacochaperoning ActionsShahrooz Nasrollahi-Shirazi, Sonja Sucic, Qiong Yang, Michael Freissmuth and Christian NanoffJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 73-81; DOI: https://doi.org/10.1124/jpet.116.232884
Sullivan, Kathleen A.
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Sun, Duxin
- You have accessSignificant Improvement of Antithrombotic Responses to Clopidogrel by Use of a Novel Conjugate as Revealed in an Arterial Model of ThrombosisHaoming Zhang, D. Adam Lauver, Hui Wang, Duxin Sun, Paul F. Hollenberg, Y. Eugene Chen, Yoichi Osawa and Daniel T. EitzmanJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 11-17; DOI: https://doi.org/10.1124/jpet.116.236034
Sun, Guangqiang
- You have accessThe Marine-Derived Oligosaccharide Sulfate MS80, a Novel Transforming Growth Factor β1 Inhibitor, Reverses Epithelial Mesenchymal Transition Induced by Transforming Growth Factor-β1 and Suppresses Tumor MetastasisJi Zhou, Wenjie You, Guangqiang Sun, Yixuan Li, Bi Chen, Jing Ai and Handong JiangJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 54-61; DOI: https://doi.org/10.1124/jpet.116.234799
Sutliff, Aimee K.
- You have accessRegulation of UGT2B Expression and Activity by miR-216b-5p in Liver Cancer Cell LinesDouglas F. Dluzen, Aimee K. Sutliff, Gang Chen, Christy J. W. Watson, Faoud T. Ishmael and Philip LazarusJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 182-193; DOI: https://doi.org/10.1124/jpet.116.235044
Swearingen, Craig A.
- You have accessPharmacological Characterization of a Potent Inhibitor of Autotaxin in Animal Models of Inflammatory Bowel Disease and Multiple SclerosisKannan Thirunavukkarasu, Bailin Tan, Craig A. Swearingen, Guilherme Rocha, Hai H. Bui, Denis J. McCann, Spencer B. Jones, Bryan H. Norman, Lance A. Pfeifer and Joy K. SahaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 207-214; DOI: https://doi.org/10.1124/jpet.116.234013
T
Tan, Bailin
- You have accessPharmacological Characterization of a Potent Inhibitor of Autotaxin in Animal Models of Inflammatory Bowel Disease and Multiple SclerosisKannan Thirunavukkarasu, Bailin Tan, Craig A. Swearingen, Guilherme Rocha, Hai H. Bui, Denis J. McCann, Spencer B. Jones, Bryan H. Norman, Lance A. Pfeifer and Joy K. SahaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 207-214; DOI: https://doi.org/10.1124/jpet.116.234013
Tang, Haifeng
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Thirunavukkarasu, Kannan
- You have accessPharmacological Characterization of a Potent Inhibitor of Autotaxin in Animal Models of Inflammatory Bowel Disease and Multiple SclerosisKannan Thirunavukkarasu, Bailin Tan, Craig A. Swearingen, Guilherme Rocha, Hai H. Bui, Denis J. McCann, Spencer B. Jones, Bryan H. Norman, Lance A. Pfeifer and Joy K. SahaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 207-214; DOI: https://doi.org/10.1124/jpet.116.234013
Thomas-Fowlkes, Brande
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Tong, Vince
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Toriyabe, Takayoshi
- You have accessActivation of p38 Mitogen-Activated Protein Kinase by Clotrimazole Induces Multidrug Resistance–Associated Protein 3 Activation through a Novel Transcriptional ElementTakamitsu Sasaki, Keita Inami, Yoshihiro Numata, Kodai Funakoshi, Midori Yoshida, Takeshi Kumagai, Shuichi Kanno, Satomi Matsui, Takayoshi Toriyabe, Yasushi Yamazoe, Kouichi Yoshinari and Kiyoshi NagataJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 102-109; DOI: https://doi.org/10.1124/jpet.115.231589
V
Váradi, András
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Venkataramani, Sathyadevi
- You have accessUnexpected Potency Differences between B-Cell–Activating Factor (BAFF) Antagonist Antibodies against Various Forms of BAFF: Trimer, 60-Mer, and Membrane-BoundAmy M. Nicoletti, Cynthia Hess Kenny, Ashraf M. Khalil, Qi Pan, Kerry L. M. Ralph, Julie Ritchie, Sathyadevi Venkataramani, David H. Presky, Scott M. DeWire and Scott R. BrodeurJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 37-44; DOI: https://doi.org/10.1124/jpet.116.236075
Vitarelli, Giovanna
- You have accessEmpagliflozin Protects against Diet-Induced NLRP-3 Inflammasome Activation and Lipid AccumulationElisa Benetti, Raffaella Mastrocola, Giovanna Vitarelli, Juan Carlos Cutrin, Debora Nigro, Fausto Chiazza, Eric Mayoux, Massimo Collino and Roberto FantozziJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 45-53; DOI: https://doi.org/10.1124/jpet.116.235069
W
Wainer, Irving W.
