p-fluoro-hexahydro-sila-difenidol: the first M2 beta-selective muscarinic antagonist

Eur J Pharmacol. 1988 Jul 26;152(1-2):193-4. doi: 10.1016/0014-2999(88)90856-4.
No abstract available

MeSH terms

  • Animals
  • Guinea Pigs
  • Ileum / drug effects
  • Ileum / metabolism
  • In Vitro Techniques
  • Male
  • Muscle, Smooth / drug effects
  • Muscle, Smooth / metabolism
  • Myocardium / metabolism
  • Parasympatholytics / pharmacology*
  • Piperidines / pharmacology*
  • Pirenzepine / pharmacology
  • Rabbits
  • Receptors, Muscarinic / drug effects*
  • Vas Deferens / drug effects

Substances

  • Parasympatholytics
  • Piperidines
  • Receptors, Muscarinic
  • 4-fluorohexahydrosiladifenidol
  • Pirenzepine