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Journal of Pharmacology and Experimental Therapeutics

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Table of Contents

December 01, 2001; Volume 299,Issue 3

PERSPECTIVES IN PHARMACOLOGY

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    Pharmacology of Opioid and Nonopioid Analgesics in Chronic Pain States
    Thomas J. Martin and James C. Eisenach
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 811-817;
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    Post-Translational Control of Endothelial Nitric Oxide Synthase: Why Isn't Calcium/Calmodulin Enough?
    David Fulton, Jean-Philippe Gratton and William C. Sessa
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 818-824;

ABSORPTION, DISTRIBUTION, METABOLISM, AND EXCRETION

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    Identification of Variants of CYP3A4 and Characterization of Their Abilities to Metabolize Testosterone and Chlorpyrifos
    Diana Dai, Jun Tang, Randy Rose, Ernest Hodgson, Rachelle J. Bienstock, Harvey W. Mohrenweiser and Joyce A. Goldstein
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 825-831;
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    Rifampin Is a Selective, Pleiotropic Inducer of Drug Metabolism Genes in Human Hepatocytes: Studies with cDNA and Oligonucleotide Expression Arrays
    James M. Rae, Michael D. Johnson, Marc E. Lippman and David A. Flockhart
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 849-857;
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    Differential Inhibition and Inactivation of Human CYP1 Enzymes bytrans-Resveratrol: Evidence for Mechanism-Based Inactivation of CYP1A2
    Thomas K. H. Chang, Jie Chen and Wendy B. K. Lee
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 874-882;
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    Improved Blood-Brain Barrier Penetration and Enhanced Analgesia of an Opioid Peptide by Glycosylation
    R. D. Egleton, S. A. Mitchell, J. D. Huber, M. M. Palian, R. Polt and T. P. Davis
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 967-972;
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    Interindividual Variability in Acetaminophen Glucuronidation by Human Liver Microsomes: Identification of Relevant Acetaminophen UDP-Glucuronosyltransferase Isoforms
    Michael H. Court, Su X. Duan, Lisa L. von Moltke, David J. Greenblatt, Christopher J. Patten, John O. Miners and Peter I. Mackenzie
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 998-1006;

BEHAVIORAL PHARMACOLOGY

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    Multiple Behavioral Effects of Cocaine- and Amphetamine-Regulated Transcript (CART) Peptides in Mice: CART 42–89 and CART 49–89 Differ in Potency and Activity
    Anthony W. Bannon, Jennifer Seda, Michelle Carmouche, Jonathan M. Francis, Mark A. Jarosinski and James Douglass
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1021-1026;

CARDIOVASCULAR

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    An Up-Regulation of Renal α2A-Adrenoceptors Is Associated with Resistance to Salt-Induced Hypertension in Sabra Rats
    Mostafa Khalid, Yves Giudicelli and Jean-Pierre Dausse
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 928-933;
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    Gastrointestinal Prokinetic Drugs have Different Affinity for the Human Cardiac Human Ether-à-gogo K+ Channel
    Franck Potet, Thierry Bouyssou, Denis Escande and Isabelle Baró
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1007-1012;
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    Interaction of the Sulfonylthiourea HMR 1833 with Sulfonylurea Receptors and Recombinant ATP-Sensitive K+ Channels: Comparison with Glibenclamide
    Ulrich Russ, Ulf Lange, Cornelia Löffler-Walz, Annette Hambrock and Ulrich Quast
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1049-1055;
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    Vascular Endothelial Growth Factor (VEGF) Receptor-2 Antagonists Inhibit VEGF- and Basic Fibroblast Growth Factor-Induced Angiogenesis in Vivo and in Vitro
    J.-C. Tille, J. Wood, S.J. Mandriota, C. Schnell, S. Ferrari, J. Mestan, Z. Zhu, L. Witte and M. S. Pepper
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1073-1085;
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    Functional Calcitonin Gene-Related Peptide Subtype 2 Receptors in Porcine Coronary Arteries Are Identified as Calcitonin Gene-Related Peptide Subtype 1 Receptors by Radioligand Binding and Reverse Transcription-Polymerase Chain Reaction
    Boyd R. Rorabaugh, Margaret A. Scofield, D. David Smith, William B. Jeffries and Peter W. Abel
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1086-1094;
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    Effects of Heart Rate Reduction with Ivabradine on Exercise-Induced Myocardial Ischemia and Stunning
    Xavier Monnet, Bijan Ghaleh, Patrice Colin, Olivier Parent de Curzon, Jean-François Giudicelli and Alain Berdeaux
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1133-1139;

