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Journal of Pharmacology and Experimental Therapeutics

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Table of Contents

October 01, 2001; Volume 299,Issue 1

PERSPECTIVES IN PHARMACOLOGY

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    Transgenic Studies of Cardiac Adrenergic Receptor Regulation
    Andrea D. Eckhart and Walter J. Koch
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 1-5;
  • You have access
    Mechanisms of Induction of Persistent Nociception by Dynorphin
    Tinna M. Laughlin, Alice A. Larson and George L. Wilcox
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 6-11;
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    Unveiling the Functions of Presynaptic Metabotropic Glutamate Receptors in the Central Nervous System
    Darryle D. Schoepp
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 12-20;

ABSORPTION, DISTRIBUTION, METABOLISM, AND EXCRETION

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    Preclinical Studies to Predict the Disposition of Apo2L/Tumor Necrosis Factor-Related Apoptosis-Inducing Ligand in Humans: Characterization of in Vivo Efficacy, Pharmacokinetics, and Safety
    Sean K. Kelley, Louise A. Harris, David Xie, Laura DeForge, Klara Totpal, Jeanine Bussiere and Judith A. Fox
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 31-38;
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    Identification and Localization of Five CYP2Cs in Murine Extrahepatic Tissues and Their Metabolism of Arachidonic Acid to Regio- and Stereoselective Products
    Cheng-Chung Tsao, Sherry J. Coulter, Anna Chien, Gang Luo, Natasha P. Clayton, Robert Maronpot, Joyce A. Goldstein and Darryl C. Zeldin
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 39-47;
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    Multispecific Substrate Recognition of Kidney-Specific Organic Anion Transporters OAT-K1 and OAT-K2
    Ayako Takeuchi, Satohiro Masuda, Hideyuki Saito, Takaaki Abe and Ken-ichi Inui
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 261-267;
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    Flavonoids with Epidermal Growth Factor-Receptor Tyrosine Kinase Inhibitory Activity Stimulate PEPT1-Mediated Cefixime Uptake into Human Intestinal Epithelial Cells
    Uwe Wenzel, Sabine Kuntz and Hannelore Daniel
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 351-357;
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    Functional Characteristics and Steroid Hormone-Mediated Regulation of an Organic Cation Transporter in Madin-Darby Canine Kidney Cells
    Yan Shu, Carlo L. Bello, Lara M. Mangravite, Bo Feng and Kathleen M. Giacomini
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 392-398;

CARDIOVASCULAR

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    N,N′-Diacetyl-l-cystine (DiNAC), the Disulphide Dimer of N-Acetylcysteine, Inhibits Atherosclerosis in WHHL Rabbits: Evidence for Immunomodulatory Agents as a New Approach to Prevent Atherosclerosis
    Maria Wågberg, Anne-Heléne Jansson, Christer Westerlund, Ann-Margret Östlund-Lindqvist, Bengt Särnstrand, Håkan Bergstrand and Knut Pettersson
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 76-82;
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    Effects of Cocaine and Its Major Metabolites on the HERG-Encoded Potassium Channel
    Scott Ferreira, William J. Crumb, Carol G. Carlton and Craig W. Clarkson
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 220-226;
  • You have access
    Interactions of the Antimalarial Drug Mefloquine with the Human Cardiac Potassium Channels KvLQT1/minK and HERG
    Jiesheng Kang, Xiao-Liang Chen, Lin Wang and David Rampe
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 290-296;
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    Inhibition of Ca2+-Induced Relaxation by Oxidized Tungsten Wires and Paratungstate
    Richard D. Bukoski, Simoneque Shearin, William F. Jackson and Mohan F. Pamarthi
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 343-350;
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    Differential Effects of U46619 on Renal Regional Hemodynamics in the Rat: Involvement of Endothelin
    Hercule Hantz, Ajayi Adesuyi and Oyekan Adebayo
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 372-376;

