Journal of Pharmacology and Experimental Therapeutics: 299 (3)

December 01, 2001; Volume 299,Issue 3

PERSPECTIVES IN PHARMACOLOGY

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Pharmacology of Opioid and Nonopioid Analgesics in Chronic Pain States
Thomas J. Martin and James C. Eisenach

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 811-817;
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Post-Translational Control of Endothelial Nitric Oxide Synthase: Why Isn't Calcium/Calmodulin Enough?
David Fulton, Jean-Philippe Gratton and William C. Sessa

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 818-824;

ABSORPTION, DISTRIBUTION, METABOLISM, AND EXCRETION

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Identification of Variants of CYP3A4 and Characterization of Their Abilities to Metabolize Testosterone and Chlorpyrifos
Diana Dai, Jun Tang, Randy Rose, Ernest Hodgson, Rachelle J. Bienstock, Harvey W. Mohrenweiser and Joyce A. Goldstein

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 825-831;
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Rifampin Is a Selective, Pleiotropic Inducer of Drug Metabolism Genes in Human Hepatocytes: Studies with cDNA and Oligonucleotide Expression Arrays
James M. Rae, Michael D. Johnson, Marc E. Lippman and David A. Flockhart

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 849-857;
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Differential Inhibition and Inactivation of Human CYP1 Enzymes bytrans-Resveratrol: Evidence for Mechanism-Based Inactivation of CYP1A2
Thomas K. H. Chang, Jie Chen and Wendy B. K. Lee

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 874-882;
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Improved Blood-Brain Barrier Penetration and Enhanced Analgesia of an Opioid Peptide by Glycosylation
R. D. Egleton, S. A. Mitchell, J. D. Huber, M. M. Palian, R. Polt and T. P. Davis

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 967-972;
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Interindividual Variability in Acetaminophen Glucuronidation by Human Liver Microsomes: Identification of Relevant Acetaminophen UDP-Glucuronosyltransferase Isoforms
Michael H. Court, Su X. Duan, Lisa L. von Moltke, David J. Greenblatt, Christopher J. Patten, John O. Miners and Peter I. Mackenzie

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 998-1006;

BEHAVIORAL PHARMACOLOGY

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Multiple Behavioral Effects of Cocaine- and Amphetamine-Regulated Transcript (CART) Peptides in Mice: CART 42–89 and CART 49–89 Differ in Potency and Activity
Anthony W. Bannon, Jennifer Seda, Michelle Carmouche, Jonathan M. Francis, Mark A. Jarosinski and James Douglass

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1021-1026;

CARDIOVASCULAR

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An Up-Regulation of Renal α₂A-Adrenoceptors Is Associated with Resistance to Salt-Induced Hypertension in Sabra Rats
Mostafa Khalid, Yves Giudicelli and Jean-Pierre Dausse

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 928-933;
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Gastrointestinal Prokinetic Drugs have Different Affinity for the Human Cardiac Human Ether-à-gogo K⁺ Channel
Franck Potet, Thierry Bouyssou, Denis Escande and Isabelle Baró

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1007-1012;
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Interaction of the Sulfonylthiourea HMR 1833 with Sulfonylurea Receptors and Recombinant ATP-Sensitive K⁺ Channels: Comparison with Glibenclamide
Ulrich Russ, Ulf Lange, Cornelia Löffler-Walz, Annette Hambrock and Ulrich Quast

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1049-1055;
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Vascular Endothelial Growth Factor (VEGF) Receptor-2 Antagonists Inhibit VEGF- and Basic Fibroblast Growth Factor-Induced Angiogenesis in Vivo and in Vitro
J.-C. Tille, J. Wood, S.J. Mandriota, C. Schnell, S. Ferrari, J. Mestan, Z. Zhu, L. Witte and M. S. Pepper

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1073-1085;
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Functional Calcitonin Gene-Related Peptide Subtype 2 Receptors in Porcine Coronary Arteries Are Identified as Calcitonin Gene-Related Peptide Subtype 1 Receptors by Radioligand Binding and Reverse Transcription-Polymerase Chain Reaction
Boyd R. Rorabaugh, Margaret A. Scofield, D. David Smith, William B. Jeffries and Peter W. Abel

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1086-1094;
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Effects of Heart Rate Reduction with Ivabradine on Exercise-Induced Myocardial Ischemia and Stunning
Xavier Monnet, Bijan Ghaleh, Patrice Colin, Olivier Parent de Curzon, Jean-François Giudicelli and Alain Berdeaux

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1133-1139;

CELLULAR AND MOLECULAR

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Ca²⁺ Influx through Nonselective Cation Channels Plays an Essential Role in Noradrenaline-Induced Arachidonic Acid Release in Chinese Hamster Ovary Cells Expressing α_1A-, α_1B-, or α_1D-Adrenergic Receptors
Yoshifumi Kawanabe, Nobuo Hashimoto, Tomoh Masaki and Soichi Miwa