CELLULAR AND MOLECULAR

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    Ca2+ Influx through Nonselective Cation Channels Plays an Essential Role in Noradrenaline-Induced Arachidonic Acid Release in Chinese Hamster Ovary Cells Expressing α1A-, α1B-, or α1D-Adrenergic Receptors
    Yoshifumi Kawanabe, Nobuo Hashimoto, Tomoh Masaki and Soichi Miwa
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 901-907;
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    Constitutive Activity of Histamine H3 Receptors Stably Expressed in SK-N-MC Cells: Display of Agonism and Inverse Agonism by H3 Antagonists
    Kerstin Wieland, Gerold Bongers, Yumiko Yamamoto, Takeshi Hashimoto, Atsushi Yamatodani, Wiro M. B. P. Menge, Henk Timmerman, Timothy W. Lovenberg and Rob Leurs
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 908-914;
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    Inhibition of Rat C6 Glioma Cell Proliferation by Endogenous and Synthetic Cannabinoids. Relative Involvement of Cannabinoid and Vanilloid Receptors
    Stig O. P. Jacobsson, Thomas Wallin and Christopher J. Fowler
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 951-959;
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    Kinetics of Modulation of Tetrodotoxin-Sensitive and Tetrodotoxin-Resistant Sodium Channels by Tetramethrin and Deltamethrin
    Iustin V. Tabarean and Toshio Narahashi
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 988-997;
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    Similar Apparent Constitutive Activity of Human Histamine H2-Receptor Fused to Long and Short Splice Variants of Gsα
    Katharina Wenzel-Seifert, Melissa T. Kelley, Armin Buschauer and Roland Seifert
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1013-1020;

CHEMOTHERAPY, ANTIBIOTICS, AND GENE THERAPY

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    Model for Time Dependency of Cytotoxic Effect of CHS 828 in Vitro Suggests Two Different Mechanisms of Action
    Saadia B. Hassan, Elin Jonsson, Rolf Larsson and Mats O. Karlsson
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1140-1147;
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    CI-988 Inhibits Growth of Small Cell Lung Cancer Cells
    Terry W. Moody and Robert T. Jensen
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1154-1160;

ENDOCRINE AND REPRODUCTIVE

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    Increase in Neurokinin B Expression and in Tachykinin NK3 Receptor-Mediated Response and Expression in the Rat Uterus with Age
    Cristina G. Cintado, Francisco M. Pinto, Philippe Devillier, Angel Merida and M. Luz Candenas
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 934-938;
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    2-Hydroxyestradiol Attenuates the Development of Obesity, the Metabolic Syndrome, and Vascular and Renal Dysfunction in Obese ZSF1 Rats
    Stevan P. Tofovic, Raghvendra K. Dubey and Edwin K. Jackson
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 973-977;

