How should values of pA2 and affinity constants for pharmacological competitive antagonists be estimated?
J Pharm Pharmacol
.
1978 May;30(5):312-3.
doi: 10.1111/j.2042-7158.1978.tb13237.x.
Author
D MacKay
PMID:
26747
DOI:
10.1111/j.2042-7158.1978.tb13237.x
No abstract available
MeSH terms
Binding, Competitive
Drug Antagonism*
Mathematics
Models, Biological
Pharmaceutical Preparations / metabolism*
Receptors, Drug / metabolism*
Substances
Pharmaceutical Preparations
Receptors, Drug