Research ArticleDrug Discovery and Translational Medicine
Inhibition of Btk with CC-292 Provides Early Pharmacodynamic Assessment of Activity in Mice and Humans
Erica K. Evans, Richland Tester, Sharon Aslanian, Russell Karp, Michael Sheets, Matthew T. Labenski, Steven R. Witowski, Heather Lounsbury, Prasoon Chaturvedi, Hormoz Mazdiyasni, Zhendong Zhu, Mariana Nacht, Martin I. Freed, Russell C. Petter, Alex Dubrovskiy, Juswinder Singh and William F. Westlin
Journal of Pharmacology and Experimental Therapeutics August 2013, 346 (2) 219-228; DOI: https://doi.org/10.1124/jpet.113.203489
Erica K. Evans
Celgene Avilomics Research, Bedford, Massachusetts
Richland Tester
Celgene Avilomics Research, Bedford, Massachusetts
Sharon Aslanian
Celgene Avilomics Research, Bedford, Massachusetts
Russell Karp
Celgene Avilomics Research, Bedford, Massachusetts
Michael Sheets
Celgene Avilomics Research, Bedford, Massachusetts
Matthew T. Labenski
Celgene Avilomics Research, Bedford, Massachusetts
Steven R. Witowski
Celgene Avilomics Research, Bedford, Massachusetts
Heather Lounsbury
Celgene Avilomics Research, Bedford, Massachusetts
Prasoon Chaturvedi
Celgene Avilomics Research, Bedford, Massachusetts
Hormoz Mazdiyasni
Celgene Avilomics Research, Bedford, Massachusetts
Zhendong Zhu
Celgene Avilomics Research, Bedford, Massachusetts
Mariana Nacht
Celgene Avilomics Research, Bedford, Massachusetts
Martin I. Freed
Celgene Avilomics Research, Bedford, Massachusetts
Russell C. Petter
Celgene Avilomics Research, Bedford, Massachusetts
Alex Dubrovskiy
Celgene Avilomics Research, Bedford, Massachusetts
Juswinder Singh
Celgene Avilomics Research, Bedford, Massachusetts
William F. Westlin
Celgene Avilomics Research, Bedford, Massachusetts

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Research ArticleDrug Discovery and Translational Medicine
Btk Inhibition with the Covalent Inhibitor CC-292
Erica K. Evans, Richland Tester, Sharon Aslanian, Russell Karp, Michael Sheets, Matthew T. Labenski, Steven R. Witowski, Heather Lounsbury, Prasoon Chaturvedi, Hormoz Mazdiyasni, Zhendong Zhu, Mariana Nacht, Martin I. Freed, Russell C. Petter, Alex Dubrovskiy, Juswinder Singh and William F. Westlin
Journal of Pharmacology and Experimental Therapeutics August 1, 2013, 346 (2) 219-228; DOI: https://doi.org/10.1124/jpet.113.203489
Research ArticleDrug Discovery and Translational Medicine
Btk Inhibition with the Covalent Inhibitor CC-292
Erica K. Evans, Richland Tester, Sharon Aslanian, Russell Karp, Michael Sheets, Matthew T. Labenski, Steven R. Witowski, Heather Lounsbury, Prasoon Chaturvedi, Hormoz Mazdiyasni, Zhendong Zhu, Mariana Nacht, Martin I. Freed, Russell C. Petter, Alex Dubrovskiy, Juswinder Singh and William F. Westlin
Journal of Pharmacology and Experimental Therapeutics August 1, 2013, 346 (2) 219-228; DOI: https://doi.org/10.1124/jpet.113.203489
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