GASTROINTESTINAL, HEPATIC, PULMONARY, AND RENAL

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    Cyclosporin A Causes a Hypermetabolic State and Hypoxia in the Liver: Prevention by Dietary Glycine
    Zhi Zhong, Xiangli Li, Shunhei Yamashina, Moritz von Frankenberg, Nobuyuki Enomoto, Kenichi Ikejima, Monica Kolinsky, James A. Raleigh and Ronald G. Thurman
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 858-865;
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    Bid Antisense Attenuates Bile Acid-Induced Apoptosis and Cholestatic Liver Injury
    Hajime Higuchi, Hideyuki Miyoshi, Steven F. Bronk, Hong Zhang, Nicholas Dean and Gregory J. Gores
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 866-873;
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    Sodium Salicylate Inhibits Prostaglandin Formation without Affecting the Induction of Cyclooxygenase-2 by Bacterial Lipopolysaccharide in Vivo
    Francesco Giuliano, Jane A. Mitchell and Timothy D. Warner
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 894-900;
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    Evidence for the Interaction between Nitric Oxide and Vasoactive Intestinal Polypeptide in the Mouse Gastric Fundus
    Yusuf Ergün and Nuran Öğülener
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 945-950;
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    A1 Receptor Blockade Induces Natriuresis with a Favorable Renal Hemodynamic Profile in SHHF/Mcc-facp Rats Chronically Treated with Salt and Furosemide
    Edwin K. Jackson, Curtis K. Kost, William A. Herzer, Glenn J. Smits and Stevan P. Tofovic
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 978-987;
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    N-[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]-N-(2-nitrophenyl) Cyclohexanecarboxamide: A Novel Pre- and Postsynaptic 5-Hydroxytryptamine1A Receptor Antagonist Active on the Lower Urinary Tract
    A. Leonardi, L. Guarneri, E. Poggesi, P. Angelico, C. Velasco, A. Cilia and R. Testa
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1027-1037;
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    Acetylcholine-Induced Desensitization of Muscarinic Contractile Response in Guinea Pig Ileum Is Inhibited by Pertussis Toxin Treatment
    Frederick J. Ehlert, Khurram Z. Ansari, Darakhshanda Shehnaz, Gregory W. Sawyer and Michael T. Griffin
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1126-1132;

INFLAMMATION AND IMMUNOPHARMACOLOGY

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    Caffeic Acid Phenethyl Ester, an Inhibitor of Nuclear Factor-κB, Attenuates Bacterial Peptidoglycan Polysaccharide-Induced Colitis in Rats
    Leo R. Fitzpatrick, Jian Wang and Truc Le
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 915-920;
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    Pregabalin Enhances Nonrapid Eye Movement Sleep
    Takeshi Kubota, Jidong Fang, Leonard T. Meltzer and James M. Krueger
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1095-1105;

NEUROPHARMACOLOGY

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    Colocalization of μ-Opioid Receptors and Activated G-Proteins in Rat Cingulate Cortex
    Leslie J. Vogt, Laura J. Sim-Selley, Steven R. Childers, Ronald G. Wiley and Brent A. Vogt
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 840-848;
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    The Pharmacological Profile of (R)-3,4-Dihydro-N-isopropyl-3-(N-isopropyl-N-propylamino)-2H-1-benzopyran-5-carboxamide, a Selective 5-Hydroxytryptamine1A Receptor Agonist
    Lucy Rënyi, John L. Evenden, Christopher J. Fowler, Eva Jerning, Diana Kelder, Desmond Lake-Bakaar, Lars-Gunnar Larsson, Nina Mohell, Maria Sällemark and Svante B. Ross
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 883-893;
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    α2A-Adrenoceptor Stimulation Reduces Capsaicin-Induced Glutamate Release from Spinal Cord Synaptosomes
    Xinhui Li and James C. Eisenach
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 939-944;
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    M2 Muscarinic Autoreceptors Modulate Acetylcholine Release in Prefrontal Cortex of C57BL/6J Mouse
    Christopher L. Douglas, Helen A. Baghdoyan and Ralph Lydic
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 960-966;
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    Local Anesthetics Noncompetitively Inhibit Function of Four Distinct Nicotinic Acetylcholine Receptor Subtypes
    Cynthia L. Gentry and Ronald J. Lukas
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1038-1048;
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    Effects of Infusion Rate of Intravenously Administered Morphine on Physiological, Psychomotor, and Self-Reported Measures in Humans
    Lisa A. Marsch, Warren K. Bickel, Gary J. Badger, James P. Rathmell, Michael D. B. Swedberg, Bror Jonzon and Carina Norsten-Höög
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1056-1065;
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    Selective and Divergent Regulation of Cortical 5-HT2AReceptors in Rabbit
    Vincent J. Aloyo, Kuldip D. Dave, Tariq Rahman and John A. Harvey
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1066-1072;
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    Inhibitory Presynaptic 5-Hydroxytryptamine2AReceptors Regulate Evoked Glutamate Release from Rat Cerebellar Mossy Fibers
    Manuela Marcoli, Christian Rosu, Andrea Bonfanti, Maurizio Raiteri and Guido Maura
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1106-1111;
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    Benzylidene Analogs of Anabaseine Display Partial Agonist and Antagonist Properties at the Mouse 5-Hydroxytryptamine3AReceptor
    Tina K. Machu, Margaret E. Hamilton, Tonia F. Frye, Christopher L. Shanklin, Michael C. Harris, Hongwei Sun, Thomas E. Tenner, Ferenc S. Soti and William R. Kem
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1112-1119;
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    Acute Antinociceptive Tolerance and Asymmetric Cross-Tolerance between Endomorphin-1 and Endomorphin-2 Given Intracerebroventricularly in the Mouse
    Hsiang-en Wu, Kuei-chun Hung, Hirokazu Mizoguchi, James M. Fujimoto and Leon F. Tseng
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1120-1125;
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    Binding Characteristics of the γ-Hydroxybutyric Acid Receptor Antagonist [3H](2E)-(5-Hydroxy-5,7,8,9-tetrahydro-6H-benzo[a][7]annulen-6-ylidene) Ethanoic Acid in the Rat Brain
    Ashok K. Mehta, Nicole M. Muschaweck, Dean Y. Maeda, Andrew Coop and Maharaj K. Ticku
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1148-1153;
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    Insights into the Mechanisms of Ifosfamide Encephalopathy: Drug Metabolites Have Agonistic Effects on α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA)/Kainate Receptors and Induce Cellular Acidification in Mouse Cortical Neurons
    Jean-Yves Chatton, Jeffrey R. Idle, Cathrine Broberg Vågbø and Pierre J. Magistretti
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1161-1168;

