Anti-inflammatory effects of the novel phosphodiesterase IV inhibitor RP 73401

Int Arch Allergy Immunol. 1995 May-Jun;107(1-3):425-6. doi: 10.1159/000237066.
No abstract available

MeSH terms

  • 3',5'-Cyclic-AMP Phosphodiesterases*
  • Animals
  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology*
  • Aorta / enzymology
  • Benzamides / pharmacology*
  • Bronchial Spasm / drug therapy
  • Bronchial Spasm / prevention & control
  • Cyclic AMP / metabolism
  • Cyclic Nucleotide Phosphodiesterases, Type 4
  • Drug Evaluation, Preclinical
  • Eosinophils / enzymology
  • Eosinophils / metabolism
  • Granulocytes / drug effects
  • Granulocytes / enzymology
  • Guinea Pigs
  • Humans
  • Isoenzymes / antagonists & inhibitors
  • Leukotriene B4 / pharmacology
  • Phosphodiesterase Inhibitors / pharmacology*
  • Phosphoric Diester Hydrolases*
  • Pyridines / pharmacology*
  • Pyrrolidinones / pharmacology
  • Rolipram
  • Swine

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Benzamides
  • Isoenzymes
  • Phosphodiesterase Inhibitors
  • Pyridines
  • Pyrrolidinones
  • Leukotriene B4
  • Cyclic AMP
  • Phosphoric Diester Hydrolases
  • 3',5'-Cyclic-AMP Phosphodiesterases
  • Cyclic Nucleotide Phosphodiesterases, Type 4
  • Rolipram
  • piclamilast