Naltrindole, a highly selective and potent non-peptide delta opioid receptor antagonist

Eur J Pharmacol. 1988 Jan 27;146(1):185-6. doi: 10.1016/0014-2999(88)90502-x.
No abstract available

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Guinea Pigs
  • Ileum / drug effects
  • Ileum / metabolism
  • In Vitro Techniques
  • Indoles / metabolism*
  • Indoles / pharmacology
  • Male
  • Mice
  • Morphinans / metabolism*
  • Morphinans / pharmacology
  • Muscle Contraction / drug effects
  • Muscle, Smooth, Vascular / drug effects
  • Muscle, Smooth, Vascular / metabolism*
  • Naltrexone* / analogs & derivatives*
  • Narcotic Antagonists / metabolism*
  • Narcotic Antagonists / pharmacology
  • Rats
  • Receptors, Opioid / metabolism*
  • Receptors, Opioid, delta
  • Vas Deferens / drug effects
  • Vas Deferens / metabolism

Substances

  • Indoles
  • Morphinans
  • Narcotic Antagonists
  • Receptors, Opioid
  • Receptors, Opioid, delta
  • Naltrexone
  • naltrindole