OtherNEUROPHARMACOLOGY
Begacestat (GSI-953): A Novel, Selective Thiophene Sulfonamide Inhibitor of Amyloid Precursor Protein γ-Secretase for the Treatment of Alzheimer's Disease
Robert L. Martone, Hua Zhou, Kevin Atchison, Thomas Comery, Jane Z. Xu, Xinyi Huang, Xioahai Gong, Mei Jin, Anthony Kreft, Boyd Harrison, Scott C. Mayer, Suzan Aschmies, Cathleen Gonzales, Margaret M. Zaleska, David R. Riddell, Erik Wagner, Peimin Lu, Shaiu-Ching Sun, June Sonnenberg-Reines, Aram Oganesian, Karissa Adkins, Michael W. Leach, David W. Clarke, Donna Huryn, Magid Abou-Gharbia, Ronald Magolda, Jonathan Bard, Glen Frick, Sangeeta Raje, S. Bradley Forlow, Carrie Balliet, Michael E. Burczynski, Peter H. Reinhart, Hong I. Wan, Menelas N. Pangalos and J. Steven Jacobsen
Journal of Pharmacology and Experimental Therapeutics November 2009, 331 (2) 598-608; DOI: https://doi.org/10.1124/jpet.109.152975
Robert L. Martone
Hua Zhou
Kevin Atchison
Thomas Comery
Jane Z. Xu
Xinyi Huang
Xioahai Gong
Mei Jin
Anthony Kreft
Boyd Harrison
Scott C. Mayer
Suzan Aschmies
Cathleen Gonzales
Margaret M. Zaleska
David R. Riddell
Erik Wagner
Peimin Lu
Shaiu-Ching Sun
June Sonnenberg-Reines
Aram Oganesian
Karissa Adkins
Michael W. Leach
David W. Clarke
Donna Huryn
Magid Abou-Gharbia
Ronald Magolda
Jonathan Bard
Glen Frick
Sangeeta Raje
S. Bradley Forlow
Carrie Balliet
Michael E. Burczynski
Peter H. Reinhart
Hong I. Wan
Menelas N. Pangalos
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OtherNEUROPHARMACOLOGY
Begacestat (GSI-953): A Novel, Selective Thiophene Sulfonamide Inhibitor of Amyloid Precursor Protein γ-Secretase for the Treatment of Alzheimer's Disease
Robert L. Martone, Hua Zhou, Kevin Atchison, Thomas Comery, Jane Z. Xu, Xinyi Huang, Xioahai Gong, Mei Jin, Anthony Kreft, Boyd Harrison, Scott C. Mayer, Suzan Aschmies, Cathleen Gonzales, Margaret M. Zaleska, David R. Riddell, Erik Wagner, Peimin Lu, Shaiu-Ching Sun, June Sonnenberg-Reines, Aram Oganesian, Karissa Adkins, Michael W. Leach, David W. Clarke, Donna Huryn, Magid Abou-Gharbia, Ronald Magolda, Jonathan Bard, Glen Frick, Sangeeta Raje, S. Bradley Forlow, Carrie Balliet, Michael E. Burczynski, Peter H. Reinhart, Hong I. Wan, Menelas N. Pangalos and J. Steven Jacobsen
Journal of Pharmacology and Experimental Therapeutics November 1, 2009, 331 (2) 598-608; DOI: https://doi.org/10.1124/jpet.109.152975
OtherNEUROPHARMACOLOGY
Begacestat (GSI-953): A Novel, Selective Thiophene Sulfonamide Inhibitor of Amyloid Precursor Protein γ-Secretase for the Treatment of Alzheimer's Disease
Robert L. Martone, Hua Zhou, Kevin Atchison, Thomas Comery, Jane Z. Xu, Xinyi Huang, Xioahai Gong, Mei Jin, Anthony Kreft, Boyd Harrison, Scott C. Mayer, Suzan Aschmies, Cathleen Gonzales, Margaret M. Zaleska, David R. Riddell, Erik Wagner, Peimin Lu, Shaiu-Ching Sun, June Sonnenberg-Reines, Aram Oganesian, Karissa Adkins, Michael W. Leach, David W. Clarke, Donna Huryn, Magid Abou-Gharbia, Ronald Magolda, Jonathan Bard, Glen Frick, Sangeeta Raje, S. Bradley Forlow, Carrie Balliet, Michael E. Burczynski, Peter H. Reinhart, Hong I. Wan, Menelas N. Pangalos and J. Steven Jacobsen
Journal of Pharmacology and Experimental Therapeutics November 1, 2009, 331 (2) 598-608; DOI: https://doi.org/10.1124/jpet.109.152975
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