- You have accessEffects of Ketamine and Ketamine Metabolites on Evoked Striatal Dopamine Release, Dopamine Receptors, and Monoamine TransportersAdem Can, Panos Zanos, Ruin Moaddel, Hye Jin Kang, Katinia S. S. Dossou, Irving W. Wainer, Joseph F. Cheer, Douglas O. Frost, Xi-Ping Huang and Todd D. GouldJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 159-170; DOI: https://doi.org/10.1124/jpet.116.235838
Wang, Hui
- You have accessSignificant Improvement of Antithrombotic Responses to Clopidogrel by Use of a Novel Conjugate as Revealed in an Arterial Model of ThrombosisHaoming Zhang, D. Adam Lauver, Hui Wang, Duxin Sun, Paul F. Hollenberg, Y. Eugene Chen, Yoichi Osawa and Daniel T. EitzmanJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 11-17; DOI: https://doi.org/10.1124/jpet.116.236034
Wang, Zaijie Jim
- You have accessInhibition of CaMKIIα in the Central Nucleus of Amygdala Attenuates Fentanyl-Induced Hyperalgesia in RatsZhen Li, Chenhong Li, Pingping Yin, Zaijie Jim Wang and Fang LuoJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 82-89; DOI: https://doi.org/10.1124/jpet.116.233817
Watson, Christy J. W.
- You have accessRegulation of UGT2B Expression and Activity by miR-216b-5p in Liver Cancer Cell LinesDouglas F. Dluzen, Aimee K. Sutliff, Gang Chen, Christy J. W. Watson, Faoud T. Ishmael and Philip LazarusJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 182-193; DOI: https://doi.org/10.1124/jpet.116.235044
Weldon, Steven M.
- You have accessSelectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman PrimatesSteven M. Weldon, Matthew A. Cerny, Kristina Gueneva-Boucheva, Derek Cogan, Xin Guo, Neil Moss, Jean-Hugues Parmentier, Jeremy R. Richman, Glenn A. Reinhart and Nicholas F. BrownJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 142-150; DOI: https://doi.org/10.1124/jpet.116.236463
Wu, Wei
- You have accessMolecular Properties of Drugs Interacting with SLC22 Transporters OAT1, OAT3, OCT1, and OCT2: A Machine-Learning ApproachHenry C. Liu, Anne Goldenberg, Yuchen Chen, Christina Lun, Wei Wu, Kevin T. Bush, Natasha Balac, Paul Rodriguez, Ruben Abagyan and Sanjay K. NigamJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 215-229; DOI: https://doi.org/10.1124/jpet.116.232660
X
Xiao, Jianying
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
Y
Yamazoe, Yasushi
- You have accessActivation of p38 Mitogen-Activated Protein Kinase by Clotrimazole Induces Multidrug Resistance–Associated Protein 3 Activation through a Novel Transcriptional ElementTakamitsu Sasaki, Keita Inami, Yoshihiro Numata, Kodai Funakoshi, Midori Yoshida, Takeshi Kumagai, Shuichi Kanno, Satomi Matsui, Takayoshi Toriyabe, Yasushi Yamazoe, Kouichi Yoshinari and Kiyoshi NagataJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 102-109; DOI: https://doi.org/10.1124/jpet.115.231589
Yang, Qiong
- You have accessComparison of the β-Adrenergic Receptor Antagonists Landiolol and Esmolol: Receptor Selectivity, Partial Agonism, and Pharmacochaperoning ActionsShahrooz Nasrollahi-Shirazi, Sonja Sucic, Qiong Yang, Michael Freissmuth and Christian NanoffJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 73-81; DOI: https://doi.org/10.1124/jpet.116.232884
Yin, Pingping
- You have accessInhibition of CaMKIIα in the Central Nucleus of Amygdala Attenuates Fentanyl-Induced Hyperalgesia in RatsZhen Li, Chenhong Li, Pingping Yin, Zaijie Jim Wang and Fang LuoJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 82-89; DOI: https://doi.org/10.1124/jpet.116.233817
Yoshida, Midori
- You have accessActivation of p38 Mitogen-Activated Protein Kinase by Clotrimazole Induces Multidrug Resistance–Associated Protein 3 Activation through a Novel Transcriptional ElementTakamitsu Sasaki, Keita Inami, Yoshihiro Numata, Kodai Funakoshi, Midori Yoshida, Takeshi Kumagai, Shuichi Kanno, Satomi Matsui, Takayoshi Toriyabe, Yasushi Yamazoe, Kouichi Yoshinari and Kiyoshi NagataJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 102-109; DOI: https://doi.org/10.1124/jpet.115.231589