CELLULAR AND MOLECULAR

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    Neuronal Apoptosis Resulting from High Doses of the Isoflavone Genistein: Role for Calcium and P42/44 Mitogen-Activated Protein Kinase
    Nancy J. Linford, Yaxiong Yang, David G. Cook and Daniel M. Dorsa
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 67-75;
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    Dual Action of Octopamine on Glucose Transport into Adipocytes: Inhibition via β3-Adrenoceptor Activation and Stimulation via Oxidation by Amine Oxidases
    Virgile Visentin, Nathalie Morin, Emi Fontana, Danielle Prévot, Jeremie Boucher, Isabelle Castan, Philippe Valet, Danica Grujic and Christian Carpéné
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 96-104;
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    SLC-1 Receptor Mediates Effect of Melanin-Concentrating Hormone on Feeding Behavior in Rat: A Structure-Activity Study
    Thomas Suply, Odile Della Zuana, Valérie Audinot, Marianne Rodriguez, Philippe Beauverger, Jacques Duhault, Emmanuel Canet, Jean-Pierre Galizzi, Jean-Louis Nahon, Nigel Levens and Jean A. Boutin
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 137-146;
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    Activation of p42/p44 Mitogen-Activated Protein Kinase and Contraction by Prostaglandin F2α, Ionomycin, and Thapsigargin in Cat Iris Sphincter Smooth Muscle: Inhibition by PD98059, KN-93, and Isoproterenol
    Habib R. Ansari, Shahid Husain and Ata A. Abdel-Latif
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 178-186;
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    Calcilytic Compounds: Potent and Selective Ca2+Receptor Antagonists That Stimulate Secretion of Parathyroid Hormone
    Edward F. Nemeth, Eric G. Delmar, William L. Heaton, Michael A. Miller, Lyssa D. Lambert, Rebecca L. Conklin, Maxine Gowen, John G. Gleason, Pradip K. Bhatnagar and John Fox
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 323-331;
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    Determinants of Agonist Binding Affinity on Neuronal Nicotinic Receptor β Subunits
    Michael J. Parker, Scott C. Harvey and Charles W. Luetje
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 385-391;

GASTROINTESTINAL, HEPATIC, PULMONARY, AND RENAL

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    Recombinant Human Interleukin-11 Restores Smooth Muscle Function in the Jejunum and Colon of Human Leukocyte Antigen-B27 Rats with Intestinal Inflammation
    Beverley Greenwood-Van Meerveld, Kalina Venkova and James C. Keith
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 58-66;
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    Nizatidine Enhances the Gastrocolonic Response and the Colonic Peristaltic Reflex in Humans
    Wei Ming Sun, William L. Hasler, Han-Chung Lien, Jared Montague and Chung Owyang
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 159-163;
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    Correlation of Gene Expression of Ten Drug Efflux Proteins of the ATP-Binding Cassette Transporter Family in Normal Human Jejunum and in Human Intestinal Epithelial Caco-2 Cell Monolayers
    Jan Taipalensuu, Hans Törnblom, Greger Lindberg, Curt Einarsson, Folke Sjöqvist, Håkan Melhus, Per Garberg, Brita Sjöström, Bo Lundgren and Per Artursson
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 164-170;
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    Nepadutant Pharmacokinetics and Dose-Effect Relationships as Tachykinin NK2 Receptor Antagonist Are Altered by Intestinal Inflammation in Rodent Models
    Alessandro Lecci, Francesca Carini, Manuela Tramontana, Vincenzo D'Aranno, Erica Marinoni, Attilio Crea, Lionel Bueno, Jean Fioramonti, Marco Criscuoli, Sandro Giuliani and Carlo Alberto Maggi
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 247-254;
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    Role of Sodium Depletion in Acute Antidiuretic Effect of Bendroflumethiazide in Rats with Nephrogenic Diabetes Insipidus
    Nadeem R. Janjua, Thomas E. N. Jonassen, Susanna Langhoff, Klaus Thomsen and Sten Christensen
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 307-313;

