New bradykinin antagonists having very high potency at B1 receptors

Immunopharmacology. 1996 Jun;33(1-3):183-5. doi: 10.1016/0162-3109(96)00100-2.
No abstract available

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Aorta / drug effects
  • Aorta / physiology
  • Bradykinin / antagonists & inhibitors*
  • Bradykinin / chemistry
  • Bradykinin / metabolism
  • CHO Cells
  • Cell Line
  • Cricetinae
  • Guinea Pigs
  • Humans
  • Ileum / metabolism
  • In Vitro Techniques
  • Molecular Structure
  • Oligopeptides / chemistry
  • Oligopeptides / metabolism*
  • Oligopeptides / pharmacology*
  • Rabbits
  • Receptor, Bradykinin B1
  • Receptors, Bradykinin / metabolism*
  • Structure-Activity Relationship
  • Vasodilation / drug effects

Substances

  • Oligopeptides
  • Receptor, Bradykinin B1
  • Receptors, Bradykinin
  • Bradykinin