Yoshinari, Kouichi
- You have accessActivation of p38 Mitogen-Activated Protein Kinase by Clotrimazole Induces Multidrug Resistance–Associated Protein 3 Activation through a Novel Transcriptional ElementTakamitsu Sasaki, Keita Inami, Yoshihiro Numata, Kodai Funakoshi, Midori Yoshida, Takeshi Kumagai, Shuichi Kanno, Satomi Matsui, Takayoshi Toriyabe, Yasushi Yamazoe, Kouichi Yoshinari and Kiyoshi NagataJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 102-109; DOI: https://doi.org/10.1124/jpet.115.231589
You, Wenjie
- You have accessThe Marine-Derived Oligosaccharide Sulfate MS80, a Novel Transforming Growth Factor β1 Inhibitor, Reverses Epithelial Mesenchymal Transition Induced by Transforming Growth Factor-β1 and Suppresses Tumor MetastasisJi Zhou, Wenjie You, Guangqiang Sun, Yixuan Li, Bi Chen, Jing Ai and Handong JiangJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 54-61; DOI: https://doi.org/10.1124/jpet.116.234799
Z
Zádori, Zoltán Sándor
- You have accessNew Morphine Analogs Produce Peripheral Antinociception within a Certain Dose Range of Their Systemic AdministrationErzsébet Lackó, Pál Riba, Zoltán Giricz, András Váradi, Laura Cornic, Mihály Balogh, Kornél Király, Kata Csekő, Shaaban A. Mousa, Sándor Hosztafi, Michael Schäfer, Zoltán Sándor Zádori, Zsuzsanna Helyes, Péter Ferdinandy, Susanna Fürst and Mahmoud Al-KhrasaniJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 171-181; DOI: https://doi.org/10.1124/jpet.116.233551
Zanos, Panos
- You have accessEffects of Ketamine and Ketamine Metabolites on Evoked Striatal Dopamine Release, Dopamine Receptors, and Monoamine TransportersAdem Can, Panos Zanos, Ruin Moaddel, Hye Jin Kang, Katinia S. S. Dossou, Irving W. Wainer, Joseph F. Cheer, Douglas O. Frost, Xi-Ping Huang and Todd D. GouldJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 159-170; DOI: https://doi.org/10.1124/jpet.116.235838
Zhang, Haoming
- You have accessSignificant Improvement of Antithrombotic Responses to Clopidogrel by Use of a Novel Conjugate as Revealed in an Arterial Model of ThrombosisHaoming Zhang, D. Adam Lauver, Hui Wang, Duxin Sun, Paul F. Hollenberg, Y. Eugene Chen, Yoichi Osawa and Daniel T. EitzmanJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 11-17; DOI: https://doi.org/10.1124/jpet.116.236034
Zhao, Angela
- You have accessPregnane X Receptor Activation Attenuates Inflammation-Associated Intestinal Epithelial Barrier Dysfunction by Inhibiting Cytokine-Induced Myosin Light-Chain Kinase Expression and c-Jun N-Terminal Kinase 1/2 ActivationAditya Garg, Angela Zhao, Sarah L. Erickson, Subhajit Mukherjee, Aik Jiang Lau, Laurie Alston, Thomas K. H. Chang, Sridhar Mani and Simon A. HirotaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 91-101; DOI: https://doi.org/10.1124/jpet.116.234096
Zhou, Ji
- You have accessThe Marine-Derived Oligosaccharide Sulfate MS80, a Novel Transforming Growth Factor β1 Inhibitor, Reverses Epithelial Mesenchymal Transition Induced by Transforming Growth Factor-β1 and Suppresses Tumor MetastasisJi Zhou, Wenjie You, Guangqiang Sun, Yixuan Li, Bi Chen, Jing Ai and Handong JiangJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 54-61; DOI: https://doi.org/10.1124/jpet.116.234799
Zhou, Xiaoyan
- You have accessThe Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter’s Syndrome Type II PhenotypeCaryn Hampton, Xiaoyan Zhou, Birgit T. Priest, Lee-Yuh Pai, John P. Felix, Brande Thomas-Fowlkes, Jessica Liu, Martin Kohler, Jianying Xiao, Aaron Corona, Olga Price, Charles Gill, Kashmira Shah, Cordelia Rasa, Vince Tong, Karen Owens, James Ormes, Haifeng Tang, Sophie Roy, Kathleen A. Sullivan, Joseph M. Metzger, Magdalena Alonso-Galicia, Gregory J. Kaczorowski, Alexander Pasternak and Maria L. GarciaJournal of Pharmacology and Experimental Therapeutics October 2016, 359 (1) 194-206; DOI: https://doi.org/10.1124/jpet.116.235150
In this issue

Advertisement