Inhibition of Organic Anion Transporting Polypeptide-Mediated Hepatic Uptake Is the Major Determinant in the Pharmacokinetic Interaction between Bosentan and Cyclosporin A in the Rat

Address correspondence to:
Dr. Alexander Treiber, Department of Preclinical Pharmacokinetics and Metabolism, Actelion Pharmaceuticals Ltd., Gewerbestrasse 16, 4123 Allschwil, Switzerland. E-mail: alexander.treiber{at}actelion.com

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Oct 2020	12	3	3
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Dec 2020	14	5	4
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