Dopamine transporter mutants, small molecules, and approaches to cocaine antagonist/dopamine transporter disinhibitor development

Methods Enzymol. 1998:296:456-65. doi: 10.1016/s0076-6879(98)96033-5.
No abstract available

Publication types

  • Research Support, U.S. Gov't, P.H.S.
  • Review

MeSH terms

  • Animals
  • Carrier Proteins / chemistry*
  • Carrier Proteins / genetics*
  • Carrier Proteins / metabolism
  • Cocaine / antagonists & inhibitors*
  • Cocaine / chemistry
  • Cocaine / pharmacokinetics*
  • Dopamine / metabolism
  • Dopamine Plasma Membrane Transport Proteins
  • Drug Design
  • Membrane Glycoproteins*
  • Membrane Transport Proteins*
  • Models, Molecular
  • Molecular Conformation
  • Mutagenesis, Site-Directed
  • Nerve Tissue Proteins*
  • Protein Conformation
  • Protein Structure, Secondary
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / metabolism
  • Structure-Activity Relationship
  • Transfection

Substances

  • Carrier Proteins
  • Dopamine Plasma Membrane Transport Proteins
  • Membrane Glycoproteins
  • Membrane Transport Proteins
  • Nerve Tissue Proteins
  • Recombinant Proteins
  • Cocaine
  • Dopamine