INFLAMMATION AND IMMUNOPHARMACOLOGY

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    Nonpeptide CXCR2 Antagonist Prevents Neutrophil Accumulation in Hyperoxia-Exposed Newborn Rats
    Richard L. Auten, Ricardo M. Richardson, John R. White, S. Nicholas Mason, Michael A. Vozzelli and Mary H. Whorton
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 90-95;
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    Comparison of Human, Mouse, Rat, and Guinea Pig Histamine H4 Receptors Reveals Substantial Pharmacological Species Variation
    Changlu Liu, Sandy J. Wilson, Chester Kuei and Timothy W. Lovenberg
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 121-130;
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    Identification and Characterization of a Novel Class of Interleukin-1 Post-Translational Processing Inhibitors
    David G. Perregaux, Patricia McNiff, Ronald Laliberte, Natalie Hawryluk, Heather Peurano, Ethan Stam, Jim Eggler, Richard Griffiths, Mark A. Dombroski and Christopher A. Gabel
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 187-197;
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    Peroxynitrite-Induced Nitrotyrosination of Proteins Is Blocked by Direct 5-Lipoxygenase Inhibitor Zileuton
    Michael J. Coffey, Susan M. Phare and Marc Peters-Golden
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 198-203;
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    Capsaicin Inhibits Jurkat T-Cell Activation by Blocking Calcium Entry Current ICRAC
    Bruce S. Fischer, Danmei Qin, Kami Kim and Thomas V. McDonald
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 238-246;
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    Inverse Agonist Activity of Selected Ligands of Platelet-Activating Factor Receptor
    Denis J. Dupré, Christian Le Gouill, Marek Rola-Pleszczynski and Jana Staňková
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 358-365;

