Research ArticleMinireviews
Endogenous Allosteric Modulators of G Protein–Coupled Receptors
Emma T. van der Westhuizen, Celine Valant, Patrick M. Sexton and Arthur Christopoulos
Journal of Pharmacology and Experimental Therapeutics May 2015, 353 (2) 246-260; DOI: https://doi.org/10.1124/jpet.114.221606
Emma T. van der Westhuizen
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
Celine Valant
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
Patrick M. Sexton
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
Arthur Christopoulos
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
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Research ArticleMinireviews
Endogenous GPCR Allosteric Modulators
Emma T. van der Westhuizen, Celine Valant, Patrick M. Sexton and Arthur Christopoulos
Journal of Pharmacology and Experimental Therapeutics May 1, 2015, 353 (2) 246-260; DOI: https://doi.org/10.1124/jpet.114.221606
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- Article
- Abstract
- Introduction
- G Proteins as Endogenous Allosteric Modulators
- GPCR–Accessory Protein Interactions
- Ions as Allosteric Modulators
- Lipids as Allosteric Modulators
- Amino Acids and Peptides as Allosteric Modulators
- Allosteric Autoantibodies
- Concluding Remarks
- Authorship Contributions
- Footnotes
- Abbreviations
- References
- Figures & Data
- Info & Metrics
- eLetters
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