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 901-907;
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Constitutive Activity of Histamine H₃ Receptors Stably Expressed in SK-N-MC Cells: Display of Agonism and Inverse Agonism by H₃ Antagonists
Kerstin Wieland, Gerold Bongers, Yumiko Yamamoto, Takeshi Hashimoto, Atsushi Yamatodani, Wiro M. B. P. Menge, Henk Timmerman, Timothy W. Lovenberg and Rob Leurs

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 908-914;
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Inhibition of Rat C6 Glioma Cell Proliferation by Endogenous and Synthetic Cannabinoids. Relative Involvement of Cannabinoid and Vanilloid Receptors
Stig O. P. Jacobsson, Thomas Wallin and Christopher J. Fowler

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 951-959;
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Kinetics of Modulation of Tetrodotoxin-Sensitive and Tetrodotoxin-Resistant Sodium Channels by Tetramethrin and Deltamethrin
Iustin V. Tabarean and Toshio Narahashi

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 988-997;
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Similar Apparent Constitutive Activity of Human Histamine H₂-Receptor Fused to Long and Short Splice Variants of G_sα
Katharina Wenzel-Seifert, Melissa T. Kelley, Armin Buschauer and Roland Seifert

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1013-1020;

CHEMOTHERAPY, ANTIBIOTICS, AND GENE THERAPY

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Model for Time Dependency of Cytotoxic Effect of CHS 828 in Vitro Suggests Two Different Mechanisms of Action
Saadia B. Hassan, Elin Jonsson, Rolf Larsson and Mats O. Karlsson

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1140-1147;
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CI-988 Inhibits Growth of Small Cell Lung Cancer Cells
Terry W. Moody and Robert T. Jensen

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1154-1160;

ENDOCRINE AND REPRODUCTIVE

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Increase in Neurokinin B Expression and in Tachykinin NK₃ Receptor-Mediated Response and Expression in the Rat Uterus with Age
Cristina G. Cintado, Francisco M. Pinto, Philippe Devillier, Angel Merida and M. Luz Candenas

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 934-938;
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2-Hydroxyestradiol Attenuates the Development of Obesity, the Metabolic Syndrome, and Vascular and Renal Dysfunction in Obese ZSF1 Rats
Stevan P. Tofovic, Raghvendra K. Dubey and Edwin K. Jackson

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 973-977;

GASTROINTESTINAL, HEPATIC, PULMONARY, AND RENAL

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Cyclosporin A Causes a Hypermetabolic State and Hypoxia in the Liver: Prevention by Dietary Glycine
Zhi Zhong, Xiangli Li, Shunhei Yamashina, Moritz von Frankenberg, Nobuyuki Enomoto, Kenichi Ikejima, Monica Kolinsky, James A. Raleigh and Ronald G. Thurman

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 858-865;
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Bid Antisense Attenuates Bile Acid-Induced Apoptosis and Cholestatic Liver Injury
Hajime Higuchi, Hideyuki Miyoshi, Steven F. Bronk, Hong Zhang, Nicholas Dean and Gregory J. Gores

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 866-873;
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Sodium Salicylate Inhibits Prostaglandin Formation without Affecting the Induction of Cyclooxygenase-2 by Bacterial Lipopolysaccharide in Vivo
Francesco Giuliano, Jane A. Mitchell and Timothy D. Warner

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 894-900;
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Evidence for the Interaction between Nitric Oxide and Vasoactive Intestinal Polypeptide in the Mouse Gastric Fundus
Yusuf Ergün and Nuran Öğülener

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 945-950;
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A₁ Receptor Blockade Induces Natriuresis with a Favorable Renal Hemodynamic Profile in SHHF/Mcc-fa^cp Rats Chronically Treated with Salt and Furosemide
Edwin K. Jackson, Curtis K. Kost, William A. Herzer, Glenn J. Smits and Stevan P. Tofovic

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 978-987;
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N-[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]-N-(2-nitrophenyl) Cyclohexanecarboxamide: A Novel Pre- and Postsynaptic 5-Hydroxytryptamine_1A Receptor Antagonist Active on the Lower Urinary Tract
A. Leonardi, L. Guarneri, E. Poggesi, P. Angelico, C. Velasco, A. Cilia and R. Testa

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1027-1037;
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Acetylcholine-Induced Desensitization of Muscarinic Contractile Response in Guinea Pig Ileum Is Inhibited by Pertussis Toxin Treatment
Frederick J. Ehlert, Khurram Z. Ansari, Darakhshanda Shehnaz, Gregory W. Sawyer and Michael T. Griffin

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1126-1132;

INFLAMMATION AND IMMUNOPHARMACOLOGY

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Caffeic Acid Phenethyl Ester, an Inhibitor of Nuclear Factor-κB, Attenuates Bacterial Peptidoglycan Polysaccharide-Induced Colitis in Rats
Leo R. Fitzpatrick, Jian Wang and Truc Le

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 915-920;
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Pregabalin Enhances Nonrapid Eye Movement Sleep
Takeshi Kubota, Jidong Fang, Leonard T. Meltzer and James M. Krueger

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1095-1105;

NEUROPHARMACOLOGY

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Colocalization of μ-Opioid Receptors and Activated G-Proteins in Rat Cingulate Cortex
Leslie J. Vogt, Laura J. Sim-Selley, Steven R. Childers, Ronald G. Wiley and Brent A. Vogt