NEUROPHARMACOLOGY

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    The Noradrenergic Inhibition of an Apamin-Sensitive, Small-Conductance Ca2+-Activated K+ Channel in Hypothalamic γ-Aminobutyric Acid Neurons: Pharmacology, Estrogen Sensitivity, and Relevance to the Control of the Reproductive Axis
    Edward J. Wagner, Oline K. Rønnekleiv and Martin J. Kelly
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 21-30;
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    Electroencephalogram Analysis and Neuroprotective Profile of theN-Acetylated-α-Linked Acidic Dipeptidase Inhibitor, GPI5232, in Normal and Brain-Injured Rats ,
    A. J. Williams, X. M. Lu, B. Slusher and F. C. Tortella
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 48-57;
  • You have access
    Inverse Agonist Actions of Typical and Atypical Antipsychotic Drugs at the Human 5-Hydroxytryptamine2C Receptor
    Laura Rauser, Jason E. Savage, Herbert Y. Meltzer and Bryan L. Roth
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 83-89;
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    Combinations of Neurokinin Receptor Antagonists Reduce Visceral Hyperalgesia
    Elizabeth H. Kamp, Daniel R. Beck and G. F. Gebhart
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 105-113;
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    Effects of Saline Substitution on Responding and Plasma Corticosterone in Rats Trained to Self-Administer Different Doses of Cocaine
    Rachel L. Peltier, Glenn F. Guerin, Nandakumar Dorairaj and Nick E. Goeders
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 114-120;
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    Selective Agonism of Group I P2X Receptors by Dinucleotides Dependent on a Single Adenine Moiety
    Okan Cinkilic, Brian F. King, Markus van der Giet, Hartmut Schlüter, Walter Zidek and Geoffrey Burnstock
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 131-136;
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    Enadoline and Butorphanol: Evaluation of κ-Agonists on Cocaine Pharmacodynamics and Cocaine Self-Administration in Humans
    Sharon L. Walsh, Beth Geter-Douglas, Eric C. Strain and George E. Bigelow
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 147-158;
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    Nanomolar Concentrations of Tri-n-butyltin Facilitate γ-Aminobutyric Acidergic Synaptic Transmission in Rat Hypothalamic Neurons
    Kiyonori Kishimoto, Shin-Ichiro Matsuo, Yumiko Kanemoto, Hitoshi Ishibashi, Yasuo Oyama and Norio Akaike
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 171-177;
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    Functional Expression of P-glycoprotein in Rat Brain Microglia
    Gloria Lee, Lyanne Schlichter, Moise Bendayan and Reina Bendayan
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 204-212;
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    Pronociceptive Effects of Nociceptin/Orphanin FQ (13–17) at Peripheral and Spinal Level in Mice
    Makoto Inoue, Shinobu Matsunaga, M. Harunor Rashid, Akira Yoshida, Kiyonobu Mizuno, Tsukasa Sakurada, Hiroshi Takeshima and Hiroshi Ueda
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 213-219;
  • You have access
    Neuroprotective Agent Riluzole Dramatically Slows Inactivation of Kv1.4 Potassium Channels by a Voltage-Dependent Oxidative Mechanism
    Lin Xu, Judith A. Enyeart and John J. Enyeart
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 227-237;
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    Inhibition by Tramadol of Muscarinic Receptor-Induced Responses in Cultured Adrenal Medullary Cells and in Xenopus laevis Oocytes Expressing Cloned M1Receptors
    Munehiro Shiraishi, Kouichiro Minami, Yasuhito Uezono, Nobuyuki Yanagihara and Akio Shigematsu
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 255-260;
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    5-Hydroxytryptamine2A Receptor Inverse Agonists as Antipsychotics
    D. M. Weiner, E. S. Burstein, N. Nash, G. E. Croston, E. A. Currier, K. E. Vanover, S. C. Harvey, E. Donohue, H. C. Hansen, C. M. Andersson, T. A. Spalding, D. F. C. Gibson, K. Krebs-Thomson, S. B. Powell, M. A. Geyer, U. Hacksell and M. R. Brann
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 268-276;
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    Bidirectional Changes in Ethanol Consumption in Rats with Site-Specific Antisense Down-Regulation of 5-Hydroxytryptamine2A Receptors in Brain
    Gregory G. Blakley, Larissa A. Pohorecky and Daniel Benjamin
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 277-289;
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    SIB-1553A, (±)-4-{[2-(1-Methyl-2-pyrrolidinyl)ethyl]thio}phenol Hydrochloride, a Subtype-Selective Ligand for Nicotinic Acetylcholine Receptors with Putative Cognitive-Enhancing Properties: Effects on Working and Reference Memory Performances in Aged Rodents and Nonhuman Primates
    Bruno Bontempi, Kevin T. Whelan, Victoria B. Risbrough, Tadimeti S. Rao, Jerry J. Buccafusco, G. Kenneth Lloyd and Frédérique Menzaghi
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 297-306;
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    RPR 119990, a Novel α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid Antagonist: Synthesis, Pharmacological Properties, and Activity in an Animal Model of Amyotrophic Lateral Sclerosis
    Thierry Canton, Georg Andrees Böhme, Alain Boireau, Françoise Bordier, Serge Mignani, Patrick Jimonet, Ghafoor Jahn, Mohammad Alavijeh, James Stygall, Simon Roberts, Clive Brealey, Marc Vuilhorgne, Marc-William Debono, Sylvain Le Guern, Michel Laville, Dominique Briet, Michel Roux, Jean-Marie Stutzmann and Jeremy Pratt
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 314-322;
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    Behavioral Evidence for the Interaction of Oleamide with Multiple Neurotransmitter Systems
    Irina Fedorova, Akihiro Hashimoto, Robert A. Fecik, Michael P. Hedrick, Lumı́r O. Hanuš, Dale L. Boger, Kenner C. Rice and Anthony S. Basile
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 332-342;
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    Blockade of Rat α3β4 Nicotinic Receptor Function by Methadone, Its Metabolites, and Structural Analogs
    Yingxian Xiao, Richard D. Smith, Frank S. Caruso and Kenneth J. Kellar
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 366-371;
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    Complestatin Is a Noncompetitive Peptide Antagonist of N-Methyl-d-aspartate and α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid/Kainate Receptors: Secure Blockade of Ischemic Neuronal Death
    So Young Seo, Bong-Sik Yun, In-Ja Ryoo, Jun-Sub Choi, Choun-Ki Joo, Su-Youne Chang, Jun-Mo Chung, Seikwan Oh, Byoung Joo Gwag and Ick Dong Yoo
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 377-384;

Erratum

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    Correction to “Actions of pyrethroid insecticides on sodium currents, action potentials, and contractile rhythm in isolated mammalian ventricular myocytes and perfused hearts”
    Journal of Pharmacology and Experimental Therapeutics October 2001, 299 (1) 399;
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Journal of Pharmacology and Experimental Therapeutics: 299 (1)
Journal of Pharmacology and Experimental Therapeutics
Vol. 299, Issue 1
1 Oct 2001
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  • INFLAMMATION AND IMMUNOPHARMACOLOGY
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