Characterization of the Interaction of Indiplon, a Novel Pyrazolopyrimidine Sedative-Hypnotic, with the GABAA Receptor

Departments of Pharmacology (S.K.S., D.E.G.), Neuroscience (R.E.P., G.V., A.C.F.), and Medicinal Chemistry (R.S.G.), Neurocrine Biosciences Inc., San Diego, California

Address correspondence to:
Dr. Dimitri E. Grigoriadis, 12790 El Camino Real, San Diego, CA 92130. E-mail: dgrigoriadis{at}neurocrine.com

View Full Text

Statistics from Altmetric.com

Article usage

Article usage: July 2004 to January 2021

	Abstract	Full	Pdf
Jul 2004	62	0	74
Aug 2004	61	0	96
Sep 2004	32	0	67
Oct 2004	165	88	74
Nov 2004	93	116	95
Dec 2004	97	127	27
Jan 2005	69	90	38
Feb 2005	43	63	26
Mar 2005	56	77	35
Apr 2005	31	65	40
May 2005	44	51	13
Jun 2005	33	92	26
Jul 2005	20	59	19
Aug 2005	23	50	27
Sep 2005	33	52	20
Oct 2005	41	78	26
Nov 2005	50	81	65
Dec 2005	40	51	39
Jan 2006	44	76	55
Feb 2006	38	65	39
Mar 2006	50	78	46
Apr 2006	45	59	53
May 2006	65	83	54
Jun 2006	22	43	77
Jul 2006	21	41	28
Aug 2006	28	32	32
Sep 2006	18	25	22
Oct 2006	27	41	23
Nov 2006	25	29	14
Dec 2006	7	27	9
Jan 2007	15	26	18
Feb 2007	6	15	10
Mar 2007	7	29	15
Apr 2007	15	25	21
May 2007	11	37	19
Jun 2007	9	17	11
Jul 2007	14	17	21
Aug 2007	8	9	12
Sep 2007	4	7	8
Oct 2007	11	17	26
Nov 2007	11	19	12
Dec 2007	9	29	10
Jan 2008	7	9	10
Feb 2008	3	5	5
Mar 2008	15	13	10
Apr 2008	10	11	23
May 2008	9	13	16
Jun 2008	22	18	17
Jul 2008	10	14	7
Aug 2008	3	15	16
Sep 2008	3	20	11
Oct 2008	20	13	9
Nov 2008	15	9	10
Dec 2008	8	6	7
Jan 2009	6	10	8
Feb 2009	7	8	14
Mar 2009	11	7	14
Apr 2009	30	9	9
May 2009	3	3	5
Jun 2009	13	9	6
Jul 2009	9	10	6
Aug 2009	10	27	17
Sep 2009	5	9	8
Oct 2009	12	5	5
Nov 2009	15	10	6
Dec 2009	7	5	3
Jan 2010	14	7	9
Feb 2010	7	7	9
Mar 2010	12	7	8
Apr 2010	7	13	5
May 2010	10	6	5
Jun 2010	10	4	5
Jul 2010	15	6	6
Aug 2010	7	9	3
Sep 2010	3	11	8
Oct 2010	6	16	9
Nov 2010	3	17	18
Dec 2010	15	6	5
Jan 2011	10	10	6
Feb 2011	11	10	9
Mar 2011	13	20	21
Apr 2011	7	8	7
May 2011	6	7	8
Jun 2011	12	7	14
Jul 2011	7	8	11
Aug 2011	13	9	8
Sep 2011	7	19	9
Oct 2011	13	23	13
Nov 2011	12	13	9
Dec 2011	8	9	10
Jan 2012	7	11	17
Feb 2012	9	15	21
Mar 2012	14	7	13
Apr 2012	14	11	10
May 2012	11	9	13
Jun 2012	16	20	13
Jul 2012	13	14	9
Aug 2012	5	16	13
Sep 2012	9	11	11
Oct 2012	23	13	24
Nov 2012	21	14	17
Dec 2012	14	15	13
Jan 2013	16	11	9
Feb 2013	7	9	8
Mar 2013	15	9	14
Apr 2013	10	11	18
May 2013	8	16	14
Jun 2013	7	3	4
Jul 2013	9	5	9
Aug 2013	9	5	6
Sep 2013	17	5	9
Oct 2013	7	4	6
Nov 2013	3	4	3
Dec 2013	5	2	1
Jan 2014	16	8	1
Feb 2014	10	11	7
Mar 2014	7	8	5
Apr 2014	16	9	6
May 2014	9	3	13
Jun 2014	7	4	8
Jul 2014	10	24	2
Aug 2014	1	1	4
Sep 2014	3	2	5
Oct 2014	4	9	3
Nov 2014	2	0	0
Dec 2014	3	2	5
Jan 2015	3	4	1
Feb 2015	2	1	2
Mar 2015	17	3	4
Apr 2015	2	5	1
May 2015	9	11	2
Jun 2015	4	6	3
Jul 2015	4	3	7
Aug 2015	3	5	1
Sep 2015	4	1	1
Oct 2015	4	5	4
Nov 2015	5	3	4
Dec 2015	7	1	2
Jan 2016	17	2	6
Feb 2016	6	4	6
Mar 2016	4	3	12
Apr 2016	5	5	7
May 2016	6	4	14
Jun 2016	3	9	13
Jul 2016	4	4	13
Aug 2016	9	11	11
Sep 2016	1	8	14
Oct 2016	4	10	5
Nov 2016	1	14	8
Dec 2016	1	8	4
Jan 2017	3	29	8
Feb 2017	0	9	0
Mar 2017	0	14	4
Apr 2017	0	7	2
May 2017	0	11	1
Jun 2017	0	7	4
Jul 2017	2	3	0
Aug 2017	0	9	5
Sep 2017	2	6	2
Oct 2017	6	13	4
Nov 2017	2	21	6
Dec 2017	4	8	3
Jan 2018	1	11	7
Feb 2018	2	9	8
Mar 2018	1	9	5
Apr 2018	2	26	2
May 2018	0	9	5
Jun 2018	0	9	3
Jul 2018	0	7	6
Aug 2018	1	4	1
Sep 2018	0	6	1
Oct 2018	0	8	3
Nov 2018	2	16	3
Dec 2018	10	5	1
Jan 2019	6	0	0
Feb 2019	6	1	0
Mar 2019	13	6	1
Apr 2019	8	0	0
May 2019	14	0	2
Jun 2019	4	0	0
Jul 2019	4	0	2
Aug 2019	9	1	2
Sep 2019	15	1	0
Oct 2019	10	0	1
Nov 2019	22	0	4
Dec 2019	15	1	5
Jan 2020	15	1	4
Feb 2020	19	1	1
Mar 2020	6	4	2
Apr 2020	8	2	0
May 2020	6	3	2
Jun 2020	3	1	1
Jul 2020	6	0	0
Aug 2020	4	0	1
Sep 2020	7	2	0
Oct 2020	7	2	1
Nov 2020	4	2	1
Dec 2020	13	2	2
Jan 2021	11	2	1