Research ArticleDrug Discovery and Translational Medicine
The Protease Activated Receptor 2 (PAR2) Polymorphic Variant F240S Constitutively Activates PAR2 Receptors and Potentiates Responses to Small-Molecule PAR2 Agonists
Jian-Nong Ma and Ethan S. Burstein
Journal of Pharmacology and Experimental Therapeutics December 2013, 347 (3) 697-704; DOI: https://doi.org/10.1124/jpet.113.208744