CTEP: A Novel, Potent, Long-Acting, and Orally Bioavailable Metabotropic Glutamate Receptor 5 Inhibitor

Lothar Lindemann; Georg Jaeschke; Aubin Michalon; Eric Vieira; Michael Honer; Will Spooren; Richard Porter; Thomas Hartung; Sabine Kolczewski; Bernd Büttelmann; Christophe Flament; Catherine Diener; Christophe Fischer; Silvia Gatti; Eric P. Prinssen; Neil Parrott; Gerhard Hoffmann; Joseph G. Wettstein

doi:10.1124/jpet.111.185660

Research ArticleNeuropharmacology

CTEP: A Novel, Potent, Long-Acting, and Orally Bioavailable Metabotropic Glutamate Receptor 5 Inhibitor

Lothar Lindemann, Georg Jaeschke, Aubin Michalon, Eric Vieira, Michael Honer, Will Spooren, Richard Porter, Thomas Hartung, Sabine Kolczewski, Bernd Büttelmann, Christophe Flament, Catherine Diener, Christophe Fischer, Silvia Gatti, Eric P. Prinssen, Neil Parrott, Gerhard Hoffmann and Joseph G. Wettstein

Journal of Pharmacology and Experimental Therapeutics November 2011, 339 (2) 474-486; DOI: https://doi.org/10.1124/jpet.111.185660

Lothar Lindemann

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Georg Jaeschke

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Aubin Michalon

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Eric Vieira

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Michael Honer

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Will Spooren

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Richard Porter

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Thomas Hartung

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Sabine Kolczewski

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Bernd Büttelmann

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Christophe Flament

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Catherine Diener

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Christophe Fischer

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Silvia Gatti

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Eric P. Prinssen

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Neil Parrott

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Gerhard Hoffmann

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Joseph G. Wettstein

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Journal of Pharmacology and Experimental Therapeutics

Vol. 339, Issue 2

1 Nov 2011

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Research ArticleNeuropharmacology