Research ArticleCellular and Molecular
Target Binding Properties and Cellular Activity of Afatinib (BIBW 2992), an Irreversible ErbB Family Blocker
Flavio Solca, Goeran Dahl, Andreas Zoephel, Gerd Bader, Michael Sanderson, Christian Klein, Oliver Kraemer, Frank Himmelsbach, Eric Haaksma and Guenther R. Adolf
Journal of Pharmacology and Experimental Therapeutics November 2012, 343 (2) 342-350; DOI: https://doi.org/10.1124/jpet.112.197756
Flavio Solca
Boehringer Ingelheim RCV GmbH & Co. KG., Vienna, Austria (F.S., G.D., A.Z., G.B., M.S., C.K., O.K., E.H., G.R.A.); and Boehringer Ingelheim Pharma GmbH & Co. KG., Biberach/Riss, Germany (F.H.)
Goeran Dahl
Boehringer Ingelheim RCV GmbH & Co. KG., Vienna, Austria (F.S., G.D., A.Z., G.B., M.S., C.K., O.K., E.H., G.R.A.); and Boehringer Ingelheim Pharma GmbH & Co. KG., Biberach/Riss, Germany (F.H.)
Andreas Zoephel
Boehringer Ingelheim RCV GmbH & Co. KG., Vienna, Austria (F.S., G.D., A.Z., G.B., M.S., C.K., O.K., E.H., G.R.A.); and Boehringer Ingelheim Pharma GmbH & Co. KG., Biberach/Riss, Germany (F.H.)
Gerd Bader
Boehringer Ingelheim RCV GmbH & Co. KG., Vienna, Austria (F.S., G.D., A.Z., G.B., M.S., C.K., O.K., E.H., G.R.A.); and Boehringer Ingelheim Pharma GmbH & Co. KG., Biberach/Riss, Germany (F.H.)
Michael Sanderson
Boehringer Ingelheim RCV GmbH & Co. KG., Vienna, Austria (F.S., G.D., A.Z., G.B., M.S., C.K., O.K., E.H., G.R.A.); and Boehringer Ingelheim Pharma GmbH & Co. KG., Biberach/Riss, Germany (F.H.)
Christian Klein
Boehringer Ingelheim RCV GmbH & Co. KG., Vienna, Austria (F.S., G.D., A.Z., G.B., M.S., C.K., O.K., E.H., G.R.A.); and Boehringer Ingelheim Pharma GmbH & Co. KG., Biberach/Riss, Germany (F.H.)
Oliver Kraemer
Boehringer Ingelheim RCV GmbH & Co. KG., Vienna, Austria (F.S., G.D., A.Z., G.B., M.S., C.K., O.K., E.H., G.R.A.); and Boehringer Ingelheim Pharma GmbH & Co. KG., Biberach/Riss, Germany (F.H.)
Frank Himmelsbach
Boehringer Ingelheim RCV GmbH & Co. KG., Vienna, Austria (F.S., G.D., A.Z., G.B., M.S., C.K., O.K., E.H., G.R.A.); and Boehringer Ingelheim Pharma GmbH & Co. KG., Biberach/Riss, Germany (F.H.)
Eric Haaksma
Boehringer Ingelheim RCV GmbH & Co. KG., Vienna, Austria (F.S., G.D., A.Z., G.B., M.S., C.K., O.K., E.H., G.R.A.); and Boehringer Ingelheim Pharma GmbH & Co. KG., Biberach/Riss, Germany (F.H.)
Guenther R. Adolf
Boehringer Ingelheim RCV GmbH & Co. KG., Vienna, Austria (F.S., G.D., A.Z., G.B., M.S., C.K., O.K., E.H., G.R.A.); and Boehringer Ingelheim Pharma GmbH & Co. KG., Biberach/Riss, Germany (F.H.)

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In this issue
Research ArticleCellular and Molecular
Afatinib, an Irreversible Inhibitor of EGFR, HER2, and ErbB4
Flavio Solca, Goeran Dahl, Andreas Zoephel, Gerd Bader, Michael Sanderson, Christian Klein, Oliver Kraemer, Frank Himmelsbach, Eric Haaksma and Guenther R. Adolf
Journal of Pharmacology and Experimental Therapeutics November 1, 2012, 343 (2) 342-350; DOI: https://doi.org/10.1124/jpet.112.197756
Research ArticleCellular and Molecular
Afatinib, an Irreversible Inhibitor of EGFR, HER2, and ErbB4
Flavio Solca, Goeran Dahl, Andreas Zoephel, Gerd Bader, Michael Sanderson, Christian Klein, Oliver Kraemer, Frank Himmelsbach, Eric Haaksma and Guenther R. Adolf
Journal of Pharmacology and Experimental Therapeutics November 1, 2012, 343 (2) 342-350; DOI: https://doi.org/10.1124/jpet.112.197756
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