Research ArticleDrug Discovery and Translational Medicine
Linking Phenotype to Kinase: Identification of a Novel Benzoxaborole Hinge-Binding Motif for Kinase Inhibition and Development of High-Potency Rho Kinase Inhibitors
Tsutomu Akama, Chen Dong, Charlotte Virtucio, David Sullivan, Yasheen Zhou, Yong-Kang Zhang, Fernando Rock, Yvonne Freund, Liang Liu, Wei Bu, Anne Wu, Xiao-Qing Fan and Kurt Jarnagin
Journal of Pharmacology and Experimental Therapeutics December 2013, 347 (3) 615-625; DOI: https://doi.org/10.1124/jpet.113.207662
Tsutomu Akama
Anacor Pharmaceuticals, Inc., Palo Alto, California
Chen Dong
Anacor Pharmaceuticals, Inc., Palo Alto, California
Charlotte Virtucio
Anacor Pharmaceuticals, Inc., Palo Alto, California
David Sullivan
Anacor Pharmaceuticals, Inc., Palo Alto, California
Yasheen Zhou
Anacor Pharmaceuticals, Inc., Palo Alto, California
Yong-Kang Zhang
Anacor Pharmaceuticals, Inc., Palo Alto, California
Fernando Rock
Anacor Pharmaceuticals, Inc., Palo Alto, California
Yvonne Freund
Anacor Pharmaceuticals, Inc., Palo Alto, California
Liang Liu
Anacor Pharmaceuticals, Inc., Palo Alto, California
Wei Bu
Anacor Pharmaceuticals, Inc., Palo Alto, California
Anne Wu
Anacor Pharmaceuticals, Inc., Palo Alto, California
Xiao-Qing Fan
Anacor Pharmaceuticals, Inc., Palo Alto, California
Kurt Jarnagin
Anacor Pharmaceuticals, Inc., Palo Alto, California
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Research ArticleDrug Discovery and Translational Medicine
Benzoxaborole Rho Kinase Inhibitors
Tsutomu Akama, Chen Dong, Charlotte Virtucio, David Sullivan, Yasheen Zhou, Yong-Kang Zhang, Fernando Rock, Yvonne Freund, Liang Liu, Wei Bu, Anne Wu, Xiao-Qing Fan and Kurt Jarnagin
Journal of Pharmacology and Experimental Therapeutics December 1, 2013, 347 (3) 615-625; DOI: https://doi.org/10.1124/jpet.113.207662
Research ArticleDrug Discovery and Translational Medicine
Benzoxaborole Rho Kinase Inhibitors
Tsutomu Akama, Chen Dong, Charlotte Virtucio, David Sullivan, Yasheen Zhou, Yong-Kang Zhang, Fernando Rock, Yvonne Freund, Liang Liu, Wei Bu, Anne Wu, Xiao-Qing Fan and Kurt Jarnagin
Journal of Pharmacology and Experimental Therapeutics December 1, 2013, 347 (3) 615-625; DOI: https://doi.org/10.1124/jpet.113.207662
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