TOXICOLOGY

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    Arginine Reverses Ethanol-Induced Inflammatory and Fibrotic Changes in Liver Despite Continued Ethanol Administration
    Amin A. Nanji, Kalle Jokelainen, George K. K. Lau, Amir Rahemtulla, George L. Tipoe, Rathnagiri Polavarapu and El-Nasir Lalani
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 832-839;
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    Midazolam Is a Phenobarbital-Like Cytochrome P450 Inducer in Rats
    Peter A. C. 't Hoen, Martin K. Bijsterbosch, Theo J. C. van Berkel, Nico P. E. Vermeulen and Jan N. M. Commandeur
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 921-927;

Erratum

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    Correction to “A Pharmacodynamic Analysis of Erythropoietin-Stimulated Reticulocyte Response in Phlebotomized Sheep”
    Journal of Pharmacology and Experimental Therapeutics December 2001, 299 (3) 1169;
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Journal of Pharmacology and Experimental Therapeutics: 299 (3)
Journal of Pharmacology and Experimental Therapeutics
Vol. 299, Issue 3
1 Dec 2001
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  • PERSPECTIVES IN PHARMACOLOGY
  • ABSORPTION, DISTRIBUTION, METABOLISM, AND EXCRETION
  • BEHAVIORAL PHARMACOLOGY
  • CARDIOVASCULAR
  • CELLULAR AND MOLECULAR
  • CHEMOTHERAPY, ANTIBIOTICS, AND GENE THERAPY
  • ENDOCRINE AND REPRODUCTIVE
  • GASTROINTESTINAL, HEPATIC, PULMONARY, AND RENAL
  • INFLAMMATION AND IMMUNOPHARMACOLOGY
  • NEUROPHARMACOLOGY
  • TOXICOLOGY
  • Erratum
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  • Interindividual variations in human liver cytochrome P-450 enzymes involved in the oxidation of drugs, carcinogens and toxic chemicals: studies with liver microsomes of 30 Japanese and 30 Caucasians.
  • Functional Selectivity and Classical Concepts of Quantitative Pharmacology
  • Abl Protein-Tyrosine Kinase Inhibitor STI571 Inhibits In Vitro Signal Transduction Mediated by c-Kit and Platelet-Derived Growth Factor Receptors
  • The Prediction of Human Pharmacokinetic Parameters from Preclinical and In Vitro Metabolism Data
  • A METHOD FOR DETERMINING LOSS OF PAIN SENSATION
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