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 840-848;
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The Pharmacological Profile of (R)-3,4-Dihydro-N-isopropyl-3-(N-isopropyl-N-propylamino)-2H-1-benzopyran-5-carboxamide, a Selective 5-Hydroxytryptamine_1A Receptor Agonist
Lucy Rënyi, John L. Evenden, Christopher J. Fowler, Eva Jerning, Diana Kelder, Desmond Lake-Bakaar, Lars-Gunnar Larsson, Nina Mohell, Maria Sällemark and Svante B. Ross

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 883-893;
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α2A-Adrenoceptor Stimulation Reduces Capsaicin-Induced Glutamate Release from Spinal Cord Synaptosomes
Xinhui Li and James C. Eisenach

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 939-944;
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M2 Muscarinic Autoreceptors Modulate Acetylcholine Release in Prefrontal Cortex of C57BL/6J Mouse
Christopher L. Douglas, Helen A. Baghdoyan and Ralph Lydic

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 960-966;
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Local Anesthetics Noncompetitively Inhibit Function of Four Distinct Nicotinic Acetylcholine Receptor Subtypes
Cynthia L. Gentry and Ronald J. Lukas

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1038-1048;
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Effects of Infusion Rate of Intravenously Administered Morphine on Physiological, Psychomotor, and Self-Reported Measures in Humans
Lisa A. Marsch, Warren K. Bickel, Gary J. Badger, James P. Rathmell, Michael D. B. Swedberg, Bror Jonzon and Carina Norsten-Höög

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1056-1065;
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Selective and Divergent Regulation of Cortical 5-HT_2AReceptors in Rabbit
Vincent J. Aloyo, Kuldip D. Dave, Tariq Rahman and John A. Harvey

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1066-1072;
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Inhibitory Presynaptic 5-Hydroxytryptamine_2AReceptors Regulate Evoked Glutamate Release from Rat Cerebellar Mossy Fibers
Manuela Marcoli, Christian Rosu, Andrea Bonfanti, Maurizio Raiteri and Guido Maura

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1106-1111;
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Benzylidene Analogs of Anabaseine Display Partial Agonist and Antagonist Properties at the Mouse 5-Hydroxytryptamine_3AReceptor
Tina K. Machu, Margaret E. Hamilton, Tonia F. Frye, Christopher L. Shanklin, Michael C. Harris, Hongwei Sun, Thomas E. Tenner, Ferenc S. Soti and William R. Kem

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1112-1119;
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Acute Antinociceptive Tolerance and Asymmetric Cross-Tolerance between Endomorphin-1 and Endomorphin-2 Given Intracerebroventricularly in the Mouse
Hsiang-en Wu, Kuei-chun Hung, Hirokazu Mizoguchi, James M. Fujimoto and Leon F. Tseng

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1120-1125;
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Binding Characteristics of the γ-Hydroxybutyric Acid Receptor Antagonist [³H](2E)-(5-Hydroxy-5,7,8,9-tetrahydro-6H-benzo[a][7]annulen-6-ylidene) Ethanoic Acid in the Rat Brain
Ashok K. Mehta, Nicole M. Muschaweck, Dean Y. Maeda, Andrew Coop and Maharaj K. Ticku

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1148-1153;
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Insights into the Mechanisms of Ifosfamide Encephalopathy: Drug Metabolites Have Agonistic Effects on α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA)/Kainate Receptors and Induce Cellular Acidification in Mouse Cortical Neurons
Jean-Yves Chatton, Jeffrey R. Idle, Cathrine Broberg Vågbø and Pierre J. Magistretti

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1161-1168;

TOXICOLOGY

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Arginine Reverses Ethanol-Induced Inflammatory and Fibrotic Changes in Liver Despite Continued Ethanol Administration
Amin A. Nanji, Kalle Jokelainen, George K. K. Lau, Amir Rahemtulla, George L. Tipoe, Rathnagiri Polavarapu and El-Nasir Lalani

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 832-839;
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Midazolam Is a Phenobarbital-Like Cytochrome P450 Inducer in Rats
Peter A. C. 't Hoen, Martin K. Bijsterbosch, Theo J. C. van Berkel, Nico P. E. Vermeulen and Jan N. M. Commandeur

Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 921-927;

Erratum

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Correction to “A Pharmacodynamic Analysis of Erythropoietin-Stimulated Reticulocyte Response in Phlebotomized Sheep”
Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1169;

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Table of Contents

PERSPECTIVES IN PHARMACOLOGY

ABSORPTION, DISTRIBUTION, METABOLISM, AND EXCRETION

BEHAVIORAL PHARMACOLOGY

CARDIOVASCULAR

CELLULAR AND MOLECULAR

CHEMOTHERAPY, ANTIBIOTICS, AND GENE THERAPY

ENDOCRINE AND REPRODUCTIVE

GASTROINTESTINAL, HEPATIC, PULMONARY, AND RENAL

INFLAMMATION AND IMMUNOPHARMACOLOGY

NEUROPHARMACOLOGY

TOXICOLOGY

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